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DK2058317T3 - Aminophosphorsyreesterderivat og S1P receptormodulator indeholdende samme som aktiv ingrediens - Google Patents

Aminophosphorsyreesterderivat og S1P receptormodulator indeholdende samme som aktiv ingrediens

Info

Publication number
DK2058317T3
DK2058317T3 DK07792066.8T DK07792066T DK2058317T3 DK 2058317 T3 DK2058317 T3 DK 2058317T3 DK 07792066 T DK07792066 T DK 07792066T DK 2058317 T3 DK2058317 T3 DK 2058317T3
Authority
DK
Denmark
Prior art keywords
active ingredient
acid ester
same
ester derivative
receptor modulator
Prior art date
Application number
DK07792066.8T
Other languages
English (en)
Inventor
Yasushi Kohno
Kiyoshi Fujii
Tatsuhiro Saito
Original Assignee
Kyorin Seiyaku Kk
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Kyorin Seiyaku Kk filed Critical Kyorin Seiyaku Kk
Application granted granted Critical
Publication of DK2058317T3 publication Critical patent/DK2058317T3/da

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/08—Esters of oxyacids of phosphorus
    • C07F9/09—Esters of phosphoric acids
    • C07F9/091—Esters of phosphoric acids with hydroxyalkyl compounds with further substituents on alkyl
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/06—Phosphorus compounds without P—C bonds
    • C07F9/08—Esters of oxyacids of phosphorus
    • C07F9/09—Esters of phosphoric acids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/66—Phosphorus compounds
    • A61K31/661—Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
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    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/14—Vasoprotectives; Antihaemorrhoidals; Drugs for varicose therapy; Capillary stabilisers

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  • Organic Chemistry (AREA)
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  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
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  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Immunology (AREA)
  • Diabetes (AREA)
  • Cardiology (AREA)
  • Pulmonology (AREA)
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  • Heart & Thoracic Surgery (AREA)
  • Molecular Biology (AREA)
  • Neurology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Biochemistry (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Endocrinology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Vascular Medicine (AREA)
  • Rheumatology (AREA)
  • Ophthalmology & Optometry (AREA)
  • Obesity (AREA)
  • Dermatology (AREA)
  • Hospice & Palliative Care (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Otolaryngology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
DK07792066.8T 2006-08-08 2007-08-07 Aminophosphorsyreesterderivat og S1P receptormodulator indeholdende samme som aktiv ingrediens DK2058317T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
JP2006215280 2006-08-08
PCT/JP2007/065397 WO2008018427A1 (en) 2006-08-08 2007-08-07 Aminophosphoric acid ester derivative and s1p receptor modulator containing the same as active ingredient

Publications (1)

Publication Number Publication Date
DK2058317T3 true DK2058317T3 (da) 2014-01-06

Family

ID=39032957

Family Applications (1)

Application Number Title Priority Date Filing Date
DK07792066.8T DK2058317T3 (da) 2006-08-08 2007-08-07 Aminophosphorsyreesterderivat og S1P receptormodulator indeholdende samme som aktiv ingrediens

Country Status (26)

Country Link
US (1) US8232319B2 (da)
EP (1) EP2058317B1 (da)
JP (1) JP5188972B2 (da)
KR (1) KR101339976B1 (da)
CN (1) CN101501049B (da)
CA (1) CA2659598A1 (da)
CY (1) CY1114681T1 (da)
DK (1) DK2058317T3 (da)
ES (1) ES2438265T3 (da)
HR (1) HRP20131172T1 (da)
IL (1) IL196275A (da)
MA (1) MA30663B1 (da)
ME (1) ME02095B (da)
MX (1) MX2009001456A (da)
MY (1) MY152176A (da)
NO (1) NO20090606L (da)
NZ (1) NZ574011A (da)
PL (1) PL2058317T3 (da)
PT (1) PT2058317E (da)
RS (1) RS53080B (da)
RU (1) RU2430925C2 (da)
SG (1) SG174028A1 (da)
SI (1) SI2058317T1 (da)
TN (1) TNSN08545A1 (da)
WO (1) WO2008018427A1 (da)
ZA (1) ZA200900206B (da)

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CN102863345A (zh) * 2011-07-06 2013-01-09 中国医学科学院药物研究所 胺基丙二醇类衍生物、其制备方法和其药物组合物与用途
JPWO2015194157A1 (ja) * 2014-06-16 2017-04-20 杏林製薬株式会社 ジフェニルスルフィド誘導体の製造方法及び製造中間体
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MA42807A (fr) 2015-06-22 2018-07-25 Arena Pharm Inc Sel l-arginine cristallin d'acide (r)-2-(7-(4-cyclopentyl-3-(trifluorométhyl)benzyloxy)-1,2,3,4-tétrahydrocyclo-penta[b]indol-3-yl)acétique (composé 1) pour une utilisation dans des troubles associés au récepteur de s1p1
HUE060485T2 (hu) 2016-06-07 2023-03-28 Tesla Inc Villanymotor hûtési rendszer
WO2018151873A1 (en) 2017-02-16 2018-08-23 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of primary biliary cholangitis
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US10967702B2 (en) 2017-09-07 2021-04-06 Tesla, Inc. Optimal source electric vehicle heat pump with extreme temperature heating capability and efficient thermal preconditioning
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WO2020051378A1 (en) 2018-09-06 2020-03-12 Arena Pharmaceuticals, Inc. Compounds useful in the treatment of autoimmune and inflammatory disorders
MX2021010217A (es) 2019-02-26 2021-09-21 Bayer Ag Derivados heterociclos biciclicos condensados como plaguicida.
JP2023548475A (ja) * 2020-11-09 2023-11-17 アリーナ ファーマシューティカルズ， インコーポレイテッド Ｓ１ｐ１受容体に関係する病態を治療する方法
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PT2058317E (pt) 2013-12-11
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US8232319B2 (en) 2012-07-31
US20090325907A1 (en) 2009-12-31
RU2430925C2 (ru) 2011-10-10
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