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UA104603C2 - Protein kinase inhibitors - Google Patents

Protein kinase inhibitors

Info

Publication number
UA104603C2
UA104603C2 UAA201107836A UAA201107836A UA104603C2 UA 104603 C2 UA104603 C2 UA 104603C2 UA A201107836 A UAA201107836 A UA A201107836A UA A201107836 A UAA201107836 A UA A201107836A UA 104603 C2 UA104603 C2 UA 104603C2
Authority
UA
Ukraine
Prior art keywords
protein kinase
kinase inhibitors
useful
compound
formula
Prior art date
Application number
UAA201107836A
Other languages
English (en)
Ukrainian (uk)
Inventor
Дейвид Эндрю Коутс
Диос Магана Альфонсо Де
Прадо Гонсалес Ана Де
Прадо Каталина Мириам Филадельфа Дель
Паредес Мария Кристина Гарсиа
Лоренс Марк Гелберт
Джон Монте Нобелок
Де Ла Нава Ева Мария Мартин
Ортега Фингер Мария Долорес Мартин
Перес Хосе Антонио Мартинес
Герранс Ана Изабел Матео
Мартинес Карлос Перес
Мартинес Консепсьон Санчес
Original Assignee
Эли Лилли Энд Компани
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=42267022&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UA104603(C2) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Эли Лилли Энд Компани filed Critical Эли Лилли Энд Компани
Publication of UA104603C2 publication Critical patent/UA104603C2/ru

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D401/00Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/14Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing three or more hetero rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/506Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim not condensed and containing further heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00Antineoplastic agents
    • A61P35/02Antineoplastic agents specific for leukemia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Hematology (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)

Abstract

Это изобретение предлагает соединение Формулы (I):(I)или его фармацевтически приемлемую соль, полезные при лечении заболеваний, которые характеризуются аномальной пролиферацией клеток.
UAA201107836A 2008-12-22 2009-12-15 Protein kinase inhibitors UA104603C2 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP08380343 2008-12-22
PCT/US2009/068030 WO2010075074A1 (en) 2008-12-22 2009-12-15 Protein kinase inhibitors

Publications (1)

Publication Number Publication Date
UA104603C2 true UA104603C2 (en) 2014-02-25

Family

ID=42267022

Family Applications (1)

Application Number Title Priority Date Filing Date
UAA201107836A UA104603C2 (en) 2008-12-22 2009-12-15 Protein kinase inhibitors

Country Status (40)

Country Link
US (1) US7855211B2 (ru)
EP (1) EP2379528B1 (ru)
JP (1) JP5417453B2 (ru)
KR (1) KR101297497B1 (ru)
CN (1) CN102264725B (ru)
AR (1) AR074575A1 (ru)
AU (1) AU2009330365B2 (ru)
BR (1) BRPI0924183B8 (ru)
CA (1) CA2747055C (ru)
CO (1) CO6382125A2 (ru)
CR (1) CR20110343A (ru)
CY (1) CY2019009I1 (ru)
DK (1) DK2379528T3 (ru)
DO (1) DOP2011000204A (ru)
EA (1) EA018808B1 (ru)
EC (1) ECSP11011157A (ru)
ES (1) ES2435798T3 (ru)
FI (1) FIC20190008I1 (ru)
GT (1) GT201100181A (ru)
HN (1) HN2011001701A (ru)
HR (1) HRP20131051T1 (ru)
HU (1) HUS000509I2 (ru)
IL (1) IL213350A (ru)
JO (1) JO2885B1 (ru)
MA (1) MA32903B1 (ru)
MX (1) MX2011006757A (ru)
MY (1) MY150547A (ru)
NZ (1) NZ593114A (ru)
PA (1) PA8852901A1 (ru)
PE (1) PE20120107A1 (ru)
PL (1) PL2379528T3 (ru)
PT (1) PT2379528E (ru)
RS (1) RS53061B (ru)
SG (1) SG172331A1 (ru)
SI (1) SI2379528T1 (ru)
TN (1) TN2011000293A1 (ru)
TW (1) TWI429635B (ru)
UA (1) UA104603C2 (ru)
WO (1) WO2010075074A1 (ru)
ZA (1) ZA201104505B (ru)

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