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NO20084341L - Anvendelse av DPP-IV inhibitorer - Google Patents

Anvendelse av DPP-IV inhibitorer

Info

Publication number
NO20084341L
NO20084341L NO20084341A NO20084341A NO20084341L NO 20084341 L NO20084341 L NO 20084341L NO 20084341 A NO20084341 A NO 20084341A NO 20084341 A NO20084341 A NO 20084341A NO 20084341 L NO20084341 L NO 20084341L
Authority
NO
Norway
Prior art keywords
inhibitors
dpp
risk
disorders
patients
Prior art date
Application number
NO20084341A
Other languages
English (en)
Other versions
NO345061B1 (no
Inventor
Frank Himmelsbach
Klaus Dugi
Michael Mark
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=38235138&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20084341(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of NO20084341L publication Critical patent/NO20084341L/no
Publication of NO345061B1 publication Critical patent/NO345061B1/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine
    • A61K31/522—Purines, e.g. adenine having oxo groups directly attached to the heterocyclic ring, e.g. hypoxanthine, guanine, acyclovir
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/155—Amidines (), e.g. guanidine (H2N—C(=NH)—NH2), isourea (N=C(OH)—NH2), isothiourea (—N=C(SH)—NH2)
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19—Carboxylic acids, e.g. valproic acid
    • A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
    • A61K31/197—Carboxylic acids, e.g. valproic acid having an amino group the amino and the carboxyl groups being attached to the same acyclic carbon chain, e.g. gamma-aminobutyric acid [GABA], beta-alanine, epsilon-aminocaproic acid or pantothenic acid
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4164—1,3-Diazoles
    • A61K31/4184—1,3-Diazoles condensed with carbocyclic rings, e.g. benzimidazoles
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/4985—Pyrazines or piperazines ortho- or peri-condensed with heterocyclic ring systems
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/50—Pyridazines; Hydrogenated pyridazines
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    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
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    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P5/00—Drugs for disorders of the endocrine system
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    • A61P5/50—Drugs for disorders of the endocrine system of the pancreatic hormones for increasing or potentiating the activity of insulin
    • A—HUMAN NECESSITIES
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • A61P9/00—Drugs for disorders of the cardiovascular system
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    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A61K31/52—Purines, e.g. adenine

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  • Health & Medical Sciences (AREA)
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  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Endocrinology (AREA)
  • Obesity (AREA)
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  • Emergency Medicine (AREA)
  • Hospice & Palliative Care (AREA)
  • Immunology (AREA)
  • Molecular Biology (AREA)
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  • Rheumatology (AREA)
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  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Reproductive Health (AREA)
  • Child & Adolescent Psychology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Inorganic Chemistry (AREA)

Abstract

Det beskrives anvendelse av valgte DPP IV-hemmere for behandling av fysiologiske funksjonsforstyrrelser og for reduksjon av risikoen hos risikopasienter til å utvikle slike funksjonsforstyrrelser. I tillegg beskrives anvendelse av ovennevnte DPP IV-hemmere sammen med andre aktive substanser, hvorved forbedrede behandlingsresultater kan oppnås. Disse formene for anvendelse lar seg nyttiggjøre til fremstilling av tilsvarende medikamenter.
NO20084341A 2006-05-04 2008-10-16 Anvendelse av DPP-IV inhibitorer NO345061B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP06009203 2006-05-04
PCT/EP2007/054270 WO2007128761A2 (de) 2006-05-04 2007-05-03 Verwendungen von dpp iv inhibitoren

Publications (2)

Publication Number Publication Date
NO20084341L true NO20084341L (no) 2008-12-02
NO345061B1 NO345061B1 (no) 2020-09-14

Family

ID=38235138

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20084341A NO345061B1 (no) 2006-05-04 2008-10-16 Anvendelse av DPP-IV inhibitorer

Country Status (35)

Country Link
US (9) US8232281B2 (no)
EP (5) EP2397142B1 (no)
JP (12) JP5734564B2 (no)
KR (9) KR20220140016A (no)
CN (8) CN110227078A (no)
AR (1) AR060757A1 (no)
AU (1) AU2007247141B2 (no)
BR (1) BRPI0711308A2 (no)
CA (4) CA2833705C (no)
CL (3) CL2012002527A1 (no)
CY (1) CY1115350T1 (no)
DK (1) DK2015754T3 (no)
EA (3) EA202091999A3 (no)
EC (1) ECSP088866A (no)
ES (2) ES2474866T3 (no)
HK (1) HK1204548A1 (no)
HR (1) HRP20140645T1 (no)
IL (1) IL195031A0 (no)
ME (1) ME01787B (no)
MX (4) MX2008014025A (no)
MY (3) MY174380A (no)
NO (1) NO345061B1 (no)
NZ (2) NZ609765A (no)
PE (2) PE20110235A1 (no)
PH (2) PH12013501790B1 (no)
PL (1) PL2015754T3 (no)
PT (2) PT2015754E (no)
RS (1) RS53272B (no)
SG (1) SG171648A1 (no)
SI (1) SI2015754T1 (no)
TW (2) TWI524894B (no)
UA (1) UA102669C2 (no)
UY (1) UY30321A1 (no)
WO (1) WO2007128761A2 (no)
ZA (1) ZA200808282B (no)

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CN109503584A (zh) 2006-05-04 2019-03-22 勃林格殷格翰国际有限公司 多晶型
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