DK1667975T3 - En polymorf form for 3-phenylsulfonyl-8-piperazin-1-yl-quinolin - Google Patents
En polymorf form for 3-phenylsulfonyl-8-piperazin-1-yl-quinolinInfo
- Publication number
- DK1667975T3 DK1667975T3 DK04765655T DK04765655T DK1667975T3 DK 1667975 T3 DK1667975 T3 DK 1667975T3 DK 04765655 T DK04765655 T DK 04765655T DK 04765655 T DK04765655 T DK 04765655T DK 1667975 T3 DK1667975 T3 DK 1667975T3
- Authority
- DK
- Denmark
- Prior art keywords
- phenylsulfonyl
- piperazin
- quinoline
- polymorphic form
- polymorphic
- Prior art date
Links
- JJZFWROHYSMCMU-UHFFFAOYSA-N 3-(benzenesulfonyl)-8-piperazin-1-ylquinoline Chemical compound C=1N=C2C(N3CCNCC3)=CC=CC2=CC=1S(=O)(=O)C1=CC=CC=C1 JJZFWROHYSMCMU-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
- C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
- C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D215/38—Nitrogen atoms
- C07D215/40—Nitrogen atoms attached in position 8
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Engineering & Computer Science (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Life Sciences & Earth Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Veterinary Medicine (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Public Health (AREA)
- Pharmacology & Pharmacy (AREA)
- General Health & Medical Sciences (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Psychiatry (AREA)
- Cardiology (AREA)
- Heart & Thoracic Surgery (AREA)
- Child & Adolescent Psychology (AREA)
- Hospice & Palliative Care (AREA)
- Hematology (AREA)
- Obesity (AREA)
- Diabetes (AREA)
- Pain & Pain Management (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Quinoline Compounds (AREA)
- Hydrogenated Pyridines (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GBGB0322629.7A GB0322629D0 (en) | 2003-09-26 | 2003-09-26 | Novel compound |
| PCT/EP2004/010843 WO2005040124A1 (fr) | 2003-09-26 | 2004-09-23 | Nouveau compose |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DK1667975T3 true DK1667975T3 (da) | 2008-04-14 |
Family
ID=29286934
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DK04765655T DK1667975T3 (da) | 2003-09-26 | 2004-09-23 | En polymorf form for 3-phenylsulfonyl-8-piperazin-1-yl-quinolin |
Country Status (23)
| Country | Link |
|---|---|
| US (1) | US20070032504A1 (fr) |
| EP (1) | EP1667975B1 (fr) |
| JP (1) | JP2007506702A (fr) |
| CN (1) | CN1856471A (fr) |
| AU (1) | AU2004283805A1 (fr) |
| BR (1) | BRPI0414678A (fr) |
| CA (1) | CA2540022A1 (fr) |
| CO (1) | CO5680402A2 (fr) |
| DE (1) | DE602004010410T2 (fr) |
| DK (1) | DK1667975T3 (fr) |
| ES (1) | ES2297465T3 (fr) |
| GB (1) | GB0322629D0 (fr) |
| HR (1) | HRP20080055T3 (fr) |
| IL (1) | IL174213A0 (fr) |
| IS (1) | IS8399A (fr) |
| MA (1) | MA28093A1 (fr) |
| MX (1) | MXPA06003375A (fr) |
| NO (1) | NO20061791L (fr) |
| PL (1) | PL1667975T3 (fr) |
| PT (1) | PT1667975E (fr) |
| RU (1) | RU2355681C2 (fr) |
| WO (1) | WO2005040124A1 (fr) |
| ZA (1) | ZA200601453B (fr) |
Families Citing this family (12)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| AR039127A1 (es) * | 2002-03-27 | 2005-02-09 | Glaxo Group Ltd | Compuesto de quinolina, procedimiento para su preparacion, composicion farmaceutica que lo comprende y uso del mismo para la fabricacion de un medicamento |
| MXPA06000795A (es) | 2003-07-22 | 2006-08-23 | Arena Pharm Inc | Derivados de diaril y arilheteroaril urea como moduladores del receptor 5-ht2a de serotonina utiles para la profilaxis y tratamiento de desordenes relacionados con el mismo. |
| PT1663958E (pt) | 2003-09-18 | 2015-06-01 | Virobay Inc | Compostos contendo haloalquilo como inibidores de protease de cisteína |
| BRPI0611516A2 (pt) | 2005-06-02 | 2010-09-14 | Hoffmann La Roche | 3-metanossulfonilquinolinas como realçadores ("enhancers") de gaba-b |
| GB0519758D0 (en) * | 2005-09-28 | 2005-11-09 | Glaxo Group Ltd | Novel process |
| WO2008113818A1 (fr) * | 2007-03-21 | 2008-09-25 | Glaxo Group Limited | Utilisation de composés pour le traitement de la douleur et du syndrome du côlon irritable |
| EP2508177A1 (fr) | 2007-12-12 | 2012-10-10 | Glaxo Group Limited | Associations contenant de la 3-phenylsulfonyl-8-piperazinyl-1yl-quinoline |
| US20110021538A1 (en) | 2008-04-02 | 2011-01-27 | Arena Pharmaceuticals, Inc. | Processes for the preparation of pyrazole derivatives useful as modulators of the 5-ht2a serotonin receptor |
| WO2010062321A1 (fr) | 2008-10-28 | 2010-06-03 | Arena Pharmaceuticals, Inc. | Procédés utiles pour la préparation de 1-[3-(4-bromo-2-méthyl-2h-pyrazol-3-yl)-4-méthoxy-phényl]-3-(2,4-difluoro‑phényl)-urée, et formes cristallines associées |
| MX388281B (es) | 2015-06-12 | 2025-03-11 | Axovant Sciences Gmbh | Derivados de diaril y arilheteroaril urea como moduladores del receptor 5ht2a de serotonina útiles para la profilaxis y el tratamiento de un trastorno conductual del sueño rem. |
| HK1247555A1 (zh) | 2015-07-15 | 2018-09-28 | Axovant Sciences Gmbh | 用於预防和治疗与神经变性疾病相关的幻觉的作为5-ht2a血清素受体的调节剂的二芳基脲和芳基杂芳基脲衍生物 |
| CN108290842B (zh) * | 2016-05-27 | 2021-04-06 | 深圳市塔吉瑞生物医药有限公司 | 一种取代的喹啉化合物及其药物组合物 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9818916D0 (en) * | 1998-08-28 | 1998-10-21 | Smithkline Beecham Plc | Use |
| AR039127A1 (es) * | 2002-03-27 | 2005-02-09 | Glaxo Group Ltd | Compuesto de quinolina, procedimiento para su preparacion, composicion farmaceutica que lo comprende y uso del mismo para la fabricacion de un medicamento |
| GB0321473D0 (en) * | 2003-09-12 | 2003-10-15 | Glaxo Group Ltd | Novel compounds |
-
2003
- 2003-09-26 GB GBGB0322629.7A patent/GB0322629D0/en not_active Ceased
- 2003-09-26 PT PT04765655T patent/PT1667975E/pt unknown
-
2004
- 2004-09-23 EP EP04765655A patent/EP1667975B1/fr not_active Expired - Lifetime
- 2004-09-23 MX MXPA06003375A patent/MXPA06003375A/es active IP Right Grant
- 2004-09-23 DE DE602004010410T patent/DE602004010410T2/de not_active Expired - Fee Related
- 2004-09-23 US US10/572,670 patent/US20070032504A1/en not_active Abandoned
- 2004-09-23 CA CA002540022A patent/CA2540022A1/fr not_active Abandoned
- 2004-09-23 PL PL04765655T patent/PL1667975T3/pl unknown
- 2004-09-23 WO PCT/EP2004/010843 patent/WO2005040124A1/fr not_active Ceased
- 2004-09-23 JP JP2006527373A patent/JP2007506702A/ja not_active Withdrawn
- 2004-09-23 CN CNA2004800275278A patent/CN1856471A/zh active Pending
- 2004-09-23 AU AU2004283805A patent/AU2004283805A1/en not_active Abandoned
- 2004-09-23 DK DK04765655T patent/DK1667975T3/da active
- 2004-09-23 ES ES04765655T patent/ES2297465T3/es not_active Expired - Lifetime
- 2004-09-23 RU RU2006114024/04A patent/RU2355681C2/ru active
- 2004-09-23 HR HR20080055T patent/HRP20080055T3/xx unknown
- 2004-09-23 BR BRPI0414678-6A patent/BRPI0414678A/pt not_active IP Right Cessation
-
2006
- 2006-02-20 ZA ZA200601453A patent/ZA200601453B/en unknown
- 2006-03-09 IL IL174213A patent/IL174213A0/en unknown
- 2006-03-27 CO CO06030123A patent/CO5680402A2/es not_active Application Discontinuation
- 2006-04-05 IS IS8399A patent/IS8399A/is unknown
- 2006-04-13 MA MA28933A patent/MA28093A1/fr unknown
- 2006-04-24 NO NO20061791A patent/NO20061791L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| CA2540022A1 (fr) | 2005-05-06 |
| MA28093A1 (fr) | 2006-08-01 |
| HRP20080055T3 (en) | 2008-02-29 |
| IL174213A0 (en) | 2006-08-01 |
| BRPI0414678A (pt) | 2006-11-28 |
| CO5680402A2 (es) | 2006-09-29 |
| DE602004010410D1 (en) | 2008-01-10 |
| EP1667975A1 (fr) | 2006-06-14 |
| DE602004010410T2 (de) | 2008-10-16 |
| RU2355681C2 (ru) | 2009-05-20 |
| CN1856471A (zh) | 2006-11-01 |
| NO20061791L (no) | 2006-04-24 |
| MXPA06003375A (es) | 2006-06-08 |
| PT1667975E (pt) | 2008-02-29 |
| HK1094190A1 (en) | 2007-03-23 |
| WO2005040124A1 (fr) | 2005-05-06 |
| ZA200601453B (en) | 2007-04-25 |
| GB0322629D0 (en) | 2003-10-29 |
| ES2297465T3 (es) | 2008-05-01 |
| US20070032504A1 (en) | 2007-02-08 |
| RU2006114024A (ru) | 2007-11-10 |
| EP1667975B1 (fr) | 2007-11-28 |
| IS8399A (is) | 2006-04-05 |
| AU2004283805A1 (en) | 2005-05-06 |
| PL1667975T3 (pl) | 2008-04-30 |
| JP2007506702A (ja) | 2007-03-22 |
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