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HN2005036113A - Macrolidos - Google Patents

Macrolidos

Info

Publication number
HN2005036113A
HN2005036113A HN2005036113A HN2005036113A HN2005036113A HN 2005036113 A HN2005036113 A HN 2005036113A HN 2005036113 A HN2005036113 A HN 2005036113A HN 2005036113 A HN2005036113 A HN 2005036113A HN 2005036113 A HN2005036113 A HN 2005036113A
Authority
HN
Honduras
Prior art keywords
macrolidos
antiprotozoar
antibacterial
animals
agents
Prior art date
Application number
HN2005036113A
Other languages
English (en)
Inventor
Stanley Chupak Lous
Edward Flanagan Mark
Kaneko Takushi
Victor Magee Thomas
Carl Noe Mark
Reilly Usa
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=35809765&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HN2005036113(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of HN2005036113A publication Critical patent/HN2005036113A/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/70Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00Antiparasitic agents
    • A61P33/02Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Polysaccharides And Polysaccharide Derivatives (AREA)
  • Tires In General (AREA)
  • Cephalosporin Compounds (AREA)

Abstract

ESTA INVENCION SE REFIERE A COMPUESTOS MACROLIDOS Y A SU USO, POR EJEMPLO, COMO AGENTES ANTIBACTERIANOS Y ANTIPROTOZOARIOS EN ANIMALES, INCLUYENDO SERES HUMANOS.
HN2005036113A 2004-12-21 2005-12-19 Macrolidos HN2005036113A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US63809704P 2004-12-21 2004-12-21
US71753005P 2005-09-14 2005-09-14

Publications (1)

Publication Number Publication Date
HN2005036113A true HN2005036113A (es) 2010-12-06

Family

ID=35809765

Family Applications (1)

Application Number Title Priority Date Filing Date
HN2005036113A HN2005036113A (es) 2004-12-21 2005-12-19 Macrolidos

Country Status (35)

Country Link
US (1) US7462600B2 (es)
EP (2) EP1836211B1 (es)
JP (1) JP4111994B1 (es)
KR (1) KR100897678B1 (es)
CN (1) CN101120011A (es)
AP (1) AP2007004026A0 (es)
AR (1) AR052824A1 (es)
AT (1) ATE459633T1 (es)
AU (1) AU2005317735B2 (es)
BR (1) BRPI0519135A2 (es)
CA (1) CA2591746A1 (es)
CR (1) CR9202A (es)
DE (1) DE602005019786D1 (es)
DK (1) DK1836211T3 (es)
EA (1) EA011281B1 (es)
ES (1) ES2339871T3 (es)
GE (1) GEP20094834B (es)
GT (1) GT200500378A (es)
HN (1) HN2005036113A (es)
HR (1) HRP20100253T1 (es)
IL (1) IL183661A0 (es)
MA (1) MA29108B1 (es)
MX (1) MX2007007598A (es)
NL (1) NL1030713C2 (es)
NO (1) NO20073367L (es)
PE (1) PE20060948A1 (es)
PL (1) PL1836211T3 (es)
PT (1) PT1836211E (es)
SI (1) SI1836211T1 (es)
TN (1) TNSN07233A1 (es)
TW (1) TW200626608A (es)
UA (1) UA85937C2 (es)
UY (1) UY29285A1 (es)
WO (1) WO2006067589A1 (es)
ZA (1) ZA200705108B (es)

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US9133212B1 (en) 2005-06-15 2015-09-15 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
US8367669B2 (en) * 2005-06-15 2013-02-05 Vanderbilt University Inhibitors of hemeprotein-catalyzed lipid peroxidation
WO2007025098A2 (en) 2005-08-24 2007-03-01 Rib-X Pharmaceuticals, Inc. Triazole compounds and methods of making and using the same
JP4468487B1 (ja) * 2007-03-13 2010-05-26 ファイザー・プロダクツ・インク エリスロマイシンをベースとするマクロライド
EP2136806A4 (en) * 2007-03-21 2011-11-23 Creative Antibiotics Sweden Ab METHOD AND MEANS FOR PREVENTING AND SUPPRESSING TYPE III SECRETION IN INFECTIONS BY GRAM-NEGATIVE BACTERIA
US9453042B2 (en) 2007-10-25 2016-09-27 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
WO2009053259A1 (en) * 2007-10-25 2009-04-30 Sandoz Ag Process for the production of telithromycin
CN101903382B (zh) 2007-12-21 2012-11-28 弗·哈夫曼-拉罗切有限公司 杂环抗病毒化合物
US8865662B2 (en) 2009-08-13 2014-10-21 Basilea Pharmaceutica Ag Macrolides and their use
JP5711352B2 (ja) * 2010-03-22 2015-04-30 センプラ ファーマシューティカルズ,インコーポレイテッド マクロライドの結晶形、およびその使用
CN106974913A (zh) * 2011-04-12 2017-07-25 美国卫生和人力服务部 用于治疗或预防疟疾的疟原虫表面阴离子通道抑制剂
CN102558047B (zh) * 2011-12-14 2013-10-30 天津药物研究院药业有限责任公司 3-甲基喹啉的制备方法
IN2014DN08939A (es) 2012-03-27 2015-05-22 Cempra Pharmaceuticals Inc
US9611224B2 (en) 2012-07-13 2017-04-04 Hoffmann-La Roche Inc. Antiproliferative benzo [B] azepin-2-ones
KR101663864B1 (ko) * 2013-04-19 2016-10-07 영남대학교 산학협력단 아미도피리딘올 유도체 또는 이의 약제학적 허용가능한 염을 유효성분으로 함유하는 염증성 장질환의 예방 또는 치료용 약학조성물
TW201534586A (zh) 2013-06-11 2015-09-16 Orion Corp 新穎cyp17抑制劑/抗雄激素劑
CN103739643A (zh) * 2013-12-30 2014-04-23 华东理工大学 利用分子印迹技术对红霉素进行回收分离纯化的方法
CN104230891B (zh) * 2014-08-27 2016-03-30 于宗光 一种托匹司他的制备方法
JP2019533669A (ja) 2016-10-04 2019-11-21 バイオファーマティ ソシエテ アノニム 抗菌活性を有するケトライド
AU2020286381C1 (en) 2019-06-04 2025-07-10 Hager Biosciences, Llc Imidazolo derivatives, compositions and methods as orexin antagonists
AU2020288559C1 (en) * 2019-06-04 2025-07-24 Hager Biosciences, Llc Pyrazole and imidazole derivatives, compositions and methods as orexin antagonists
CN111793022A (zh) * 2020-04-27 2020-10-20 滁州拜奥生物科技有限公司 一种3-甲基喹啉的制备方法
JP2025530768A (ja) * 2022-09-01 2025-09-17 ヘイガー バイオサイエンシズ,エルエルシー 神経疾患および精神疾患の治療のための、オレキシン受容体およびカッパオピオイド受容体に対する二重調節剤としてのピラゾール誘導体およびイミダゾール誘導体、組成物、ならびに治療法

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Also Published As

Publication number Publication date
CA2591746A1 (en) 2006-06-29
ATE459633T1 (de) 2010-03-15
US20060135447A1 (en) 2006-06-22
DE602005019786D1 (de) 2010-04-15
AP2007004026A0 (en) 2007-06-30
GT200500378A (es) 2006-11-28
IL183661A0 (en) 2007-09-20
TNSN07233A1 (fr) 2008-11-21
AR052824A1 (es) 2007-04-04
KR100897678B1 (ko) 2009-05-14
AU2005317735B2 (en) 2009-06-04
MA29108B1 (fr) 2007-12-03
PL1836211T3 (pl) 2010-07-30
TW200626608A (en) 2006-08-01
DK1836211T3 (da) 2010-05-17
NL1030713A1 (nl) 2006-06-22
EA200701113A1 (ru) 2007-12-28
WO2006067589A1 (en) 2006-06-29
HRP20100253T1 (hr) 2010-06-30
PE20060948A1 (es) 2006-10-11
MX2007007598A (es) 2007-07-25
KR20070089191A (ko) 2007-08-30
AU2005317735A1 (en) 2006-06-29
JP2008524319A (ja) 2008-07-10
NO20073367L (no) 2007-09-05
CR9202A (es) 2007-07-16
UA85937C2 (uk) 2009-03-10
BRPI0519135A2 (pt) 2008-12-23
EP2233493A1 (en) 2010-09-29
SI1836211T1 (sl) 2010-04-30
ZA200705108B (en) 2009-01-28
PT1836211E (pt) 2010-04-08
US7462600B2 (en) 2008-12-09
UY29285A1 (es) 2006-07-31
EP1836211B1 (en) 2010-03-03
CN101120011A (zh) 2008-02-06
ES2339871T3 (es) 2010-05-26
EA011281B1 (ru) 2009-02-27
GEP20094834B (en) 2009-11-25
NL1030713C2 (nl) 2006-12-12
JP4111994B1 (ja) 2008-07-02
EP1836211A1 (en) 2007-09-26

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