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MX2007010072A - Derivados de piperidina antibacterianos. - Google Patents

Derivados de piperidina antibacterianos.

Info

Publication number
MX2007010072A
MX2007010072A MX2007010072A MX2007010072A MX2007010072A MX 2007010072 A MX2007010072 A MX 2007010072A MX 2007010072 A MX2007010072 A MX 2007010072A MX 2007010072 A MX2007010072 A MX 2007010072A MX 2007010072 A MX2007010072 A MX 2007010072A
Authority
MX
Mexico
Prior art keywords
antibacterial
piperidine derivatives
formula
medicaments
compounds
Prior art date
Application number
MX2007010072A
Other languages
English (en)
Inventor
Greg Basarab
Brian Dangel
Paul Robert Fleming
Michael Barry Gravestock
Oluyinka Green
Sheila Irene Hauck
Pamela Hill
Kenneth Gregory Hull
George Mullen
Brian Sherer
Fei Zhou
Haihong Ni
Original Assignee
Astrazeneca Ab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=36218455&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=MX2007010072(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Astrazeneca Ab filed Critical Astrazeneca Ab
Publication of MX2007010072A publication Critical patent/MX2007010072A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing three or more hetero rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/541—Non-condensed thiazines containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Hydrogenated Pyridines (AREA)

Abstract

Se describen compuestos de la formula (I) y sus sales farmaceuticamente aceptables (ver formula (I)): Tambien se describen procesos para su preparacion, composiciones farmaceuticas que los contienen, su uso como medicamentos, y su uso en el tratamiento de infecciones bacterianas.
MX2007010072A 2005-02-18 2006-02-16 Derivados de piperidina antibacterianos. MX2007010072A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US65467005P 2005-02-18 2005-02-18
PCT/GB2006/000529 WO2006087543A1 (en) 2005-02-18 2006-02-16 Antibacterial piperidine derivatives

Publications (1)

Publication Number Publication Date
MX2007010072A true MX2007010072A (es) 2008-01-28

Family

ID=36218455

Family Applications (1)

Application Number Title Priority Date Filing Date
MX2007010072A MX2007010072A (es) 2005-02-18 2006-02-16 Derivados de piperidina antibacterianos.

Country Status (21)

Country Link
US (2) US8399489B2 (es)
EP (1) EP1853586B1 (es)
JP (4) JP4058106B2 (es)
KR (2) KR101422432B1 (es)
CN (1) CN101163693B (es)
AR (1) AR053683A1 (es)
AU (1) AU2006215399B2 (es)
BR (1) BRPI0607756A2 (es)
CA (1) CA2598423C (es)
ES (1) ES2430569T3 (es)
IL (1) IL185306A (es)
MX (1) MX2007010072A (es)
NO (1) NO20074703L (es)
NZ (1) NZ561613A (es)
RU (1) RU2424240C2 (es)
SA (1) SA06270020B1 (es)
TW (1) TWI402263B (es)
UA (1) UA94901C2 (es)
UY (1) UY29384A1 (es)
WO (1) WO2006087543A1 (es)
ZA (1) ZA200706920B (es)

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WO2006087543A1 (en) * 2005-02-18 2006-08-24 Astrazeneca Ab Antibacterial piperidine derivatives
US20090253671A1 (en) * 2005-03-04 2009-10-08 Astrazeneca Ab Tricyclic derivatives of azetidine and pyrrole with antibacterial activity
MY150958A (en) 2005-06-16 2014-03-31 Astrazeneca Ab Compounds for the treatment of multi-drug resistant bacterial infections
TW200819437A (en) * 2006-08-17 2008-05-01 Astrazeneca Ab Chemical compounds
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TW201026694A (en) 2008-12-12 2010-07-16 Astrazeneca Ab Compound 468
US8071605B2 (en) 2008-12-12 2011-12-06 Astrazeneca Ab Piperidine compounds for use in the treatment of bacterial infections
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Also Published As

Publication number Publication date
KR20070113233A (ko) 2007-11-28
AR053683A1 (es) 2007-05-16
HK1114376A1 (en) 2008-10-31
US8399489B2 (en) 2013-03-19
JP4058106B2 (ja) 2008-03-05
AU2006215399B2 (en) 2010-12-09
CA2598423A1 (en) 2006-08-24
JP2008024715A (ja) 2008-02-07
NZ561613A (en) 2010-12-24
RU2424240C2 (ru) 2011-07-20
CN101163693A (zh) 2008-04-16
US20100179150A1 (en) 2010-07-15
KR101422432B1 (ko) 2014-07-22
UY29384A1 (es) 2006-10-02
ZA200706920B (en) 2008-06-25
WO2006087543A1 (en) 2006-08-24
IL185306A0 (en) 2008-02-09
AU2006215399A1 (en) 2006-08-24
BRPI0607756A2 (pt) 2010-05-18
CA2598423C (en) 2014-05-27
TW200640908A (en) 2006-12-01
ES2430569T3 (es) 2013-11-21
US20130150366A1 (en) 2013-06-13
RU2007134380A (ru) 2009-03-27
EP1853586B1 (en) 2013-07-24
KR20130093174A (ko) 2013-08-21
IL185306A (en) 2012-05-31
JP2007326882A (ja) 2007-12-20
EP1853586A1 (en) 2007-11-14
JP2007326883A (ja) 2007-12-20
JP2008500321A (ja) 2008-01-10
NO20074703L (no) 2007-11-14
WO2006087543A8 (en) 2007-10-18
TWI402263B (zh) 2013-07-21
UA94901C2 (ru) 2011-06-25
SA06270020B1 (ar) 2010-10-23
CN101163693B (zh) 2013-03-06

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