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IL155335A0 - Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament - Google Patents

Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament

Info

Publication number
IL155335A0
IL155335A0 IL15533501A IL15533501A IL155335A0 IL 155335 A0 IL155335 A0 IL 155335A0 IL 15533501 A IL15533501 A IL 15533501A IL 15533501 A IL15533501 A IL 15533501A IL 155335 A0 IL155335 A0 IL 155335A0
Authority
IL
Israel
Prior art keywords
medicament
producing
production
same
crystalline monohydrate
Prior art date
Application number
IL15533501A
Other languages
English (en)
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=7659568&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=IL155335(A0) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of IL155335A0 publication Critical patent/IL155335A0/xx

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D451/00Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06Oxygen atoms
    • C07D451/10Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/06Antiasthmatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • A61P11/16Central respiratory analeptics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pulmonology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IL15533501A 2000-10-12 2001-09-28 Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament IL155335A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10050621 2000-10-12
PCT/EP2001/011225 WO2002030928A1 (de) 2000-10-12 2001-09-28 Kristallines monohydrat, verfahren zu dessen herstellung und dessen verwendung zur herstellung eines arzneimittels

Publications (1)

Publication Number Publication Date
IL155335A0 true IL155335A0 (en) 2003-11-23

Family

ID=7659568

Family Applications (2)

Application Number Title Priority Date Filing Date
IL15533501A IL155335A0 (en) 2000-10-12 2001-09-28 Crystalline monohydrate, method for producing the same and the use thereof in the production of a medicament
IL155335A IL155335A (en) 2000-10-12 2003-04-10 Crystalline monohydrate of tiotropium bromide, method for producing the same and the use thereof in the production of a medicament

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL155335A IL155335A (en) 2000-10-12 2003-04-10 Crystalline monohydrate of tiotropium bromide, method for producing the same and the use thereof in the production of a medicament

Country Status (46)

Country Link
EP (2) EP1468998A1 (sk)
JP (1) JP3764422B2 (sk)
KR (1) KR100823860B1 (sk)
CN (2) CN1221549C (sk)
AP (1) AP1572A (sk)
AR (2) AR034389A1 (sk)
AT (1) ATE276253T1 (sk)
AU (2) AU2002214996B2 (sk)
BG (1) BG66161B1 (sk)
BR (1) BR0114584A (sk)
CA (1) CA2425539C (sk)
CR (1) CR6938A (sk)
CZ (1) CZ301841B6 (sk)
DE (1) DE50103666D1 (sk)
DK (1) DK1326862T3 (sk)
DZ (1) DZ3478A1 (sk)
EA (1) EA004381B1 (sk)
EC (1) ECSP034540A (sk)
EE (1) EE04567B1 (sk)
EG (1) EG24142A (sk)
ES (1) ES2228965T3 (sk)
GE (1) GEP20063905B (sk)
HR (1) HRP20030276B1 (sk)
HU (1) HU226830B1 (sk)
IL (2) IL155335A0 (sk)
IS (1) IS2339B (sk)
MA (1) MA25842A1 (sk)
ME (2) ME00243B (sk)
MX (1) MXPA03003221A (sk)
MY (1) MY126931A (sk)
NO (1) NO328465B1 (sk)
NZ (1) NZ525733A (sk)
OA (1) OA12403A (sk)
PE (1) PE20020422A1 (sk)
PL (1) PL207870B1 (sk)
PT (1) PT1326862E (sk)
RS (1) RS50218B (sk)
SA (1) SA01220412B1 (sk)
SI (1) SI1326862T1 (sk)
SK (1) SK287009B6 (sk)
TR (1) TR200402579T4 (sk)
TW (1) TW589313B (sk)
UA (1) UA74215C2 (sk)
UY (2) UY26962A1 (sk)
WO (1) WO2002030928A1 (sk)
ZA (1) ZA200302500B (sk)

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US7244415B2 (en) 2002-03-28 2007-07-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg HFA suspension formulations of an anhydrate
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Also Published As

Publication number Publication date
KR20030042008A (ko) 2003-05-27
SK287009B6 (sk) 2009-09-07
YU27303A (sh) 2006-05-25
AR068527A2 (es) 2009-11-18
NO20031694D0 (no) 2003-04-11
BG107687A (bg) 2003-09-30
TW589313B (en) 2004-06-01
CN100519558C (zh) 2009-07-29
AU2002214996B2 (en) 2007-03-15
IL155335A (en) 2009-02-11
NZ525733A (en) 2005-01-28
PT1326862E (pt) 2004-11-30
WO2002030928A1 (de) 2002-04-18
ATE276253T1 (de) 2004-10-15
BR0114584A (pt) 2003-08-26
KR100823860B1 (ko) 2008-04-21
HUP0301022A2 (hu) 2003-10-28
TR200402579T4 (tr) 2004-12-21
ZA200302500B (en) 2004-04-22
HRP20030276B1 (en) 2006-02-28
DE50103666D1 (de) 2004-10-21
SI1326862T1 (sl) 2005-02-28
AU1499602A (en) 2002-04-22
AR034389A1 (es) 2004-02-25
AP1572A (en) 2006-02-13
RS50218B (sr) 2009-07-15
MA25842A1 (fr) 2003-07-01
EP1326862B1 (de) 2004-09-15
NO20031694L (no) 2003-04-11
PL366041A1 (en) 2005-01-24
CZ301841B6 (cs) 2010-07-07
IS2339B (is) 2008-02-15
HRP20030276A2 (en) 2005-02-28
JP2004526668A (ja) 2004-09-02
CN1733761A (zh) 2006-02-15
JP3764422B2 (ja) 2006-04-05
CA2425539A1 (en) 2003-04-11
CN1469877A (zh) 2004-01-21
HUP0301022A3 (en) 2005-12-28
EA004381B1 (ru) 2004-04-29
ECSP034540A (es) 2003-07-25
EP1326862A1 (de) 2003-07-16
EP1468998A1 (de) 2004-10-20
ES2228965T3 (es) 2005-04-16
HU226830B1 (en) 2009-11-30
UY26962A1 (es) 2002-06-20
CR6938A (es) 2004-10-28
PE20020422A1 (es) 2002-06-28
MXPA03003221A (es) 2004-12-03
MEP40008A (en) 2011-02-10
PL207870B1 (pl) 2011-02-28
HK1086557A1 (zh) 2006-09-22
GEP20063905B (en) 2006-08-25
SA01220412B1 (ar) 2006-11-05
DZ3478A1 (fr) 2002-04-18
MY126931A (en) 2006-10-31
UY34901A (es) 2015-02-27
EG24142A (en) 2008-08-06
IS6772A (is) 2003-04-09
NO328465B1 (no) 2010-02-22
UA74215C2 (uk) 2005-11-15
DK1326862T3 (da) 2004-11-22
ME00243B (me) 2011-05-10
EA200300457A1 (ru) 2003-10-30
CA2425539C (en) 2007-04-03
EE04567B1 (et) 2005-12-15
AP2003002775A0 (en) 2003-03-31
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OA12403A (en) 2006-04-18
CN1221549C (zh) 2005-10-05
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BG66161B1 (bg) 2011-09-30
SK4362003A3 (en) 2003-08-05

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