TN2011000070A1 - Picolinamide derivatives as kinase inhibitors - Google Patents
Picolinamide derivatives as kinase inhibitorsInfo
- Publication number
- TN2011000070A1 TN2011000070A1 TN2011000070A TN2011000070A TN2011000070A1 TN 2011000070 A1 TN2011000070 A1 TN 2011000070A1 TN 2011000070 A TN2011000070 A TN 2011000070A TN 2011000070 A TN2011000070 A TN 2011000070A TN 2011000070 A1 TN2011000070 A1 TN 2011000070A1
- Authority
- TN
- Tunisia
- Prior art keywords
- kinase
- compositions
- compounds
- kinase inhibitors
- picolinamide
- Prior art date
Links
- IBBMAWULFFBRKK-UHFFFAOYSA-N picolinamide Chemical class NC(=O)C1=CC=CC=N1 IBBMAWULFFBRKK-UHFFFAOYSA-N 0.000 title abstract 2
- 229940043355 kinase inhibitor Drugs 0.000 title 1
- 239000003757 phosphotransferase inhibitor Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 abstract 3
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 2
- 208000005623 Carcinogenesis Diseases 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 108091000080 Phosphotransferase Proteins 0.000 abstract 1
- MTCFGRXMJLQNBG-UHFFFAOYSA-N Serine Natural products OCC(N)C(O)=O MTCFGRXMJLQNBG-UHFFFAOYSA-N 0.000 abstract 1
- AYFVYJQAPQTCCC-UHFFFAOYSA-N Threonine Natural products CC(O)C(N)C(O)=O AYFVYJQAPQTCCC-UHFFFAOYSA-N 0.000 abstract 1
- 239000004473 Threonine Substances 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 230000036952 cancer formation Effects 0.000 abstract 1
- 231100000504 carcinogenesis Toxicity 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000005764 inhibitory process Effects 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
- 102000020233 phosphotransferase Human genes 0.000 abstract 1
- 230000010469 pro-virus integration Effects 0.000 abstract 1
- 102000027426 receptor tyrosine kinases Human genes 0.000 abstract 1
- 108091008598 receptor tyrosine kinases Proteins 0.000 abstract 1
Landscapes
- Pyridine Compounds (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| PCT/EP2009/061205 WO2010026124A1 (fr) | 2008-09-02 | 2009-08-31 | Dérivés de picolinamide en tant qu’inhibiteurs de kinase |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| TN2011000070A1 true TN2011000070A1 (en) | 2012-09-05 |
Family
ID=55024382
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| TN2011000070A TN2011000070A1 (en) | 2009-08-31 | 2011-02-11 | Picolinamide derivatives as kinase inhibitors |
Country Status (1)
| Country | Link |
|---|---|
| TN (1) | TN2011000070A1 (fr) |
-
2011
- 2011-02-11 TN TN2011000070A patent/TN2011000070A1/fr unknown
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