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CY1117279T1 - Διμηλεϊνκο αλας μιας αμινοκροτονυλικης ενωσης και μεθοδος για την παραγωγη τους - Google Patents

Διμηλεϊνκο αλας μιας αμινοκροτονυλικης ενωσης και μεθοδος για την παραγωγη τους

Info

Publication number
CY1117279T1
CY1117279T1 CY20161100212T CY161100212T CY1117279T1 CY 1117279 T1 CY1117279 T1 CY 1117279T1 CY 20161100212 T CY20161100212 T CY 20161100212T CY 161100212 T CY161100212 T CY 161100212T CY 1117279 T1 CY1117279 T1 CY 1117279T1
Authority
CY
Cyprus
Prior art keywords
production
aminocrotonylic
salon
silence
union
Prior art date
Application number
CY20161100212T
Other languages
English (en)
Inventor
Werner Rall
Christian Kulinna
Juergen Schnaubelt
Peter Sieger
Rainer Soyka
Original Assignee
Boehringer Ingelheim International Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=34428508&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CY1117279(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Boehringer Ingelheim International Gmbh filed Critical Boehringer Ingelheim International Gmbh
Publication of CY1117279T1 publication Critical patent/CY1117279T1/el

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D405/00—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom
    • C07D405/02—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings
    • C07D405/12—Heterocyclic compounds containing both one or more hetero rings having oxygen atoms as the only ring hetero atoms, and one or more rings having nitrogen as the only ring hetero atom containing two hetero rings linked by a chain containing hetero atoms as chain links
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16—Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Pulmonology (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Urology & Nephrology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pyrrole Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)

Abstract

Η εφεύρεση αφορά μια βελτιωμένη μέθοδο για την παραγωγή της 4-[(3-χλωρο-4-φθοροφαινυλ)αμινο]-6-{[4-(Ν,Ν-διμεθυλαμινο)-1-οξο-2-βουτεν-1-υλ]αμινο}-7-((S)-τετραϋδροφουραν-3-υλ-οξυ)-κιναζολίνης και συγγενών αμινοκροτονυλικών ενώσεων και την παραγωγή ενός κατάλληλου άλατος της 4-[(3-χλωρο-4-φθοροφαινυλ)αμινο]-6-{[4-(Ν,Ν-διμεθυλαμινο)-1-οξο-2-βουτεν-1-υλ]αμινο}-7-((S)-τετραϋδροφουραν-3-υλ-οξυ)-κιναζολίνης για χρήση ως δραστικής ουσίας για φάρμακα.
CY20161100212T 2003-10-17 2016-03-11 Διμηλεϊνκο αλας μιας αμινοκροτονυλικης ενωσης και μεθοδος για την παραγωγη τους CY1117279T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10349113A DE10349113A1 (de) 2003-10-17 2003-10-17 Verfahren zur Herstellung von Aminocrotonylverbindungen
EP12155662.5A EP2508521B2 (de) 2003-10-17 2004-10-12 Dimaleat einer Aminocrotonylverbindung und Verfahren zu ihrer Herstellung

Publications (1)

Publication Number Publication Date
CY1117279T1 true CY1117279T1 (el) 2017-04-26

Family

ID=34428508

Family Applications (2)

Application Number Title Priority Date Filing Date
CY20131101112T CY1114866T1 (el) 2003-10-17 2013-12-09 Μεθοδος για την παραγωγη αμινοκροτονυλικων ενωσεων
CY20161100212T CY1117279T1 (el) 2003-10-17 2016-03-11 Διμηλεϊνκο αλας μιας αμινοκροτονυλικης ενωσης και μεθοδος για την παραγωγη τους

Family Applications Before (1)

Application Number Title Priority Date Filing Date
CY20131101112T CY1114866T1 (el) 2003-10-17 2013-12-09 Μεθοδος για την παραγωγη αμινοκροτονυλικων ενωσεων

Country Status (34)

Country Link
US (2) US20050085495A1 (el)
EP (2) EP1678165B1 (el)
JP (2) JP4594317B2 (el)
KR (2) KR101180752B1 (el)
CN (2) CN101402631A (el)
AR (1) AR046118A1 (el)
AU (2) AU2004281938B2 (el)
BR (2) BR122013033343B8 (el)
CA (2) CA2759063C (el)
CY (2) CY1114866T1 (el)
DE (1) DE10349113A1 (el)
DK (2) DK2508521T4 (el)
EA (1) EA016624B1 (el)
EC (1) ECSP066509A (el)
ES (2) ES2440466T3 (el)
HR (2) HRP20160246T4 (el)
HU (1) HUE028254T2 (el)
IL (2) IL174951A (el)
ME (1) ME00341B (el)
MX (2) MXPA06004076A (el)
MY (2) MY149921A (el)
NO (2) NO333971B1 (el)
NZ (2) NZ583049A (el)
PE (2) PE20100267A1 (el)
PL (2) PL2508521T5 (el)
PT (2) PT2508521E (el)
RS (3) RS53398B (el)
SG (1) SG139743A1 (el)
SI (2) SI1678165T1 (el)
TW (2) TWI348468B (el)
UA (2) UA91006C2 (el)
UY (2) UY28559A1 (el)
WO (1) WO2005037824A2 (el)
ZA (1) ZA200602234B (el)

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