NO20035486D0 - Benzodiazepinderivater og deres anvendelse som AMPA- reseptorstimulatorer - Google Patents

Benzodiazepinderivater og deres anvendelse som AMPA- reseptorstimulatorer

Info

Publication number: NO20035486D0
Authority: NO; Norway
Prior art keywords: ampa receptor; benzodiazepine derivatives; receptor stimulators; stimulators; benzodiazepine
Prior art date: 2001-06-11

Application number

NO20035486A

Other languages

English (en)

Other versions

NO328705B1 (no

Inventor

Simon James Anthony Grove

Mingqiang Zhang

Mohammad Shahid

Original Assignee

Akzo Nobel Nv

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2001-06-11

Filing date

2003-12-10

Publication date

2003-12-10

2003-12-10 Application filed by Akzo Nobel Nv filed Critical Akzo Nobel Nv

2003-12-10 Publication of NO20035486D0 publication Critical patent/NO20035486D0/no

2010-05-03 Publication of NO328705B1 publication Critical patent/NO328705B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D515/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
- C07D515/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen, oxygen, and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
- C07D515/04—Ortho-condensed systems
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D498/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D498/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
- C07D498/04—Ortho-condensed systems
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/10—Drugs for genital or sexual disorders; Contraceptives for impotence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/08—Antiepileptics; Anticonvulsants
- A61P25/12—Antiepileptics; Anticonvulsants for grand-mal
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/22—Anxiolytics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/24—Antidepressants
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/32—Alcohol-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence
- A61P25/36—Opioid-abuse
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

Health & Medical Sciences (AREA)
Organic Chemistry (AREA)
Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Pharmacology & Pharmacy (AREA)
Chemical Kinetics & Catalysis (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Neurosurgery (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Psychiatry (AREA)
Addiction (AREA)
Pain & Pain Management (AREA)
Heart & Thoracic Surgery (AREA)
Hospice & Palliative Care (AREA)
Cardiology (AREA)
Gynecology & Obstetrics (AREA)
Endocrinology (AREA)
Reproductive Health (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Plural Heterocyclic Compounds (AREA)

NO20035486A 2001-06-11 2003-12-10 Benzodiazepinderivater og deres anvendelse som AMPA-reseptorstimulatorer NO328705B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP01202215		2001-06-11
PCT/EP2002/006185 WO2002100865A1 (en)	2001-06-11	2002-06-05	Benzoxazepine derivatives and their use as ampa receptor stimulators

Publications (2)

Publication Number	Publication Date
NO20035486D0 true NO20035486D0 (no)	2003-12-10
NO328705B1 NO328705B1 (no)	2010-05-03

Family

ID=8180450

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20035486A NO328705B1 (no)	2001-06-11	2003-12-10	Benzodiazepinderivater og deres anvendelse som AMPA-reseptorstimulatorer

Country Status (29)

Country	Link
US (2)	US7307073B2 (no)
EP (1)	EP1399450B1 (no)
JP (1)	JP4435561B2 (no)
KR (1)	KR100863255B1 (no)
CN (1)	CN1257908C (no)
AR (1)	AR036092A1 (no)
AT (1)	ATE389659T1 (no)
AU (1)	AU2002314144B2 (no)
BR (1)	BR0210222A (no)
CA (1)	CA2450274C (no)
CO (1)	CO5550447A2 (no)
CZ (1)	CZ300052B6 (no)
DE (1)	DE60225689T2 (no)
EC (1)	ECSP034891A (no)
ES (1)	ES2301651T3 (no)
HR (1)	HRP20031007A2 (no)
HU (1)	HUP0400154A3 (no)
IL (2)	IL158905A0 (no)
IS (1)	IS2526B (no)
MX (1)	MXPA03011563A (no)
NO (1)	NO328705B1 (no)
NZ (1)	NZ529670A (no)
PE (1)	PE20030097A1 (no)
PL (1)	PL366721A1 (no)
RU (1)	RU2279434C2 (no)
SK (1)	SK287150B6 (no)
TW (1)	TWI232863B (no)
WO (1)	WO2002100865A1 (no)
ZA (1)	ZA200309382B (no)

Families Citing this family (10)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PL367185A1 (en)	2001-06-14	2005-02-21	Akzo Nobel, N.V.	(pyrido/thieno)-[f]-oxazepin-5-one derivatives
WO2010054336A2 (en) *	2008-11-10	2010-05-14	The Regents Of The University Of California	Therapeutic uses of ampa receptor modulators for treatment of motor dysfunction
WO2011036280A1 (en) *	2009-09-28	2011-03-31	F. Hoffmann-La Roche Ag	Benzoxazepin pi3k inhibitor compounds and methods of use
FR2964969B1 (fr)	2010-09-16	2012-08-24	Servier Lab	Nouveaux derives dihydrobenzoxathiazepines, leur procede de preparation et les compositions pharmaceutiques qui les contiennent
JP2016521755A (ja)	2013-06-13	2016-07-25	ヴェロサイエンス，リミテッド・ライアビリティー・カンパニー	代謝障害を治療するための組成物および方法
CN110114071B (zh)	2016-11-07	2023-07-04	爱彼特生物制药公司	含有取代的吡啶酮的三环化合物以及使用其的方法
US11702427B2 (en)	2018-03-12	2023-07-18	Arbutus Biopharma Corporation	Substituted 2-pyridone tricyclic compounds, analogues thereof, and methods using same
AU2019252441A1 (en)	2018-04-12	2020-10-22	Arbutus Biopharma Corporation	Methods for preparing substituted pyridinone-containing tricyclic compounds
JP7138246B2 (ja)	2018-11-22	2022-09-15	福建▲広▼生中霖生物科技有限公司	Ｂ型肝炎表面抗原阻害剤の結晶形
US20230218632A1 (en) *	2020-03-20	2023-07-13	Amathus Therapeutics, Inc.	Cyclic sulfonamide derivatives as trap1 modulators and uses thereof

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB1238719A (no)	1968-11-01	1971-07-07
PT651746E (pt)	1992-07-24	2002-09-30	Univ California	Drogas que intensificam as respostas sinapticas mediadas por receptores de ampa
DK0801651T3 (da) *	1995-01-06	2001-10-22	Hoffmann La Roche	Hydroxymethyl-imidazodiazepiner og deres estere
US5650409A (en) *	1995-06-02	1997-07-22	Cortex Pharmaceuticals, Inc.	Benzoyl piperidines/pyrrolidines for enhancing synaptic response
US5736543A (en) *	1996-04-03	1998-04-07	The Regents Of The University Of California	Benzoxazines for enhancing synaptic response
ATE303997T1 (de)	1997-06-09	2005-09-15	Pfizer Prod Inc	Chinazolin-4-on ampa antagonisten
US5985871A (en) *	1997-12-24	1999-11-16	Cortex Pharmaceuticals, Inc.	Benzoxazine compounds for enhancing synaptic response
ZA991301B (en) *	1998-02-18	1999-09-13	Neurosearch As	Glutamate receptor modulators.
US6124278A (en)	1998-04-03	2000-09-26	The Regents Of The University Of California	Acylbenzoxazines for enhancing synaptic response

2002
- 2002-05-31 TW TW091111746A patent/TWI232863B/zh not_active IP Right Cessation
- 2002-06-05 CA CA2450274A patent/CA2450274C/en not_active Expired - Lifetime
- 2002-06-05 RU RU2004100310/04A patent/RU2279434C2/ru not_active IP Right Cessation
- 2002-06-05 KR KR1020037016150A patent/KR100863255B1/ko not_active Expired - Fee Related
- 2002-06-05 MX MXPA03011563A patent/MXPA03011563A/es active IP Right Grant
- 2002-06-05 CN CNB028116410A patent/CN1257908C/zh not_active Expired - Lifetime
- 2002-06-05 SK SK1518-2003A patent/SK287150B6/sk not_active IP Right Cessation
- 2002-06-05 WO PCT/EP2002/006185 patent/WO2002100865A1/en not_active Ceased
- 2002-06-05 PL PL02366721A patent/PL366721A1/xx not_active IP Right Cessation
- 2002-06-05 AT AT02740691T patent/ATE389659T1/de active
- 2002-06-05 HU HU0400154A patent/HUP0400154A3/hu unknown
- 2002-06-05 CZ CZ20033376A patent/CZ300052B6/cs not_active IP Right Cessation
- 2002-06-05 IL IL15890502A patent/IL158905A0/xx unknown
- 2002-06-05 BR BR0210222-6A patent/BR0210222A/pt not_active Application Discontinuation
- 2002-06-05 EP EP02740691A patent/EP1399450B1/en not_active Expired - Lifetime
- 2002-06-05 ES ES02740691T patent/ES2301651T3/es not_active Expired - Lifetime
- 2002-06-05 NZ NZ529670A patent/NZ529670A/en unknown
- 2002-06-05 JP JP2003503632A patent/JP4435561B2/ja not_active Expired - Lifetime
- 2002-06-05 DE DE60225689T patent/DE60225689T2/de not_active Expired - Lifetime
- 2002-06-05 US US10/480,623 patent/US7307073B2/en not_active Expired - Lifetime
- 2002-06-05 HR HR20031007A patent/HRP20031007A2/xx not_active Application Discontinuation
- 2002-06-05 AU AU2002314144A patent/AU2002314144B2/en not_active Expired
- 2002-06-10 PE PE2002000495A patent/PE20030097A1/es not_active Application Discontinuation
- 2002-06-10 AR ARP020102171A patent/AR036092A1/es unknown
2003
- 2003-11-13 IS IS7036A patent/IS2526B/is unknown
- 2003-11-17 IL IL158905A patent/IL158905A/en not_active IP Right Cessation
- 2003-12-02 ZA ZA200309382A patent/ZA200309382B/en unknown
- 2003-12-04 CO CO03107046A patent/CO5550447A2/es not_active Application Discontinuation
- 2003-12-10 NO NO20035486A patent/NO328705B1/no not_active IP Right Cessation
- 2003-12-11 EC EC2003004891A patent/ECSP034891A/es unknown
2007
- 2007-10-25 US US11/924,451 patent/US7504390B2/en not_active Expired - Lifetime

Also Published As

Publication number	Publication date
CO5550447A2 (es)	2005-08-31
HRP20031007A2 (en)	2005-10-31
ECSP034891A (es)	2004-01-28
ES2301651T3 (es)	2008-07-01
SK287150B6 (sk)	2010-01-07
SK15182003A3 (sk)	2004-05-04
BR0210222A (pt)	2004-04-13
RU2004100310A (ru)	2005-06-10
JP4435561B2 (ja)	2010-03-17
HK1061858A1 (en)	2004-10-08
CZ300052B6 (cs)	2009-01-21
EP1399450B1 (en)	2008-03-19
AR036092A1 (es)	2004-08-11
WO2002100865A1 (en)	2002-12-19
NZ529670A (en)	2006-02-24
PL366721A1 (en)	2005-02-07
DE60225689T2 (de)	2008-07-17
KR100863255B1 (ko)	2008-10-15
US7307073B2 (en)	2007-12-11
NO328705B1 (no)	2010-05-03
DE60225689D1 (de)	2008-04-30
RU2279434C2 (ru)	2006-07-10
HUP0400154A3 (en)	2007-05-02
IL158905A0 (en)	2004-05-12
JP2004533466A (ja)	2004-11-04
CZ20033376A3 (en)	2004-04-14
US20080139529A1 (en)	2008-06-12
US20040171605A1 (en)	2004-09-02
EP1399450A1 (en)	2004-03-24
CN1257908C (zh)	2006-05-31
TWI232863B (en)	2005-05-21
PE20030097A1 (es)	2003-02-08
ZA200309382B (en)	2005-03-02
ATE389659T1 (de)	2008-04-15
KR20040006030A (ko)	2004-01-16
AU2002314144B2 (en)	2008-01-31
HUP0400154A2 (hu)	2004-07-28
IL158905A (en)	2008-12-29
US7504390B2 (en)	2009-03-17
CA2450274C (en)	2010-12-21
MXPA03011563A (es)	2004-03-18
IS7036A (is)	2003-11-13
CA2450274A1 (en)	2002-12-19
CN1514835A (zh)	2004-07-21
IS2526B (is)	2009-07-15

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NO20035486D0 (no)	2003-12-10	Benzodiazepinderivater og deres anvendelse som AMPA- reseptorstimulatorer
NO20004144D0 (no)	2000-08-18	Heterocykliske forbindelser, deres fremstilling og anvendelse som takykinin reseptor antagonister
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Legal Events

Date	Code	Title	Description
2013-02-04	MM1K	Lapsed by not paying the annual fees