UY29285A1 - Macrolidos - Google Patents
MacrolidosInfo
- Publication number
- UY29285A1 UY29285A1 UY29285A UY29285A UY29285A1 UY 29285 A1 UY29285 A1 UY 29285A1 UY 29285 A UY29285 A UY 29285A UY 29285 A UY29285 A UY 29285A UY 29285 A1 UY29285 A1 UY 29285A1
- Authority
- UY
- Uruguay
- Prior art keywords
- compounds
- methods
- macrolidos
- famraceutical
- intermediates
- Prior art date
Links
- 150000001875 compounds Chemical class 0.000 abstract 3
- 241001465754 Metazoa Species 0.000 abstract 1
- 239000003242 anti bacterial agent Substances 0.000 abstract 1
- 230000000844 anti-bacterial effect Effects 0.000 abstract 1
- 239000003904 antiprotozoal agent Substances 0.000 abstract 1
- 201000010099 disease Diseases 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 239000000543 intermediate Substances 0.000 abstract 1
- 239000003120 macrolide antibiotic agent Substances 0.000 abstract 1
- 239000000203 mixture Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
- C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P33/00—Antiparasitic agents
- A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Molecular Biology (AREA)
- Public Health (AREA)
- Medicinal Chemistry (AREA)
- Pharmacology & Pharmacy (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Biotechnology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Genetics & Genomics (AREA)
- Engineering & Computer Science (AREA)
- Biochemistry (AREA)
- Communicable Diseases (AREA)
- Oncology (AREA)
- Tropical Medicine & Parasitology (AREA)
- Epidemiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Saccharide Compounds (AREA)
- Cephalosporin Compounds (AREA)
- Tires In General (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Polysaccharides And Polysaccharide Derivatives (AREA)
Abstract
Compuestos macrólidos per se, como se muestran a continuación y se definen en esta memoria, y su uso, p. ej., como agentes antibacterianos y antiprotozoarios en animales, incluyendo seres humanos: También se describen métodos para preparar los compuestos, productos intermedios y sus composiciones famracéuticas, y métodos para tratar o prevenir la enfermedad por administración de los compuestos a los sujetos que lo necesiten, Este resumen es sólo un extracto y no limita la invención.
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US63809704P | 2004-12-21 | 2004-12-21 | |
| US71753005P | 2005-09-14 | 2005-09-14 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| UY29285A1 true UY29285A1 (es) | 2006-07-31 |
Family
ID=35809765
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY29285A UY29285A1 (es) | 2004-12-21 | 2005-12-21 | Macrolidos |
Country Status (35)
| Country | Link |
|---|---|
| US (1) | US7462600B2 (es) |
| EP (2) | EP2233493A1 (es) |
| JP (1) | JP4111994B1 (es) |
| KR (1) | KR100897678B1 (es) |
| CN (1) | CN101120011A (es) |
| AP (1) | AP2007004026A0 (es) |
| AR (1) | AR052824A1 (es) |
| AT (1) | ATE459633T1 (es) |
| AU (1) | AU2005317735B2 (es) |
| BR (1) | BRPI0519135A2 (es) |
| CA (1) | CA2591746A1 (es) |
| CR (1) | CR9202A (es) |
| DE (1) | DE602005019786D1 (es) |
| DK (1) | DK1836211T3 (es) |
| EA (1) | EA011281B1 (es) |
| ES (1) | ES2339871T3 (es) |
| GE (1) | GEP20094834B (es) |
| GT (1) | GT200500378A (es) |
| HN (1) | HN2005036113A (es) |
| HR (1) | HRP20100253T1 (es) |
| IL (1) | IL183661A0 (es) |
| MA (1) | MA29108B1 (es) |
| MX (1) | MX2007007598A (es) |
| NL (1) | NL1030713C2 (es) |
| NO (1) | NO20073367L (es) |
| PE (1) | PE20060948A1 (es) |
| PL (1) | PL1836211T3 (es) |
| PT (1) | PT1836211E (es) |
| SI (1) | SI1836211T1 (es) |
| TN (1) | TNSN07233A1 (es) |
| TW (1) | TW200626608A (es) |
| UA (1) | UA85937C2 (es) |
| UY (1) | UY29285A1 (es) |
| WO (1) | WO2006067589A1 (es) |
| ZA (1) | ZA200705108B (es) |
Families Citing this family (23)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US9133212B1 (en) | 2005-06-15 | 2015-09-15 | Vanderbilt University | Inhibitors of hemeprotein-catalyzed lipid peroxidation |
| US8367669B2 (en) * | 2005-06-15 | 2013-02-05 | Vanderbilt University | Inhibitors of hemeprotein-catalyzed lipid peroxidation |
| HRP20171285T1 (hr) | 2005-08-24 | 2017-10-20 | Melinta Therapeutics, Inc. | Spojevi triazola i postupci dobivanja i njihova upotreba |
| WO2008110918A2 (en) * | 2007-03-13 | 2008-09-18 | Pfizer Products Inc. | Erythromycin-based macrolides |
| AU2008227216A1 (en) * | 2007-03-21 | 2008-09-25 | Creative Antibiotics Sweden Ab | Method and means for preventing and inhibiting type III secretion in infections caused by gram-negative bacteria |
| WO2009053259A1 (en) * | 2007-10-25 | 2009-04-30 | Sandoz Ag | Process for the production of telithromycin |
| AU2008316830B2 (en) | 2007-10-25 | 2016-03-17 | Cempra Pharmaceuticals, Inc. | Process for the preparation of macrolide antibacterial agents |
| EP2225239B1 (en) | 2007-12-21 | 2014-10-22 | F. Hoffmann-La Roche AG | Heterocyclic antiviral compounds |
| WO2011018510A1 (en) * | 2009-08-13 | 2011-02-17 | Basilea Pharmaceutica Ag | New macrolides and their use |
| NZ602544A (en) * | 2010-03-22 | 2014-11-28 | Cempra Pharmaceuticals Inc | Crystalline forms of a macrolide, and uses therefor |
| WO2012142125A2 (en) | 2011-04-12 | 2012-10-18 | The United States Of America, As Represented By The Secretary, Department Of Health And Human Services | Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria |
| CN102558047B (zh) * | 2011-12-14 | 2013-10-30 | 天津药物研究院药业有限责任公司 | 3-甲基喹啉的制备方法 |
| SG11201405895UA (en) | 2012-03-27 | 2014-10-30 | Cempra Pharmaceuticals Inc | Parenteral formulations for administering macrolide antibiotics |
| RU2015103119A (ru) | 2012-07-13 | 2016-08-27 | Ф. Хоффманн-Ля Рош Аг | Антипролиферативные бензо[в]азепин-2-оны |
| KR101612179B1 (ko) * | 2013-04-19 | 2016-04-12 | 영남대학교 산학협력단 | 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 암질환 예방 또는 치료용 약학조성물 |
| TW201534586A (zh) | 2013-06-11 | 2015-09-16 | Orion Corp | 新穎cyp17抑制劑/抗雄激素劑 |
| CN103739643A (zh) * | 2013-12-30 | 2014-04-23 | 华东理工大学 | 利用分子印迹技术对红霉素进行回收分离纯化的方法 |
| CN104230891B (zh) * | 2014-08-27 | 2016-03-30 | 于宗光 | 一种托匹司他的制备方法 |
| EP3522896A4 (en) | 2016-10-04 | 2020-06-17 | Biopharmati SA | KETOLID WITH ANTIBACTERIAL EFFECT |
| CN114340616A (zh) * | 2019-06-04 | 2022-04-12 | 海格生物科学有限责任公司 | 作为食欲肽拮抗剂的吡唑和咪唑衍生物、组合物以及方法 |
| SG11202112827QA (en) | 2019-06-04 | 2021-12-30 | Hager Biosciences Llc | Imidazolo derivatives, compositions and methods as orexin antagonists |
| CN111793022A (zh) * | 2020-04-27 | 2020-10-20 | 滁州拜奥生物科技有限公司 | 一种3-甲基喹啉的制备方法 |
| CN120417896A (zh) * | 2022-09-01 | 2025-08-01 | 海格生物科学有限责任公司 | 作为食欲素和κ-阿片受体双重调节剂的吡唑和咪唑衍生物、组合物、用于治疗神经和精神病患的方法 |
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|---|---|---|---|---|
| US2653899A (en) | 1952-04-14 | 1953-09-29 | Lilly Co Eli | Erythromycin, its salts, and method of preparation |
| US2823203A (en) | 1954-06-24 | 1958-02-11 | Abbott Lab | Method of producing substantially pure erythromycin a |
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| US4474768A (en) | 1982-07-19 | 1984-10-02 | Pfizer Inc. | N-Methyl 11-aza-10-deoxo-10-dihydro-erytromycin A, intermediates therefor |
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| IE70593B1 (en) | 1989-09-29 | 1996-12-11 | Eisai Co Ltd | Biphenylmethane derivative the use of it and pharmacological compositions containing same |
| US5523399A (en) | 1991-12-27 | 1996-06-04 | Taisho Pharmaceutical Co., Ltd. | 5-O-desosaminylerythronolide derivatives |
| FR2697524B1 (fr) | 1992-11-05 | 1994-12-23 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
| US5527780A (en) | 1992-11-05 | 1996-06-18 | Roussel Uclaf | Erythromycin derivatives |
| FR2719587B1 (fr) | 1994-05-03 | 1996-07-12 | Roussel Uclaf | Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments. |
| US5629322A (en) | 1994-11-15 | 1997-05-13 | Merck & Co., Inc. | Cyclic amidine analogs as inhibitors of nitric oxide synthase |
| FR2727969B1 (fr) | 1994-12-09 | 1997-01-17 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| US5747466A (en) | 1995-11-08 | 1998-05-05 | Abbott Laboratories | 3-deoxy-3-descladinose derivatives of erythromycins A and B |
| FR2742757B1 (fr) | 1995-12-22 | 1998-01-30 | Roussel Uclaf | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| US5750510A (en) | 1997-04-04 | 1998-05-12 | Abbott Laboratories | 3-descladinose-2,3-anhydroerythromycin derivatives |
| JP2000509712A (ja) | 1996-05-07 | 2000-08-02 | アボツト・ラボラトリーズ | 6―o―置換エリスロマイシン及びその製造方法 |
| FR2748746B1 (fr) | 1996-05-14 | 1998-08-14 | Hoechst Marion Roussel Inc | Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine |
| US6271255B1 (en) | 1996-07-05 | 2001-08-07 | Biotica Technology Limited | Erythromycins and process for their preparation |
| FR2751656B1 (fr) | 1996-07-24 | 1998-10-16 | Hoechst Marion Roussel Inc | Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments |
| CN1273475C (zh) | 1996-09-04 | 2006-09-06 | 艾博特公司 | 具有抗细菌活性的6-0-取代的酮基内酯类化合物 |
| US5804565A (en) | 1996-09-24 | 1998-09-08 | Taisho Pharmaceutical Co., Ltd. | Erythromycin A derivatives |
| CN1238777A (zh) | 1996-11-27 | 1999-12-15 | 大正制药株式会社 | 红霉素a衍生物 |
| US6140479A (en) | 1997-03-24 | 2000-10-31 | Taisho Pharmaceuticals Co., Ltd. | Erythromycin a derivatives |
| US6162794A (en) | 1997-05-09 | 2000-12-19 | Pfizer Inc. | Erythromycin derivatives |
| US20020025937A1 (en) | 2000-03-20 | 2002-02-28 | Yong-Jin Wu | 9-oxime erythromycin derivatives |
| EP0895999A1 (en) | 1997-08-06 | 1999-02-10 | Pfizer Products Inc. | C-4" substituted macrolide antibiotics |
| ZA987689B (en) | 1997-09-02 | 1999-02-24 | Abbott Lab | 3-descladinose 6-O substituted erythromycin derivatives |
| US6034069A (en) | 1997-09-30 | 2000-03-07 | Abbott Laboratories | 3-'N-modified 6-O-substituted erythromycin ketolide derivatives having antibacterial activity |
| PA8461401A1 (es) | 1997-10-29 | 2000-05-24 | Pfizer Prod Inc | Derivados de eritromicina triciclicos |
| HN1998000159A (es) | 1997-10-29 | 1999-02-09 | Monsanto Co | Derivados de 9- amino - 3 ceto eritromicina |
| ZA989835B (en) | 1997-10-29 | 1999-05-05 | Taisho Pharmaceutical Co Ltd | Erythromycin a derivatives |
| AP1060A (en) | 1998-01-02 | 2002-04-23 | Pfizer Prod Inc | Novel erythromycin derivatives. |
| AP9801420A0 (en) | 1998-01-02 | 1998-12-31 | Pfizer Prod Inc | Novel macrolides. |
| EP0941998B1 (en) | 1998-03-03 | 2004-09-01 | Pfizer Products Inc. | 3,6-ketal macrolide antibiotics |
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| AU3439899A (en) | 1998-06-03 | 1999-12-20 | Pfizer Products Inc. | Tricyclic 3-keto derivatives of 6-o-methylerythromycin |
| JP4573925B2 (ja) | 1998-07-09 | 2010-11-04 | アベンティス・ファーマ・ソシエテ・アノニム | 新規のエリスロマイシン誘導体、その製造方法及びその薬剤としての使用 |
| US6020521A (en) | 1998-08-26 | 2000-02-01 | Abbott Laboratories | Macrolide LHRH antagonists |
| US6387885B1 (en) | 1998-08-26 | 2002-05-14 | Abbott Laboratories | 3′,3′-N-bis-desmethyl-3′-N-cycloalkyl erythromycin derivatives as LHRH antagonists |
| US6262030B1 (en) | 1998-11-03 | 2001-07-17 | Pfizer Inc. | Erythromycin derivatives |
| TR200200436T2 (tr) | 1998-11-03 | 2002-06-21 | Pfizer Inc. | Yeni makrolit antibiyotikler |
| WO2000034297A1 (en) | 1998-12-10 | 2000-06-15 | Pfizer Products Inc. | Carbamate and carbazate ketolide antibiotics |
| SI1147121T1 (en) | 1999-01-27 | 2004-04-30 | Pfizer Products Inc. | Ketolide antibiotics |
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| US6939861B2 (en) | 1999-04-16 | 2005-09-06 | Kosan Biosciences, Inc. | Amido macrolides |
| CN1373767A (zh) * | 1999-04-16 | 2002-10-09 | 奥索-麦克尼尔药品公司 | 酮式大环内酯抗菌剂 |
| KR20020007374A (ko) | 1999-04-16 | 2002-01-26 | 추후제출 | 매크롤라이드 항감염제 |
| US20020077302A1 (en) | 1999-04-23 | 2002-06-20 | Yong-Jin Wu | Tricyclic erythromycin derivatives |
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| US20020115621A1 (en) | 2000-08-07 | 2002-08-22 | Wei-Gu Su | Macrolide antibiotics |
| HUP0302526A2 (hu) | 2000-12-21 | 2003-11-28 | Glaxo Group Limited | Makrolid vegyületek, eljárás az előállításukra, alkalmazásuk és ezeket tartalmazó gyógyszerkészítmények |
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| RU2397987C2 (ru) | 2004-07-28 | 2010-08-27 | Рэнбакси Лабораториз Лимитед | Кетолидные производные в качестве антибактериальных агентов |
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-
2005
- 2005-12-12 DE DE602005019786T patent/DE602005019786D1/de active Active
- 2005-12-12 DK DK05813939.5T patent/DK1836211T3/da active
- 2005-12-12 PL PL05813939T patent/PL1836211T3/pl unknown
- 2005-12-12 KR KR1020077014160A patent/KR100897678B1/ko not_active Expired - Fee Related
- 2005-12-12 AP AP2007004026A patent/AP2007004026A0/xx unknown
- 2005-12-12 AU AU2005317735A patent/AU2005317735B2/en not_active Ceased
- 2005-12-12 GE GEAP200510142A patent/GEP20094834B/en unknown
- 2005-12-12 BR BRPI0519135-1A patent/BRPI0519135A2/pt not_active IP Right Cessation
- 2005-12-12 WO PCT/IB2005/003829 patent/WO2006067589A1/en not_active Ceased
- 2005-12-12 SI SI200530941T patent/SI1836211T1/sl unknown
- 2005-12-12 CA CA002591746A patent/CA2591746A1/en not_active Abandoned
- 2005-12-12 EA EA200701113A patent/EA011281B1/ru not_active IP Right Cessation
- 2005-12-12 EP EP10154783A patent/EP2233493A1/en not_active Withdrawn
- 2005-12-12 EP EP05813939A patent/EP1836211B1/en active Active
- 2005-12-12 ES ES05813939T patent/ES2339871T3/es active Active
- 2005-12-12 CN CNA2005800482465A patent/CN101120011A/zh active Pending
- 2005-12-12 PT PT05813939T patent/PT1836211E/pt unknown
- 2005-12-12 MX MX2007007598A patent/MX2007007598A/es active IP Right Grant
- 2005-12-12 UA UAA200706959A patent/UA85937C2/uk unknown
- 2005-12-12 AT AT05813939T patent/ATE459633T1/de not_active IP Right Cessation
- 2005-12-12 HR HR20100253T patent/HRP20100253T1/hr unknown
- 2005-12-12 JP JP2007547694A patent/JP4111994B1/ja not_active Expired - Fee Related
- 2005-12-14 PE PE2005001462A patent/PE20060948A1/es not_active Application Discontinuation
- 2005-12-19 HN HN2005036113A patent/HN2005036113A/es unknown
- 2005-12-20 GT GT200500378A patent/GT200500378A/es unknown
- 2005-12-20 TW TW094145385A patent/TW200626608A/zh unknown
- 2005-12-20 AR ARP050105370A patent/AR052824A1/es unknown
- 2005-12-20 NL NL1030713A patent/NL1030713C2/nl not_active IP Right Cessation
- 2005-12-21 US US11/313,523 patent/US7462600B2/en not_active Expired - Fee Related
- 2005-12-21 UY UY29285A patent/UY29285A1/es not_active Application Discontinuation
-
2007
- 2007-06-04 IL IL183661A patent/IL183661A0/en unknown
- 2007-06-15 ZA ZA200705108A patent/ZA200705108B/xx unknown
- 2007-06-20 TN TNP2007000233A patent/TNSN07233A1/fr unknown
- 2007-06-21 CR CR9202A patent/CR9202A/es not_active Application Discontinuation
- 2007-06-21 MA MA30024A patent/MA29108B1/fr unknown
- 2007-06-29 NO NO20073367A patent/NO20073367L/no not_active Application Discontinuation
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| 109 | Application deemed to be withdrawn |
Effective date: 20160606 |