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SI1747210T1 - ali monosubstituirani fenolin in tiofenolni derivati uporabni kot ligandi H - Google Patents

ali monosubstituirani fenolin in tiofenolni derivati uporabni kot ligandi H

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Publication number
SI1747210T1
SI1747210T1 SI200531085T SI200531085T SI1747210T1 SI 1747210 T1 SI1747210 T1 SI 1747210T1 SI 200531085 T SI200531085 T SI 200531085T SI 200531085 T SI200531085 T SI 200531085T SI 1747210 T1 SI1747210 T1 SI 1747210T1
Authority
SI
Slovenia
Prior art keywords
ligands
derivatives useful
thiophenol derivatives
monosubstituted phenol
monosubstituted
Prior art date
Application number
SI200531085T
Other languages
English (en)
Inventor
P Bernardelli
A M Cronin
A Denis
S M Denton
H Jacobelli
M I Kemp
E Lorthiois
F Rousseau
D Serradeil-Civit
F Vergne
Original Assignee
Warner Lambert Co
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from EP04291187A external-priority patent/EP1593679A1/en
Priority claimed from GB0504564A external-priority patent/GB0504564D0/en
Application filed by Warner Lambert Co filed Critical Warner Lambert Co
Publication of SI1747210T1 publication Critical patent/SI1747210T1/sl

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    • C07D309/04—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
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    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings

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SI200531085T 2004-05-07 2005-04-19 ali monosubstituirani fenolin in tiofenolni derivati uporabni kot ligandi H SI1747210T1 (sl)

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EP04291187A EP1593679A1 (en) 2004-05-07 2004-05-07 3- Or 4-monosubstituted phenol derivatives useful as H3 ligands
GB0504564A GB0504564D0 (en) 2005-03-04 2005-03-04 New compounds
PCT/IB2005/001114 WO2005108384A1 (en) 2004-05-07 2005-04-19 3- or 4-monosubstituted phenol and thiophenol derivatives useful as h3 ligands
EP05718521A EP1747210B1 (en) 2004-05-07 2005-04-19 3- or 4-monosubstituted phenol and thiophenol derivatives useful as h3 ligands

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BRPI0712823A2 (pt) * 2006-06-23 2012-07-24 Abbott Lab derivados de ciclopropil amina como moduladores de receptor de histamina h3
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JP5420534B2 (ja) 2007-05-31 2014-02-19 サノビオン ファーマシューティカルズ インク モノアミン再取り込み阻害薬としてのフェニル置換シクロアルキルアミン
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MX337469B (es) * 2011-10-26 2016-03-02 Pfizer Ltd Derivados de (4-fenilimidazol-2-il)etilamina utiles como moduladores de canal de sodio.
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JP6253668B2 (ja) * 2013-01-09 2017-12-27 アリーナ ファーマシューティカルズ， インコーポレイテッド 認識障害の処置のためのヒスタミンｈ３受容体調節因子としてのビフェニル−エチル−ピロリジン誘導体
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ECSP066975A (es) 2006-12-29
TWI346549B (en) 2011-08-11
HK1100823A1 (en) 2007-09-28
RS51403B (sr) 2011-02-28
IL178433A0 (en) 2007-02-11
EP1747210A1 (en) 2007-01-31
AU2005240846A1 (en) 2005-11-17
UY28883A1 (es) 2005-12-30
TW200607494A (en) 2006-03-01
AP2006003772A0 (en) 2006-10-31
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DE602005022062D1 (de) 2010-08-12
JP2007536365A (ja) 2007-12-13
AR048939A1 (es) 2006-06-14
WO2005108384A1 (en) 2005-11-17
EP1747210B1 (en) 2010-06-30
CR8729A (es) 2006-11-30
HRP20100469T1 (hr) 2010-10-31
CA2565852C (en) 2010-08-10
BRPI0510664A (pt) 2007-12-04
CN1950351A (zh) 2007-04-18
EA200601868A1 (ru) 2007-04-27
GT200500107A (es) 2006-01-10
PA8632201A1 (es) 2006-09-22
KR100843848B1 (ko) 2008-07-03
NL1028968A1 (nl) 2005-11-08
ATE472540T1 (de) 2010-07-15
NZ550769A (en) 2010-06-25
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CY1110735T1 (el) 2015-06-10
BRPI0510664B1 (pt) 2020-04-07
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