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SV2011004077A - Derivados aminobutiricos sustituidos como inhibidores de neprilisina - Google Patents

Derivados aminobutiricos sustituidos como inhibidores de neprilisina

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Publication number
SV2011004077A
SV2011004077A SV2011004077A SV2011004077A SV2011004077A SV 2011004077 A SV2011004077 A SV 2011004077A SV 2011004077 A SV2011004077 A SV 2011004077A SV 2011004077 A SV2011004077 A SV 2011004077A SV 2011004077 A SV2011004077 A SV 2011004077A
Authority
SV
El Salvador
Prior art keywords
neprilisine
aminobutiric
inhibitors
derivatives replaced
provides
Prior art date
Application number
SV2011004077A
Other languages
English (en)
Inventor
Gary Mark Coppola
Yuki Iwaki
Rajeshri Ganesh Karki
Toshio Kawanami
Gary Michael Ksander
Muneto Mogi
Robert Sun
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of SV2011004077A publication Critical patent/SV2011004077A/es

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Abstract

LA PRESENTE INVENCIÓN PROPORCIONA UN COMPUESTO DE LA FÓRMULA (I'): (VER FORMULA); O UNA SAL FARMACÉUTICAMENTE ACEPTABLE DEL MISMO, EN DONDE R1, R2, R3, X Y N SE DEFINEN EN LA PRESENTE. LA INVENCIÓN TAMBIÉN SE REFIERE A UN MÉTODO PARA LA ELABORACIÓN DE LOS COMPUESTOS DE LA INVENCIÓN, Y A SUS USOS TERAPÉUTICOS. LA PRESENTE INVENCIÓN PROPORCIONA ADEMÁS UNA COMBINACIÓN DE AGENTES FARMACOLÓGICAMENTE ACTIVOS Y UNA COMPOSICIÓN FARMACÉUTICA
SV2011004077A 2009-05-28 2011-11-28 Derivados aminobutiricos sustituidos como inhibidores de neprilisina SV2011004077A (es)

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