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UY29384A1 - Derivados del ácido2-3s,4r)-4-(((3,4-dicloro-5-metil-1h-pirrol-2-il) carbonil)amino)-1,3-tiazol-5-carboxílico y sus sales, composiciones farmacéuticas que los contienen, procedimientos de preparación y aplicaciónes. - Google Patents

Derivados del ácido2-3s,4r)-4-(((3,4-dicloro-5-metil-1h-pirrol-2-il) carbonil)amino)-1,3-tiazol-5-carboxílico y sus sales, composiciones farmacéuticas que los contienen, procedimientos de preparación y aplicaciónes.

Info

Publication number
UY29384A1
UY29384A1 UY29384A UY29384A UY29384A1 UY 29384 A1 UY29384 A1 UY 29384A1 UY 29384 A UY29384 A UY 29384A UY 29384 A UY29384 A UY 29384A UY 29384 A1 UY29384 A1 UY 29384A1
Authority
UY
Uruguay
Prior art keywords
pharmaceutical compositions
carbonil
pirrol
tiazol
dicloro
Prior art date
Application number
UY29384A
Other languages
English (en)
Inventor
Basarab Greg
Dangel Brian
Fleming Paulrobert
Gravestock Michael Barry
Green Oluyinka
Hauck Sheila Irene
Hill Pamela
Hull Kenneth Gregory
Mullen George
Sherer Brian
Zhou Fei
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36218455&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY29384(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of UY29384A1 publication Critical patent/UY29384A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Se describen compuestos de fórmula (I) y sus sales farmacéuticamente aceptables. También se describen procesos para su preparación, composiciones farmacéuticas que los contienen, su uso como medicamento y su uso en el tratamiento de infecciones bacterianas.
UY29384A 2005-02-18 2006-02-17 Derivados del ácido2-3s,4r)-4-(((3,4-dicloro-5-metil-1h-pirrol-2-il) carbonil)amino)-1,3-tiazol-5-carboxílico y sus sales, composiciones farmacéuticas que los contienen, procedimientos de preparación y aplicaciónes. UY29384A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US65467005P 2005-02-18 2005-02-18

Publications (1)

Publication Number Publication Date
UY29384A1 true UY29384A1 (es) 2006-10-02

Family

ID=36218455

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29384A UY29384A1 (es) 2005-02-18 2006-02-17 Derivados del ácido2-3s,4r)-4-(((3,4-dicloro-5-metil-1h-pirrol-2-il) carbonil)amino)-1,3-tiazol-5-carboxílico y sus sales, composiciones farmacéuticas que los contienen, procedimientos de preparación y aplicaciónes.

Country Status (21)

Country Link
US (2) US8399489B2 (es)
EP (1) EP1853586B1 (es)
JP (4) JP4058106B2 (es)
KR (2) KR20070113233A (es)
CN (1) CN101163693B (es)
AR (1) AR053683A1 (es)
AU (1) AU2006215399B2 (es)
BR (1) BRPI0607756A2 (es)
CA (1) CA2598423C (es)
ES (1) ES2430569T3 (es)
IL (1) IL185306A (es)
MX (1) MX2007010072A (es)
NO (1) NO20074703L (es)
NZ (1) NZ561613A (es)
RU (1) RU2424240C2 (es)
SA (1) SA06270020B1 (es)
TW (1) TWI402263B (es)
UA (1) UA94901C2 (es)
UY (1) UY29384A1 (es)
WO (1) WO2006087543A1 (es)
ZA (1) ZA200706920B (es)

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Also Published As

Publication number Publication date
NO20074703L (no) 2007-11-14
SA06270020B1 (ar) 2010-10-23
TWI402263B (zh) 2013-07-21
HK1114376A1 (en) 2008-10-31
IL185306A (en) 2012-05-31
MX2007010072A (es) 2008-01-28
KR20130093174A (ko) 2013-08-21
ZA200706920B (en) 2008-06-25
CA2598423A1 (en) 2006-08-24
KR101422432B1 (ko) 2014-07-22
RU2424240C2 (ru) 2011-07-20
US8399489B2 (en) 2013-03-19
CN101163693B (zh) 2013-03-06
UA94901C2 (ru) 2011-06-25
BRPI0607756A2 (pt) 2010-05-18
IL185306A0 (en) 2008-02-09
WO2006087543A8 (en) 2007-10-18
US20100179150A1 (en) 2010-07-15
US20130150366A1 (en) 2013-06-13
ES2430569T3 (es) 2013-11-21
NZ561613A (en) 2010-12-24
CN101163693A (zh) 2008-04-16
JP2007326882A (ja) 2007-12-20
JP2008500321A (ja) 2008-01-10
AU2006215399B2 (en) 2010-12-09
CA2598423C (en) 2014-05-27
AU2006215399A1 (en) 2006-08-24
TW200640908A (en) 2006-12-01
JP2008024715A (ja) 2008-02-07
RU2007134380A (ru) 2009-03-27
JP2007326883A (ja) 2007-12-20
WO2006087543A1 (en) 2006-08-24
EP1853586A1 (en) 2007-11-14
JP4058106B2 (ja) 2008-03-05
EP1853586B1 (en) 2013-07-24
AR053683A1 (es) 2007-05-16
KR20070113233A (ko) 2007-11-28

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