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SI0719278T1 - Androstenonski derivat - Google Patents

Androstenonski derivat

Info

Publication number
SI0719278T1
SI0719278T1 SI9430130T SI9430130T SI0719278T1 SI 0719278 T1 SI0719278 T1 SI 0719278T1 SI 9430130 T SI9430130 T SI 9430130T SI 9430130 T SI9430130 T SI 9430130T SI 0719278 T1 SI0719278 T1 SI 0719278T1
Authority
SI
Slovenia
Prior art keywords
androstenone
derivative
androstenone derivative
Prior art date
Application number
SI9430130T
Other languages
English (en)
Slovenian (sl)
Inventor
Kenneth W. BATCHELOR
Stephen V. Frye
Original Assignee
Glaxo Wellcome Inc.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=22407744&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI0719278(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Glaxo Wellcome Inc. filed Critical Glaxo Wellcome Inc.
Publication of SI0719278T1 publication Critical patent/SI0719278T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J3/00—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom
    • C07J3/005—Normal steroids containing carbon, hydrogen, halogen or oxygen, substituted in position 17 beta by one carbon atom the carbon atom being part of a carboxylic function
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/26—Androgens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C235/00—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms
    • C07C235/70—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton
    • C07C235/82—Carboxylic acid amides, the carbon skeleton of the acid part being further substituted by oxygen atoms having carbon atoms of carboxamide groups and doubly-bound oxygen atoms bound to the same carbon skeleton with the carbon atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0066—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the 17-beta position being substituted by a carbon atom forming part of an amide group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J73/00—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms
    • C07J73/001—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom
    • C07J73/005—Steroids in which the cyclopenta[a]hydrophenanthrene skeleton has been modified by substitution of one or two carbon atoms by hetero atoms by one hetero atom by nitrogen as hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C2603/00—Systems containing at least three condensed rings
    • C07C2603/02—Ortho- or ortho- and peri-condensed systems
    • C07C2603/04—Ortho- or ortho- and peri-condensed systems containing three rings
    • C07C2603/06—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members
    • C07C2603/10—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings
    • C07C2603/12—Ortho- or ortho- and peri-condensed systems containing three rings containing at least one ring with less than six ring members containing five-membered rings only one five-membered ring
    • C07C2603/14—Benz[f]indenes; Hydrogenated benz[f]indenes

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SI9430130T 1993-09-17 1994-09-16 Androstenonski derivat SI0719278T1 (sl)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US12328093A 1993-09-17 1993-09-17
EP94929828A EP0719278B1 (en) 1993-09-17 1994-09-16 Androstenone derivative
PCT/US1994/010530 WO1995007927A1 (en) 1993-09-17 1994-09-16 Androstenone derivative

Publications (1)

Publication Number Publication Date
SI0719278T1 true SI0719278T1 (sl) 1998-06-30

Family

ID=22407744

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9430130T SI0719278T1 (sl) 1993-09-17 1994-09-16 Androstenonski derivat

Country Status (41)

Country Link
US (2) US5565467A (xx)
EP (1) EP0719278B1 (xx)
JP (1) JP2904310B2 (xx)
KR (1) KR100364953B1 (xx)
CN (1) CN1057771C (xx)
AP (1) AP494A (xx)
AT (1) ATE162199T1 (xx)
AU (1) AU690925B2 (xx)
BG (1) BG62363B1 (xx)
BR (1) BR1100329A (xx)
CA (2) CA2462061A1 (xx)
CY (2) CY2219B1 (xx)
CZ (1) CZ286069B6 (xx)
DE (2) DE69407978T2 (xx)
DK (1) DK0719278T3 (xx)
EE (1) EE03241B1 (xx)
ES (1) ES2113127T3 (xx)
FI (1) FI115216B (xx)
GR (1) GR3026144T3 (xx)
HK (1) HK1004334A1 (xx)
HR (1) HRP940563B1 (xx)
HU (1) HU220060B (xx)
IL (1) IL110978A (xx)
IS (1) IS1713B (xx)
LU (1) LU91027I2 (xx)
MY (1) MY119778A (xx)
NL (1) NL300122I2 (xx)
NO (2) NO306117B1 (xx)
NZ (1) NZ274642A (xx)
OA (1) OA10575A (xx)
PE (1) PE15095A1 (xx)
PL (1) PL180002B1 (xx)
RO (1) RO117455B1 (xx)
RU (1) RU2140926C1 (xx)
SA (1) SA94150231B1 (xx)
SG (1) SG52650A1 (xx)
SI (1) SI0719278T1 (xx)
SK (1) SK281869B6 (xx)
TW (1) TW369521B (xx)
WO (1) WO1995007927A1 (xx)
ZA (2) ZA947118B (xx)

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US5998427A (en) * 1998-05-14 1999-12-07 Glaxo Wellcome Inc. Androstenones
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KR102281252B1 (ko) 2018-05-21 2021-07-23 (주)인벤티지랩 두타스테라이드를 포함하는 마이크로 입자 및 이의 제조 방법
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JP2023527279A (ja) 2020-05-20 2023-06-28 ロデオ・セラピューティクス・コーポレイション 短鎖デヒドロゲナーゼ活性を調節する組成物及び方法
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