EE200200606A - Imidasopürimidiini derivaadid ja triasolopürimidiini derivaadid - Google Patents

Imidasopürimidiini derivaadid ja triasolopürimidiini derivaadid

Info

Publication number: EE200200606A
Authority: EE; Estonia
Prior art keywords: derivatives; imidazopyrimidine; triazolopyrimidine; triazolopyrimidine derivatives; imidazopyrimidine derivatives
Prior art date: 2000-04-28

Application number

EEP200200606A

Other languages

English (en)

Inventor

Yura Takeshi

B. Concepcion Arnel

Han Gyoonhee

Marumo Makiko

Katsumata Hiroko

Kawamura Norihiro

Kokubo Toshio

Komura Hiroshi

Li Yingfu

B. Lowinger Timothy

Mogi Muneto

Yamamoto Noriyuki

Yoshida Nagahiro

Miller Scott

A. Popp Margaret

M. Redmann Aniko

E. Rodriguez Martha

J. Scott William

Wang Ming

Original Assignee

Bayer Aktiengesellschaft

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-28

Filing date

2001-04-17

Publication date

2004-04-15

2001-04-17 Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft

2004-04-15 Publication of EE200200606A publication Critical patent/EE200200606A/et

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Immunology (AREA)
Pulmonology (AREA)
Hematology (AREA)
Dermatology (AREA)
Neurology (AREA)
Diabetes (AREA)
Ophthalmology & Optometry (AREA)
Physical Education & Sports Medicine (AREA)
Orthopedic Medicine & Surgery (AREA)
Biomedical Technology (AREA)
Rheumatology (AREA)
Neurosurgery (AREA)
Pain & Pain Management (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Obesity (AREA)
Child & Adolescent Psychology (AREA)
Transplantation (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

EEP200200606A 2000-04-28 2001-04-17 Imidasopürimidiini derivaadid ja triasolopürimidiini derivaadid EE200200606A (et)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP2000128870A JP2001302667A (ja)	2000-04-28	2000-04-28	イミダゾピリミジン誘導体およびトリアゾロピリミジン誘導体
PCT/EP2001/004357 WO2001083485A1 (en)	2000-04-28	2001-04-17	Imidazopyrimidine derivatives and triazolopyrimidine derivatives

Publications (1)

Publication Number	Publication Date
EE200200606A true EE200200606A (et)	2004-04-15

Family

ID=18638240

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200200606A EE200200606A (et)	2000-04-28	2001-04-17	Imidasopürimidiini derivaadid ja triasolopürimidiini derivaadid

Country Status (37)

Country	Link
US (1)	US6911443B2 (et)
EP (1)	EP1278750B1 (et)
JP (2)	JP2001302667A (et)
KR (1)	KR20030009456A (et)
CN (1)	CN1263756C (et)
AR (1)	AR033367A1 (et)
AT (1)	ATE272639T1 (et)
AU (1)	AU783043B2 (et)
BG (1)	BG107166A (et)
BR (1)	BR0110404A (et)
CA (1)	CA2407531A1 (et)
CZ (1)	CZ20023551A3 (et)
DE (1)	DE60104671T2 (et)
DK (1)	DK1278750T3 (et)
DO (1)	DOP2001000151A (et)
EE (1)	EE200200606A (et)
ES (1)	ES2225546T3 (et)
HR (1)	HRP20020943A2 (et)
HU (1)	HUP0300846A2 (et)
IL (1)	IL151919A0 (et)
MA (1)	MA25746A1 (et)
MX (1)	MXPA02010579A (et)
MY (1)	MY141578A (et)
NO (1)	NO20025154L (et)
NZ (2)	NZ526221A (et)
PE (1)	PE20011287A1 (et)
PL (1)	PL358106A1 (et)
PT (1)	PT1278750E (et)
RU (1)	RU2306313C2 (et)
SI (1)	SI1278750T1 (et)
SK (1)	SK15332002A3 (et)
SV (1)	SV2001000416A (et)
TR (1)	TR200402300T4 (et)
TW (1)	TWI222974B (et)
UA (1)	UA72615C2 (et)
WO (1)	WO2001083485A1 (et)
ZA (1)	ZA200207676B (et)

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2000
- 2000-04-28 JP JP2000128870A patent/JP2001302667A/ja active Pending
2001
- 2001-04-17 EP EP01936242A patent/EP1278750B1/en not_active Expired - Lifetime
- 2001-04-17 US US10/258,628 patent/US6911443B2/en not_active Expired - Fee Related
- 2001-04-17 CN CNB018117201A patent/CN1263756C/zh not_active Expired - Fee Related
- 2001-04-17 NZ NZ526221A patent/NZ526221A/en unknown
- 2001-04-17 WO PCT/EP2001/004357 patent/WO2001083485A1/en not_active Ceased
- 2001-04-17 NZ NZ522241A patent/NZ522241A/en unknown
- 2001-04-17 AT AT01936242T patent/ATE272639T1/de not_active IP Right Cessation
- 2001-04-17 CA CA002407531A patent/CA2407531A1/en not_active Abandoned
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- 2001-04-17 SK SK1533-2002A patent/SK15332002A3/sk unknown
- 2001-04-17 AU AU62204/01A patent/AU783043B2/en not_active Ceased
- 2001-04-17 HU HU0300846A patent/HUP0300846A2/hu unknown
- 2001-04-17 UA UA2002119418A patent/UA72615C2/uk unknown
- 2001-04-17 JP JP2002500795A patent/JP2003535067A/ja active Pending
- 2001-04-17 DE DE60104671T patent/DE60104671T2/de not_active Expired - Fee Related
- 2001-04-17 KR KR1020027014441A patent/KR20030009456A/ko not_active Ceased
- 2001-04-17 EE EEP200200606A patent/EE200200606A/et unknown
- 2001-04-17 ES ES01936242T patent/ES2225546T3/es not_active Expired - Lifetime
- 2001-04-17 MX MXPA02010579A patent/MXPA02010579A/es active IP Right Grant
- 2001-04-17 HR HR20020943A patent/HRP20020943A2/hr not_active Application Discontinuation
- 2001-04-17 PT PT01936242T patent/PT1278750E/pt unknown
- 2001-04-17 DK DK01936242T patent/DK1278750T3/da active
- 2001-04-17 RU RU2002132193/04A patent/RU2306313C2/ru not_active IP Right Cessation
- 2001-04-17 PL PL01358106A patent/PL358106A1/xx not_active Application Discontinuation
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- 2001-04-17 IL IL15191901A patent/IL151919A0/xx unknown
- 2001-04-17 SI SI200130178T patent/SI1278750T1/xx unknown
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2002
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Also Published As

Publication number	Publication date
DOP2001000151A (es)	2002-05-15
JP2001302667A (ja)	2001-10-31
DK1278750T3 (da)	2004-11-22
SK15332002A3 (sk)	2003-06-03
BG107166A (bg)	2003-06-30
ATE272639T1 (de)	2004-08-15
WO2001083485A1 (en)	2001-11-08
TWI222974B (en)	2004-11-01
PE20011287A1 (es)	2002-02-27
NO20025154D0 (no)	2002-10-25
TR200402300T4 (tr)	2004-12-21
EP1278750B1 (en)	2004-08-04
MY141578A (en)	2010-05-14
BR0110404A (pt)	2003-02-11
HRP20020943A2 (en)	2005-02-28
KR20030009456A (ko)	2003-01-29
DE60104671T2 (de)	2005-12-29
EP1278750A1 (en)	2003-01-29
HUP0300846A2 (hu)	2003-08-28
ZA200207676B (en)	2003-09-25
NZ526221A (en)	2005-01-28
HK1058362A1 (en)	2004-05-14
SI1278750T1 (en)	2005-02-28
MXPA02010579A (es)	2003-05-14
RU2306313C2 (ru)	2007-09-20
JP2003535067A (ja)	2003-11-25
DE60104671D1 (de)	2004-09-09
MA25746A1 (fr)	2003-04-01
IL151919A0 (en)	2003-04-10
CN1439009A (zh)	2003-08-27
US20040054179A1 (en)	2004-03-18
CN1263756C (zh)	2006-07-12
ES2225546T3 (es)	2005-03-16
NZ522241A (en)	2004-04-30
NO20025154L (no)	2002-10-25
US6911443B2 (en)	2005-06-28
AU6220401A (en)	2001-11-12
CZ20023551A3 (cs)	2003-01-15
CA2407531A1 (en)	2001-10-25
SV2001000416A (es)	2001-07-03
PL358106A1 (en)	2004-08-09
AR033367A1 (es)	2003-12-17
UA72615C2 (en)	2005-03-15
AU783043B2 (en)	2005-09-22
PT1278750E (pt)	2004-11-30

Publication	Publication Date	Title
EE200200606A (et)	2004-04-15	Imidasopürimidiini derivaadid ja triasolopürimidiini derivaadid
AR028622A1 (es)	2003-05-14	Derivados de tropano utiles en terapia
MA26612A1 (fr)	2004-12-20	Pyrazolopyrimidines et pyrazolotriazines
DE60026297D1 (de)	2006-04-27	Pyrrolotriazin kinasehemmer
EE200200251A (et)	2003-06-16	Uued N-asabitsükloamiidi derivaadid ja nende kasutamine
FI20000819L (fi)	2002-01-25	Menetelmä vastaanottimessa ja vastaanotin
EE200200080A (et)	2003-06-16	Imidaso[1,2a]püridiini ja pürasolo[2,3a]püridiiniderivaadid
ATE321065T1 (de)	2006-04-15	Purin-derivate
ATE238336T1 (de)	2003-05-15	Purin-derivate
EE200100681A (et)	2003-04-15	Puriinderivaadid
DE60020536D1 (de)	2005-07-07	Absorbierender artikel
DE60039814D1 (de)	2008-09-25	Absorbierender Artikel
DE60018133D1 (de)	2005-03-24	Absorbierender Artikel
DE60030038D1 (de)	2006-09-28	Absorbierender Artikel
FI19992753L (fi)	2001-06-22	Menetelmä vastaanottimessa ja vastaanotin
DE60038972D1 (de)	2008-07-03	Absorbierender artikel
DE60044183D1 (de)	2010-05-27	Absorbierender artikel
DE60032898D1 (de)	2007-02-22	Arylthiazolidindion- und aryloxazolidinderivate
DE60103909D1 (de)	2004-07-22	2-pyridinyl-6,7,8,9-tetrahydropyrimido[1,2-a]pyrimidin-4-on- und 7-pyridinyl-2,3-dihydroimidazo[1,2-a]pyrimidin-5 1honderivate
NO20025510L (no)	2003-01-14	Dibenzoazulen-derivater samt anvendelse derav
DE50208341D1 (de)	2006-11-16	Triazolopyrimidine
NO20004072D0 (no)	2000-08-15	Absorberende artikkel
DE60029170D1 (de)	2006-08-17	Absorbierender Artikel
DE60022138D1 (de)	2005-09-29	Absorbierender Artikel
DE60027963D1 (de)	2006-06-22	Absorbierender Artikel

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