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DK3030227T3 - Vedvarende frigivelses-doseringsformer for en jak1-inhibitor - Google Patents

Vedvarende frigivelses-doseringsformer for en jak1-inhibitor Download PDF

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Publication number
DK3030227T3
DK3030227T3 DK14753182.6T DK14753182T DK3030227T3 DK 3030227 T3 DK3030227 T3 DK 3030227T3 DK 14753182 T DK14753182 T DK 14753182T DK 3030227 T3 DK3030227 T3 DK 3030227T3
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Prior art keywords
dosage forms
release dosage
jak1 inhibitor
releasing release
releasing
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DK14753182.6T
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English (en)
Inventor
Krishnaswamy Yeleswaram
Bhavnish Parikh
Dilip P Modi
Trupti Sheth
Original Assignee
Incyte Corp
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Publication of DK3030227T3 publication Critical patent/DK3030227T3/da

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    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2009—Inorganic compounds
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
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    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates
    • A—HUMAN NECESSITIES
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    • A61K9/20—Pills, tablets, discs, rods
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    • A61K9/2022—Organic macromolecular compounds
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    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
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  • Health & Medical Sciences (AREA)
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  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
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  • Epidemiology (AREA)
  • Diabetes (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Immunology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Rheumatology (AREA)
  • Dermatology (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Biophysics (AREA)
  • Molecular Biology (AREA)
  • Biomedical Technology (AREA)
  • Endocrinology (AREA)
  • Neurosurgery (AREA)
  • Inorganic Chemistry (AREA)
  • Transplantation (AREA)
  • Cardiology (AREA)
  • Oncology (AREA)
  • Emergency Medicine (AREA)
  • Obesity (AREA)
  • Pulmonology (AREA)
  • Urology & Nephrology (AREA)
  • Pain & Pain Management (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hospice & Palliative Care (AREA)
DK14753182.6T 2013-08-07 2014-08-06 Vedvarende frigivelses-doseringsformer for en jak1-inhibitor DK3030227T3 (da)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US201361863325P 2013-08-07 2013-08-07
US201361913066P 2013-12-06 2013-12-06
PCT/US2014/049940 WO2015021153A1 (en) 2013-08-07 2014-08-06 Sustained release dosage forms for a jak1 inhibitor

Publications (1)

Publication Number Publication Date
DK3030227T3 true DK3030227T3 (da) 2020-04-20

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ID=51383933

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Application Number Title Priority Date Filing Date
DK14753182.6T DK3030227T3 (da) 2013-08-07 2014-08-06 Vedvarende frigivelses-doseringsformer for en jak1-inhibitor

Country Status (31)

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US (5) US9655854B2 (da)
EP (2) EP3030227B1 (da)
JP (6) JP6334700B2 (da)
KR (3) KR102419714B1 (da)
CN (3) CN105579032A (da)
AU (3) AU2014305989B2 (da)
BR (1) BR122020001831A8 (da)
CA (2) CA2920108C (da)
CL (1) CL2016000292A1 (da)
CR (3) CR20190343A (da)
CY (1) CY1123314T1 (da)
DK (1) DK3030227T3 (da)
EA (1) EA201690357A1 (da)
ES (1) ES2792549T3 (da)
HR (1) HRP20200955T1 (da)
HU (1) HUE049345T2 (da)
IL (2) IL277554B2 (da)
LT (1) LT3030227T (da)
MX (2) MX376856B (da)
MY (2) MY203694A (da)
PE (2) PE20160223A1 (da)
PH (3) PH12019502074B1 (da)
PL (1) PL3030227T3 (da)
PT (1) PT3030227T (da)
RS (1) RS60469B1 (da)
SG (3) SG11201600815WA (da)
SI (1) SI3030227T1 (da)
SM (1) SMT202000315T1 (da)
TW (3) TWI789516B (da)
UA (1) UA120499C2 (da)
WO (1) WO2015021153A1 (da)

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HUE049345T2 (hu) 2020-09-28
AU2019257368B2 (en) 2021-02-25
CA2920108C (en) 2022-07-05
CR20230316A (es) 2023-11-10
PL3030227T3 (pl) 2020-08-24
TW201529099A (zh) 2015-08-01
JP2022136270A (ja) 2022-09-15
JP6880266B2 (ja) 2021-06-02
TWI789516B (zh) 2023-01-11
TWI730935B (zh) 2021-06-21
CN114010611B (zh) 2023-11-28
SI3030227T1 (sl) 2020-08-31
ES2792549T3 (es) 2020-11-11
EP3721873A1 (en) 2020-10-14
KR102419714B1 (ko) 2022-07-13
US20170319487A1 (en) 2017-11-09
LT3030227T (lt) 2020-06-10
AU2019257368A1 (en) 2019-11-14
KR20220103810A (ko) 2022-07-22
MY195091A (en) 2023-01-10
CA2920108A1 (en) 2015-02-12
PH12016500243A1 (en) 2016-05-16
JP2021107454A (ja) 2021-07-29
CL2016000292A1 (es) 2016-08-05
JP2020079317A (ja) 2020-05-28
EP3030227A1 (en) 2016-06-15
MX2016001639A (es) 2016-10-07
US9655854B2 (en) 2017-05-23
JP2016527315A (ja) 2016-09-08
BR122020001831A2 (da) 2017-08-01
US20150065484A1 (en) 2015-03-05
RS60469B1 (sr) 2020-07-31
IL243920A0 (en) 2016-04-21
US12151026B2 (en) 2024-11-26
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EA201690357A1 (ru) 2016-07-29
JP6334700B2 (ja) 2018-05-30

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