NO20081531L - Substituerte benzimidazoler som kinaseinhibitorer - Google Patents
Substituerte benzimidazoler som kinaseinhibitorerInfo
- Publication number
- NO20081531L NO20081531L NO20081531A NO20081531A NO20081531L NO 20081531 L NO20081531 L NO 20081531L NO 20081531 A NO20081531 A NO 20081531A NO 20081531 A NO20081531 A NO 20081531A NO 20081531 L NO20081531 L NO 20081531L
- Authority
- NO
- Norway
- Prior art keywords
- kinase
- compositions
- compounds
- kinase inhibitors
- inhibiting
- Prior art date
Links
- 150000001556 benzimidazoles Chemical class 0.000 title 1
- 229940043355 kinase inhibitor Drugs 0.000 title 1
- 239000003757 phosphotransferase inhibitor Substances 0.000 title 1
- 239000000203 mixture Substances 0.000 abstract 3
- 108091000080 Phosphotransferase Proteins 0.000 abstract 2
- 150000001875 compounds Chemical class 0.000 abstract 2
- 230000000694 effects Effects 0.000 abstract 2
- 230000002401 inhibitory effect Effects 0.000 abstract 2
- 102000020233 phosphotransferase Human genes 0.000 abstract 2
- 102000027426 receptor tyrosine kinases Human genes 0.000 abstract 2
- 108091008598 receptor tyrosine kinases Proteins 0.000 abstract 2
- 208000005623 Carcinogenesis Diseases 0.000 abstract 1
- 101001059454 Homo sapiens Serine/threonine-protein kinase MARK2 Proteins 0.000 abstract 1
- 206010028980 Neoplasm Diseases 0.000 abstract 1
- 102100028904 Serine/threonine-protein kinase MARK2 Human genes 0.000 abstract 1
- 125000003785 benzimidazolyl group Chemical class N1=C(NC2=C1C=CC=C2)* 0.000 abstract 1
- 201000011510 cancer Diseases 0.000 abstract 1
- 230000036952 cancer formation Effects 0.000 abstract 1
- 231100000504 carcinogenesis Toxicity 0.000 abstract 1
- 239000003795 chemical substances by application Substances 0.000 abstract 1
- 208000037265 diseases, disorders, signs and symptoms Diseases 0.000 abstract 1
- 230000001404 mediated effect Effects 0.000 abstract 1
Landscapes
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
Nye substituerte benzimidazolforbindelser av formel (I), sammensetninger og fremgangsmåter for inhibering av kinaseaktivitet assosiert med tumorigenese i et humant individ eller dyreindivid er tilveiebrakt. I enkelte utførelsesformer er forbindelsene og sammensetningene effektive til å inhibere aktiviteten av minst en serinAreoninkinase eller reseptortyrosinkinase. De nye forbindelsene og sammensetningene kan bli benyttet enten alene eller i kombinasjon med minst et ytterligere middel for behandlingen av en serin/treoninkinase eller reseptortyrosinkinasemediert lidelse, slik som cancer.
Applications Claiming Priority (5)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US71253905P | 2005-08-30 | 2005-08-30 | |
| US71310805P | 2005-08-30 | 2005-08-30 | |
| US71359105P | 2005-10-27 | 2005-10-27 | |
| US77468406P | 2006-02-17 | 2006-02-17 | |
| PCT/US2006/034088 WO2007030377A1 (en) | 2005-08-30 | 2006-08-30 | Substituted benzimidazoles as kinase inhibitors |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| NO20081531L true NO20081531L (no) | 2008-05-29 |
Family
ID=39937548
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| NO20081531A NO20081531L (no) | 2005-08-30 | 2008-03-28 | Substituerte benzimidazoler som kinaseinhibitorer |
Country Status (2)
| Country | Link |
|---|---|
| NO (1) | NO20081531L (no) |
| SV (1) | SV2008002831A (no) |
-
2008
- 2008-02-29 SV SV2008002831A patent/SV2008002831A/es unknown
- 2008-03-28 NO NO20081531A patent/NO20081531L/no not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| SV2008002831A (es) | 2010-01-12 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC2A | Withdrawal, rejection or dismissal of laid open patent application |