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UY29285A1 - Macrolidos - Google Patents

Macrolidos

Info

Publication number
UY29285A1
UY29285A1 UY29285A UY29285A UY29285A1 UY 29285 A1 UY29285 A1 UY 29285A1 UY 29285 A UY29285 A UY 29285A UY 29285 A UY29285 A UY 29285A UY 29285 A1 UY29285 A1 UY 29285A1
Authority
UY
Uruguay
Prior art keywords
compounds
methods
macrolidos
famraceutical
intermediates
Prior art date
Application number
UY29285A
Other languages
English (en)
Inventor
Takushi Kaneko
Mark Edward Flanagan
Louis Stanley Chupak
Thomas Victor Magee
Mark Carl Noe
Usa Reilly
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35809765&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY29285(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of UY29285A1 publication Critical patent/UY29285A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Tires In General (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)

Abstract

Compuestos macrólidos per se, como se muestran a continuación y se definen en esta memoria, y su uso, p. ej., como agentes antibacterianos y antiprotozoarios en animales, incluyendo seres humanos: También se describen métodos para preparar los compuestos, productos intermedios y sus composiciones famracéuticas, y métodos para tratar o prevenir la enfermedad por administración de los compuestos a los sujetos que lo necesiten, Este resumen es sólo un extracto y no limita la invención.
UY29285A 2004-12-21 2005-12-21 Macrolidos UY29285A1 (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63809704P 2004-12-21 2004-12-21
US71753005P 2005-09-14 2005-09-14

Publications (1)

Publication Number Publication Date
UY29285A1 true UY29285A1 (es) 2006-07-31

Family

ID=35809765

Family Applications (1)

Application Number Title Priority Date Filing Date
UY29285A UY29285A1 (es) 2004-12-21 2005-12-21 Macrolidos

Country Status (35)

Country Link
US (1) US7462600B2 (es)
EP (2) EP2233493A1 (es)
JP (1) JP4111994B1 (es)
KR (1) KR100897678B1 (es)
CN (1) CN101120011A (es)
AP (1) AP2007004026A0 (es)
AR (1) AR052824A1 (es)
AT (1) ATE459633T1 (es)
AU (1) AU2005317735B2 (es)
BR (1) BRPI0519135A2 (es)
CA (1) CA2591746A1 (es)
CR (1) CR9202A (es)
DE (1) DE602005019786D1 (es)
DK (1) DK1836211T3 (es)
EA (1) EA011281B1 (es)
ES (1) ES2339871T3 (es)
GE (1) GEP20094834B (es)
GT (1) GT200500378A (es)
HN (1) HN2005036113A (es)
HR (1) HRP20100253T1 (es)
IL (1) IL183661A0 (es)
MA (1) MA29108B1 (es)
MX (1) MX2007007598A (es)
NL (1) NL1030713C2 (es)
NO (1) NO20073367L (es)
PE (1) PE20060948A1 (es)
PL (1) PL1836211T3 (es)
PT (1) PT1836211E (es)
SI (1) SI1836211T1 (es)
TN (1) TNSN07233A1 (es)
TW (1) TW200626608A (es)
UA (1) UA85937C2 (es)
UY (1) UY29285A1 (es)
WO (1) WO2006067589A1 (es)
ZA (1) ZA200705108B (es)

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US8367669B2 (en) * 2005-06-15 2013-02-05 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
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AU2008316830B2 (en) 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
EP2225239B1 (en) 2007-12-21 2014-10-22 F. Hoffmann-La Roche AG Heterocyclic antiviral compounds
WO2011018510A1 (en) * 2009-08-13 2011-02-17 Basilea Pharmaceutica Ag New macrolides and their use
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WO2012142125A2 (en) 2011-04-12 2012-10-18 The United States Of America, As Represented By The Secretary, Department Of Health And Human Services Plasmodial surface anion channel inhibitors for the treatment or prevention of malaria
CN102558047B (zh) * 2011-12-14 2013-10-30 天津药物研究院药业有限责任公司 3-甲基喹啉的制备方法
SG11201405895UA (en) 2012-03-27 2014-10-30 Cempra Pharmaceuticals Inc Parenteral formulations for administering macrolide antibiotics
RU2015103119A (ru) 2012-07-13 2016-08-27 Ф. Хоффманн-Ля Рош Аг Антипролиферативные бензо[в]азепин-2-оны
KR101612179B1 (ko) * 2013-04-19 2016-04-12 영남대학교 산학협력단 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 암질환 예방 또는 치료용 약학조성물
TW201534586A (zh) 2013-06-11 2015-09-16 Orion Corp 新穎cyp17抑制劑/抗雄激素劑
CN103739643A (zh) * 2013-12-30 2014-04-23 华东理工大学 利用分子印迹技术对红霉素进行回收分离纯化的方法
CN104230891B (zh) * 2014-08-27 2016-03-30 于宗光 一种托匹司他的制备方法
EP3522896A4 (en) 2016-10-04 2020-06-17 Biopharmati SA KETOLID WITH ANTIBACTERIAL EFFECT
CN114340616A (zh) * 2019-06-04 2022-04-12 海格生物科学有限责任公司 作为食欲肽拮抗剂的吡唑和咪唑衍生物、组合物以及方法
SG11202112827QA (en) 2019-06-04 2021-12-30 Hager Biosciences Llc Imidazolo derivatives, compositions and methods as orexin antagonists
CN111793022A (zh) * 2020-04-27 2020-10-20 滁州拜奥生物科技有限公司 一种3-甲基喹啉的制备方法
CN120417896A (zh) * 2022-09-01 2025-08-01 海格生物科学有限责任公司 作为食欲素和κ-阿片受体双重调节剂的吡唑和咪唑衍生物、组合物、用于治疗神经和精神病患的方法

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Also Published As

Publication number Publication date
JP2008524319A (ja) 2008-07-10
HN2005036113A (es) 2010-12-06
PT1836211E (pt) 2010-04-08
EP2233493A1 (en) 2010-09-29
EA011281B1 (ru) 2009-02-27
TNSN07233A1 (fr) 2008-11-21
EA200701113A1 (ru) 2007-12-28
HRP20100253T1 (hr) 2010-06-30
ZA200705108B (en) 2009-01-28
MX2007007598A (es) 2007-07-25
JP4111994B1 (ja) 2008-07-02
GEP20094834B (en) 2009-11-25
CR9202A (es) 2007-07-16
NL1030713A1 (nl) 2006-06-22
ATE459633T1 (de) 2010-03-15
SI1836211T1 (sl) 2010-04-30
IL183661A0 (en) 2007-09-20
US7462600B2 (en) 2008-12-09
KR100897678B1 (ko) 2009-05-14
AU2005317735B2 (en) 2009-06-04
MA29108B1 (fr) 2007-12-03
UA85937C2 (uk) 2009-03-10
AP2007004026A0 (en) 2007-06-30
KR20070089191A (ko) 2007-08-30
CN101120011A (zh) 2008-02-06
EP1836211A1 (en) 2007-09-26
WO2006067589A1 (en) 2006-06-29
AU2005317735A1 (en) 2006-06-29
US20060135447A1 (en) 2006-06-22
NL1030713C2 (nl) 2006-12-12
ES2339871T3 (es) 2010-05-26
BRPI0519135A2 (pt) 2008-12-23
NO20073367L (no) 2007-09-05
EP1836211B1 (en) 2010-03-03
DK1836211T3 (da) 2010-05-17
PE20060948A1 (es) 2006-10-11
GT200500378A (es) 2006-11-28
PL1836211T3 (pl) 2010-07-30
TW200626608A (en) 2006-08-01
DE602005019786D1 (de) 2010-04-15
AR052824A1 (es) 2007-04-04
CA2591746A1 (en) 2006-06-29

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