DK1278750T3 - Imidazopyrimidinderivater og triazolopyrimidinderivater - Google Patents

Imidazopyrimidinderivater og triazolopyrimidinderivater

Info

Publication number: DK1278750T3
Authority: DK; Denmark
Prior art keywords: derivatives; imidazopyrimidine; triazolopyrimidine; triazolopyrimidine derivatives; imidazopyrimidine derivatives
Prior art date: 2000-04-28

Application number

DK01936242T

Other languages

English (en)

Inventor

Ming Wang

Timothy B Lowinger

Takeshi Yura

Noriyuki Yamamoto

Arnel B Concepcion

Gyoonhee Han

Makiko Hiraoka

Hiroko Katsumata

Norihiro Kawamura

Toshio Kokubo

Hiroshi Komura

Yingfu Li

Muneto Mogi

Nagahiro Yoshida

Original Assignee

Bayer Healthcare Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2000-04-28

Filing date

2001-04-17

Publication date

2004-11-22

2001-04-17 Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag

2004-11-22 Application granted granted Critical

2004-11-22 Publication of DK1278750T3 publication Critical patent/DK1278750T3/da

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
- A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/02—Nasal agents, e.g. decongestants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/04—Antipruritics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/02—Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P21/00—Drugs for disorders of the muscular or neuromuscular system
- A61P21/04—Drugs for disorders of the muscular or neuromuscular system for myasthenia gravis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A61P27/14—Decongestants or antiallergics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/08—Antiallergic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/06—Antianaemics

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Veterinary Medicine (AREA)
Bioinformatics & Cheminformatics (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Engineering & Computer Science (AREA)
Pharmacology & Pharmacy (AREA)
Life Sciences & Earth Sciences (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Immunology (AREA)
Pulmonology (AREA)
Neurology (AREA)
Diabetes (AREA)
Dermatology (AREA)
Hematology (AREA)
Physical Education & Sports Medicine (AREA)
Ophthalmology & Optometry (AREA)
Orthopedic Medicine & Surgery (AREA)
Rheumatology (AREA)
Biomedical Technology (AREA)
Neurosurgery (AREA)
Transplantation (AREA)
Hospice & Palliative Care (AREA)
Psychiatry (AREA)
Pain & Pain Management (AREA)
Obesity (AREA)
Child & Adolescent Psychology (AREA)
Otolaryngology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Plural Heterocyclic Compounds (AREA)

DK01936242T 2000-04-28 2001-04-17 Imidazopyrimidinderivater og triazolopyrimidinderivater DK1278750T3 (da)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
JP2000128870A JP2001302667A (ja)	2000-04-28	2000-04-28	イミダゾピリミジン誘導体およびトリアゾロピリミジン誘導体
PCT/EP2001/004357 WO2001083485A1 (en)	2000-04-28	2001-04-17	Imidazopyrimidine derivatives and triazolopyrimidine derivatives

Publications (1)

Publication Number	Publication Date
DK1278750T3 true DK1278750T3 (da)	2004-11-22

Family

ID=18638240

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
DK01936242T DK1278750T3 (da)	2000-04-28	2001-04-17	Imidazopyrimidinderivater og triazolopyrimidinderivater

Country Status (37)

Country	Link
US (1)	US6911443B2 (da)
EP (1)	EP1278750B1 (da)
JP (2)	JP2001302667A (da)
KR (1)	KR20030009456A (da)
CN (1)	CN1263756C (da)
AR (1)	AR033367A1 (da)
AT (1)	ATE272639T1 (da)
AU (1)	AU783043B2 (da)
BG (1)	BG107166A (da)
BR (1)	BR0110404A (da)
CA (1)	CA2407531A1 (da)
CZ (1)	CZ20023551A3 (da)
DE (1)	DE60104671T2 (da)
DK (1)	DK1278750T3 (da)
DO (1)	DOP2001000151A (da)
EE (1)	EE200200606A (da)
ES (1)	ES2225546T3 (da)
HR (1)	HRP20020943A2 (da)
HU (1)	HUP0300846A2 (da)
IL (1)	IL151919A0 (da)
MA (1)	MA25746A1 (da)
MX (1)	MXPA02010579A (da)
MY (1)	MY141578A (da)
NO (1)	NO20025154L (da)
NZ (2)	NZ526221A (da)
PE (1)	PE20011287A1 (da)
PL (1)	PL358106A1 (da)
PT (1)	PT1278750E (da)
RU (1)	RU2306313C2 (da)
SI (1)	SI1278750T1 (da)
SK (1)	SK15332002A3 (da)
SV (1)	SV2001000416A (da)
TR (1)	TR200402300T4 (da)
TW (1)	TWI222974B (da)
UA (1)	UA72615C2 (da)
WO (1)	WO2001083485A1 (da)
ZA (1)	ZA200207676B (da)

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KR20220098759A (ko)	2019-11-08	2022-07-12	인쎄름 (엥스띠뛰 나씨오날 드 라 쌍떼 에 드 라 흐쉐르슈 메디깔)	키나제 억제제에 대해 내성을 획득한 암의 치료 방법
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2000
- 2000-04-28 JP JP2000128870A patent/JP2001302667A/ja active Pending
2001
- 2001-04-17 EP EP01936242A patent/EP1278750B1/en not_active Expired - Lifetime
- 2001-04-17 US US10/258,628 patent/US6911443B2/en not_active Expired - Fee Related
- 2001-04-17 CN CNB018117201A patent/CN1263756C/zh not_active Expired - Fee Related
- 2001-04-17 NZ NZ526221A patent/NZ526221A/en unknown
- 2001-04-17 WO PCT/EP2001/004357 patent/WO2001083485A1/en not_active Ceased
- 2001-04-17 NZ NZ522241A patent/NZ522241A/en unknown
- 2001-04-17 AT AT01936242T patent/ATE272639T1/de not_active IP Right Cessation
- 2001-04-17 CA CA002407531A patent/CA2407531A1/en not_active Abandoned
- 2001-04-17 CZ CZ20023551A patent/CZ20023551A3/cs unknown
- 2001-04-17 BR BR0110404-7A patent/BR0110404A/pt not_active IP Right Cessation
- 2001-04-17 SK SK1533-2002A patent/SK15332002A3/sk unknown
- 2001-04-17 AU AU62204/01A patent/AU783043B2/en not_active Ceased
- 2001-04-17 HU HU0300846A patent/HUP0300846A2/hu unknown
- 2001-04-17 UA UA2002119418A patent/UA72615C2/uk unknown
- 2001-04-17 JP JP2002500795A patent/JP2003535067A/ja active Pending
- 2001-04-17 DE DE60104671T patent/DE60104671T2/de not_active Expired - Fee Related
- 2001-04-17 KR KR1020027014441A patent/KR20030009456A/ko not_active Ceased
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- 2001-04-17 MX MXPA02010579A patent/MXPA02010579A/es active IP Right Grant
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- 2001-04-17 DK DK01936242T patent/DK1278750T3/da active
- 2001-04-17 RU RU2002132193/04A patent/RU2306313C2/ru not_active IP Right Cessation
- 2001-04-17 PL PL01358106A patent/PL358106A1/xx not_active Application Discontinuation
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- 2001-04-27 TW TW090110055A patent/TWI222974B/zh not_active IP Right Cessation
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2002
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- 2002-10-25 NO NO20025154A patent/NO20025154L/no not_active Application Discontinuation
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Also Published As

Publication number	Publication date
DOP2001000151A (es)	2002-05-15
JP2001302667A (ja)	2001-10-31
SK15332002A3 (sk)	2003-06-03
BG107166A (bg)	2003-06-30
ATE272639T1 (de)	2004-08-15
WO2001083485A1 (en)	2001-11-08
TWI222974B (en)	2004-11-01
PE20011287A1 (es)	2002-02-27
NO20025154D0 (no)	2002-10-25
TR200402300T4 (tr)	2004-12-21
EP1278750B1 (en)	2004-08-04
MY141578A (en)	2010-05-14
BR0110404A (pt)	2003-02-11
HRP20020943A2 (en)	2005-02-28
EE200200606A (et)	2004-04-15
KR20030009456A (ko)	2003-01-29
DE60104671T2 (de)	2005-12-29
EP1278750A1 (en)	2003-01-29
HUP0300846A2 (hu)	2003-08-28
ZA200207676B (en)	2003-09-25
NZ526221A (en)	2005-01-28
HK1058362A1 (en)	2004-05-14
SI1278750T1 (en)	2005-02-28
MXPA02010579A (es)	2003-05-14
RU2306313C2 (ru)	2007-09-20
JP2003535067A (ja)	2003-11-25
DE60104671D1 (de)	2004-09-09
MA25746A1 (fr)	2003-04-01
IL151919A0 (en)	2003-04-10
CN1439009A (zh)	2003-08-27
US20040054179A1 (en)	2004-03-18
CN1263756C (zh)	2006-07-12
ES2225546T3 (es)	2005-03-16
NZ522241A (en)	2004-04-30
NO20025154L (no)	2002-10-25
US6911443B2 (en)	2005-06-28
AU6220401A (en)	2001-11-12
CZ20023551A3 (cs)	2003-01-15
CA2407531A1 (en)	2001-10-25
SV2001000416A (es)	2001-07-03
PL358106A1 (en)	2004-08-09
AR033367A1 (es)	2003-12-17
UA72615C2 (en)	2005-03-15
AU783043B2 (en)	2005-09-22
PT1278750E (pt)	2004-11-30

Publication	Publication Date	Title
DK1278750T3 (da)	2004-11-22	Imidazopyrimidinderivater og triazolopyrimidinderivater
NO991150D0 (no)	1999-03-10	Pyrazolopyrimidiner og pyrazolotriaziner
AR028622A1 (es)	2003-05-14	Derivados de tropano utiles en terapia
IS7283A (is)	2004-05-21	3-ß-D-ríbófúranósýlþíasól[4,5-d]pýridímín kirnisleifar og notkun þeirra
DE60026297D1 (de)	2006-04-27	Pyrrolotriazin kinasehemmer
IS6385A (is)	2002-05-15	Ný notkun og nýjar N-asabísýkló-amíð afleiður
FI20000819L (fi)	2002-01-25	Menetelmä vastaanottimessa ja vastaanotin
EE200200452A (et)	2003-12-15	Puriinderivaadid
NO20041975L (no)	2005-07-16	Bicyklisk oksopyridin og oksopyrimidinderivater
DE60139930D1 (de)	2009-10-29	Desinfizieruns- und desodorierungsverfahren
DE60103537D1 (de)	2004-07-01	Purinderivate
DK1322597T3 (da)	2012-07-02	Fremgangsmåde og intermediære
DE60032898D1 (de)	2007-02-22	Arylthiazolidindion- und aryloxazolidinderivate
ATE512148T1 (de)	2011-06-15	Pyrazolo- und imidazopyrimidinderivate
DE50208341D1 (de)	2006-11-16	Triazolopyrimidine
ATE317386T1 (de)	2006-02-15	Dihydroindol- und tetrahydrochinolinderivate
DE50009171D1 (de)	2005-02-10	Co 2 - kompressor
NO20032821D0 (no)	2003-06-19	Sea-trosy og beslektede fremgangsmåter
DK1204566T3 (da)	2004-09-20	Sammenklappelig varebærer og råemne
DE60118970D1 (de)	2006-05-24	Indol- und dihydroindolderivate
GB2370001B (en)	2005-03-30	Educational aid
NO20031588D0 (no)	2003-04-08	Substituerte 3,4-dihydro-pyrimido(1,2-a)pyrimidiner og 3,4- dihydropyrazino(1,2-a)pyrimidiner
FR2815229B1 (fr)	2003-02-07	Cendrier portable
DE59905993D1 (de)	2003-07-24	Abschaltkupplung
DE50104434D1 (de)	2004-12-09	Lactam-substituierte pyrazolopyridinderivate