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NO20045521L - Diarylureaderivater anvendelige for behandling av proteinkinaseavhengige sykdommer - Google Patents

Diarylureaderivater anvendelige for behandling av proteinkinaseavhengige sykdommer

Info

Publication number
NO20045521L
NO20045521L NO20045521A NO20045521A NO20045521L NO 20045521 L NO20045521 L NO 20045521L NO 20045521 A NO20045521 A NO 20045521A NO 20045521 A NO20045521 A NO 20045521A NO 20045521 L NO20045521 L NO 20045521L
Authority
NO
Norway
Prior art keywords
treatment
diarylurea derivatives
diarylurea
derivatives
protein kinase
Prior art date
Application number
NO20045521A
Other languages
English (en)
Inventor
Guido Bold
Pascal Furet
Paul William Manley
Andreas Floersheimer
Eugen Boss
Vito Guagnano
Andrea Vaupel
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0212413A external-priority patent/GB0212413D0/en
Priority claimed from GB0305684A external-priority patent/GB0305684D0/en
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of NO20045521L publication Critical patent/NO20045521L/no

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D213/36—Radicals substituted by singly-bound nitrogen atoms
    • C07D213/40—Acylated substituent nitrogen atom
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/24—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom with substituted hydrocarbon radicals attached to ring carbon atoms
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Abstract

Foreliggende oppfinnelse angår anvendelsen av diarylureaderivater ved behandling av proteinkinaseavhengige sykdommer eller for fremstilling av farmasøytiske sammensetninger for anvendelse ved behandling av nevnte sykdommer, fremgangsmåte for anvendelse av de arylureaderivater ved behandling av nevnte sykdommer, farmasøytiske preparater som innbefatter diarylureaderivater for behandling av nevnte sykdommer, diarylureaderivater for anvendelse ved behandling av nevnte sykdommer, nye diarylureaderivater, farmasøytiske preparater som innbefatter disse nye diarylureaderivatene, fremgangsmåte for fremstilling av de nye diarylureaderivatene, anvendelsen eller fremgangsmåtene for anvendelse av de nye diarylureaderivatene som nevnt ovenfor, og/eller disse nye diarylureaderivatene for anvendelse ved behandling av en dyre- eller menneskekropp.
NO20045521A 2002-05-29 2004-12-17 Diarylureaderivater anvendelige for behandling av proteinkinaseavhengige sykdommer NO20045521L (no)

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GB0212413A GB0212413D0 (en) 2002-05-29 2002-05-29 Organic Compounds
GB0305684A GB0305684D0 (en) 2003-03-12 2003-03-12 Organic compounds
GB0309219 2003-04-23
PCT/EP2003/005634 WO2003099771A2 (en) 2002-05-29 2003-05-28 Diaryl urea derivatives useful for the treatment of protein kinase dependent diseases

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CA2484288A1 (en) 2003-12-04
JP2005527622A (ja) 2005-09-15
EP1511730B8 (en) 2009-04-08
MXPA04011789A (es) 2005-03-31
ES2318158T3 (es) 2009-05-01
CN1656073A (zh) 2005-08-17
EP1511730B1 (en) 2008-12-10
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EP1511730A2 (en) 2005-03-09
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US7652022B2 (en) 2010-01-26
CN1656073B (zh) 2010-05-26
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BR0311313A (pt) 2005-02-15
PL372426A1 (en) 2005-07-25
ATE417037T1 (de) 2008-12-15
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US20060128734A1 (en) 2006-06-15
DE60325209D1 (de) 2009-01-22
KR20050006281A (ko) 2005-01-15
KR101036394B1 (ko) 2011-05-23
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