TN2010000136A1 - Composition comprising sphingosine 1 phosphate (s1p) receptor modulators - Google Patents

Composition comprising sphingosine 1 phosphate (s1p) receptor modulators

Info

Publication number: TN2010000136A1
Authority: TN; Tunisia
Prior art keywords: sphingosine; phosphate; receptor modulators; composition; amino
Prior art date: 2007-10-12

Application number

TNP2010000136A

Other languages

English (en)

Inventor

Colleen Ruegger

Michael Ambuhl

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2007-10-12

Filing date

2010-03-26

Publication date

2011-09-26

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=40032615&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=TN2010000136(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

2010-03-26 Application filed by Novartis Ag filed Critical Novartis Ag

2011-09-26 Publication of TN2010000136A1 publication Critical patent/TN2010000136A1/fr

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline
- A61K31/137—Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/13—Amines
- A61K31/133—Amines having hydroxy groups, e.g. sphingosine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K36/00—Medicinal preparations of undetermined constitution containing material from algae, lichens, fungi or plants, or derivatives thereof, e.g. traditional herbal medicines
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/10—Alcohols; Phenols; Salts thereof, e.g. glycerol; Polyethylene glycols [PEG]; Poloxamers; PEG/POE alkyl ethers
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
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- A61K47/30—Macromolecular organic or inorganic compounds, e.g. inorganic polyphosphates
- A61K47/36—Polysaccharides; Derivatives thereof, e.g. gums, starch, alginate, dextrin, hyaluronic acid, chitosan, inulin, agar or pectin
- A61K47/38—Cellulose; Derivatives thereof
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/0012—Galenical forms characterised by the site of application
- A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
- A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
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- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
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- A61K9/2004—Excipients; Inactive ingredients
- A61K9/2013—Organic compounds, e.g. phospholipids, fats
- A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
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- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
- Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
- Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Public Health (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Bioinformatics & Cheminformatics (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Immunology (AREA)
Inorganic Chemistry (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Emergency Medicine (AREA)
Physiology (AREA)
Nutrition Science (AREA)
Zoology (AREA)
Heart & Thoracic Surgery (AREA)
Cardiology (AREA)
Botany (AREA)
Mycology (AREA)
Oil, Petroleum & Natural Gas (AREA)
Alternative & Traditional Medicine (AREA)
Biotechnology (AREA)
Natural Medicines & Medicinal Plants (AREA)
Medical Informatics (AREA)
Microbiology (AREA)
Pain & Pain Management (AREA)
Rheumatology (AREA)
Transplantation (AREA)
Hospice & Palliative Care (AREA)
Urology & Nephrology (AREA)

TNP2010000136A 2007-10-12 2010-03-26 Composition comprising sphingosine 1 phosphate (s1p) receptor modulators TN2010000136A1 (en)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US97948207P	2007-10-12	2007-10-12
PCT/US2008/079264 WO2009048993A2 (fr)	2007-10-12	2008-10-09	Compositions comprenant des modulateurs du récepteur de sphingosine 1-phosphate (s1p)

Publications (1)

Publication Number	Publication Date
TN2010000136A1 true TN2010000136A1 (en)	2011-09-26

Family

ID=40032615

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
TNP2010000136A TN2010000136A1 (en)	2007-10-12	2010-03-26	Composition comprising sphingosine 1 phosphate (s1p) receptor modulators

Country Status (32)

Country	Link
US (6)	US8673918B2 (fr)
EP (7)	EP3733161A1 (fr)
JP (2)	JP6034000B2 (fr)
KR (3)	KR101710845B1 (fr)
CN (1)	CN101820916A (fr)
AR (1)	AR068986A1 (fr)
AU (1)	AU2008310846C1 (fr)
BR (1)	BRPI0818161B8 (fr)
CA (2)	CA2925175A1 (fr)
CL (1)	CL2008003003A1 (fr)
CO (1)	CO6270342A2 (fr)
DK (1)	DK2952177T3 (fr)
EC (1)	ECSP10010169A (fr)
ES (2)	ES2545361T3 (fr)
HR (1)	HRP20150838T1 (fr)
HU (2)	HUE027696T2 (fr)
IL (3)	IL204514B (fr)
JO (2)	JOP20080436B1 (fr)
MA (1)	MA31799B1 (fr)
MX (1)	MX337152B (fr)
MY (1)	MY159358A (fr)
NZ (1)	NZ600355A (fr)
PE (2)	PE20090799A1 (fr)
PL (2)	PL2465492T3 (fr)
PT (2)	PT2952177T (fr)
RU (1)	RU2010118457A (fr)
SG (2)	SG187458A1 (fr)
SI (2)	SI2952177T1 (fr)
TN (1)	TN2010000136A1 (fr)
TW (1)	TW200927142A (fr)
WO (1)	WO2009048993A2 (fr)
ZA (1)	ZA201001819B (fr)

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US20160128951A1 (en)	2013-07-29	2016-05-12	Aizant Drug Research Solutions Pvt Ltd	Pharmaceutical compositions of fingolimod
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RS59534B1 (sr)	2014-02-13	2019-12-31	Incyte Corp	Ciklopropilamini kao lsd1 inhibitori
US9527835B2 (en)	2014-02-13	2016-12-27	Incyte Corporation	Cyclopropylamines as LSD1 inhibitors
ES2672797T3 (es)	2014-02-13	2018-06-18	Incyte Corporation	Ciclopropilaminas como inhibidores de LSD1
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CN106163502B (zh) *	2014-04-10	2020-12-01	诺华股份有限公司	免疫抑制剂配方
WO2016007722A1 (fr)	2014-07-10	2016-01-14	Incyte Corporation	Triazolopyridines et triazolopyrazines utilisables comme inhibiteurs de lsd1
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TWI687419B (zh)	2014-07-10	2020-03-11	美商英塞特公司	作為ｌｓｄ１抑制劑之咪唑并吡啶及咪唑并吡嗪
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2008
- 2008-10-09 WO PCT/US2008/079264 patent/WO2009048993A2/fr not_active Ceased
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2014
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Also Published As

Publication number	Publication date
AR068986A1 (es)	2009-12-23
KR101600098B1 (ko)	2016-03-04
CL2008003003A1 (es)	2009-05-15
IL204514B (en)	2018-01-31
JOP20210187A1 (ar)	2023-01-30
US20160296481A1 (en)	2016-10-13
AU2008310846B2 (en)	2012-06-21
US20170151195A1 (en)	2017-06-01
IL255737B (en)	2020-10-29
SI2465492T1 (sl)	2015-12-31
AU2008310846A1 (en)	2009-04-16
US20140142192A1 (en)	2014-05-22
US8673918B2 (en)	2014-03-18
WO2009048993A2 (fr)	2009-04-16
CO6270342A2 (es)	2011-04-20
BRPI0818161B1 (pt)	2020-12-22
HUE053835T2 (hu)	2021-07-28
DK2952177T3 (da)	2021-04-26
US20170368001A1 (en)	2017-12-28
RU2016138157A (ru)	2018-12-13
IL277999A (en)	2020-11-30
EP2952177A1 (fr)	2015-12-09
EP2952177B1 (fr)	2021-01-20
MX2010003925A (es)	2010-05-05
PE20090799A1 (es)	2009-07-20
ES2864671T3 (es)	2021-10-14
JP6034000B2 (ja)	2016-11-30
TW200927142A (en)	2009-07-01
EP2209493A2 (fr)	2010-07-28
EP2465492B1 (fr)	2015-07-01
CA2699788A1 (fr)	2009-04-16
EP3733161A1 (fr)	2020-11-04
CN101820916A (zh)	2010-09-01
EP2653154A1 (fr)	2013-10-23
KR101710845B1 (ko)	2017-02-27
AU2008310846C1 (en)	2022-10-06
SG187458A1 (en)	2013-02-28
PL2952177T3 (pl)	2021-07-19
HK1213768A1 (en)	2016-07-15
US20150165046A1 (en)	2015-06-18
US20100267675A1 (en)	2010-10-21
SG10201800085XA (en)	2018-02-27
ES2545361T3 (es)	2015-09-10
MA31799B1 (fr)	2010-10-01
MY159358A (en)	2016-12-30
PT2465492E (pt)	2015-10-15
WO2009048993A3 (fr)	2010-05-06
ECSP10010169A (es)	2010-06-29
PL2465492T3 (pl)	2015-11-30
BRPI0818161B8 (pt)	2021-05-25
NZ600355A (en)	2013-02-22
CA2699788C (fr)	2016-06-14
JP2015091822A (ja)	2015-05-14
KR20170021904A (ko)	2017-02-28
PT2952177T (pt)	2021-04-26
RU2016138157A3 (fr)	2020-02-10
ZA201001819B (en)	2010-12-29
BRPI0818161A2 (pt)	2017-05-16
HRP20150838T1 (hr)	2015-11-06
EP3120833A1 (fr)	2017-01-25
KR20160025633A (ko)	2016-03-08
EP3733162A1 (fr)	2020-11-04
HUE027696T2 (en)	2016-10-28
IL255737A (en)	2018-01-31
JOP20080436B1 (ar)	2023-03-28
EP2465492A1 (fr)	2012-06-20
MX337152B (es)	2016-02-15
KR20100091179A (ko)	2010-08-18
US9399066B2 (en)	2016-07-26
PE20130309A1 (es)	2013-03-30
CA2925175A1 (fr)	2009-04-16
JP2011500583A (ja)	2011-01-06
RU2010118457A (ru)	2011-11-20
SI2952177T1 (sl)	2021-07-30

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