SK284813B6 - Peleta obsahujúca itrakonazol, spôsob jej prípravy a farmaceutická dávková forma s jej obsahom - Google Patents

Peleta obsahujúca itrakonazol, spôsob jej prípravy a farmaceutická dávková forma s jej obsahom Download PDF

Info

Publication number: SK284813B6
Authority: SK; Slovakia
Prior art keywords: itraconazole; coating; pellets; water; percent
Prior art date: 1997-03-26

Application number

SK544-99A

Other languages

English (en)

Slovak (sk)

Other versions

SK54499A3 (en

Inventor

Roger Petrus Gerebern Vandecruys

Cond� Valentin Florent Victor De

Paul Marie Victor Gilis

Jozef Peeters

Original Assignee

Janssen Pharmaceutica N. V.

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1997-03-26

Filing date

1998-03-18

Publication date

2005-12-01

1998-03-18 Application filed by Janssen Pharmaceutica N. V. filed Critical Janssen Pharmaceutica N. V.

2000-01-18 Publication of SK54499A3 publication Critical patent/SK54499A3/sk

2005-12-01 Publication of SK284813B6 publication Critical patent/SK284813B6/sk

Links

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Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/50—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals
- A61K9/5073—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings
- A61K9/5078—Microcapsules having a gas, liquid or semi-solid filling; Solid microparticles or pellets surrounded by a distinct coating layer, e.g. coated microspheres, coated drug crystals having two or more different coatings optionally including drug-containing subcoatings with drug-free core
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
- A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds

Landscapes

Health & Medical Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Engineering & Computer Science (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Medicinal Chemistry (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Pharmacology & Pharmacy (AREA)
Chemical & Material Sciences (AREA)
Animal Behavior & Ethology (AREA)
Epidemiology (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Dermatology (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Agricultural Chemicals And Associated Chemicals (AREA)

SK544-99A 1997-03-26 1998-03-18 Peleta obsahujúca itrakonazol, spôsob jej prípravy a farmaceutická dávková forma s jej obsahom SK284813B6 (sk)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
EP97200914		1997-03-26
PCT/EP1998/001773 WO1998042318A1 (en)	1997-03-26	1998-03-18	Pellets having a core coated with an antifungal and a polymer

Publications (2)

Publication Number	Publication Date
SK54499A3 SK54499A3 (en)	2000-01-18
SK284813B6 true SK284813B6 (sk)	2005-12-01

Family

ID=8228147

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
SK544-99A SK284813B6 (sk)	1997-03-26	1998-03-18	Peleta obsahujúca itrakonazol, spôsob jej prípravy a farmaceutická dávková forma s jej obsahom

Country Status (30)

Country	Link
EP (1)	EP0969821B1 (cs)
JP (1)	JP3608800B2 (cs)
KR (1)	KR100520936B1 (cs)
CN (1)	CN1206984C (cs)
AP (1)	AP1227A (cs)
AT (1)	ATE241969T1 (cs)
AU (1)	AU734248B2 (cs)
BG (1)	BG64434B1 (cs)
BR (1)	BR9806174A (cs)
CA (1)	CA2269501C (cs)
CY (1)	CY2384B1 (cs)
CZ (1)	CZ295502B6 (cs)
DE (1)	DE69815316T2 (cs)
DK (1)	DK0969821T3 (cs)
EE (1)	EE03904B1 (cs)
ES (1)	ES2201485T3 (cs)
HU (1)	HU224217B1 (cs)
ID (1)	ID21477A (cs)
IL (1)	IL129575A (cs)
NO (1)	NO325102B1 (cs)
NZ (1)	NZ335364A (cs)
OA (1)	OA11162A (cs)
PL (1)	PL190566B1 (cs)
PT (1)	PT969821E (cs)
RU (1)	RU2218153C2 (cs)
SI (1)	SI0969821T1 (cs)
SK (1)	SK284813B6 (cs)
TR (1)	TR199900990T2 (cs)
UA (1)	UA60318C2 (cs)
WO (1)	WO1998042318A1 (cs)

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ES2157731B1 (es) *	1998-07-21	2002-05-01	Liconsa Liberacion Controlada	Preparacion farmaceutica oral de un compuesto de actividad antifungica y procedimiento para su preparacion.
US6497905B1 (en)	1999-03-24	2002-12-24	R.P. Scherer Technologies, Inc.	Aqueous solubility pharmaceutical formulations
KR100432949B1 (ko) *	2000-06-13	2004-05-31	코오롱제약주식회사	생체이용율이 향상된 이트라코나졸의 분립체 조성물과이를 이용한 이트라코나졸 제제 및 그 제조방법
US6663897B2 (en) *	2001-02-06	2003-12-16	Dsm Ip Assets B.V.	Oral itraconazole formulations and methods of making the same
AU2002302363B2 (en)	2001-02-14	2008-05-01	Tibotec Pharmaceuticals Ltd.	Broadspectrum 2-(substituted-amino)-benzothiazole sulfonamide HIV protease inhibitors
MXPA03009179A (es)	2001-04-09	2004-11-22	Tibotec Pharm Ltd	2-(amino sustituido)-benzoxazol sunfonamidas, inhibidores de amplio espectro de la vih proteasa.
US7622490B2 (en)	2001-05-11	2009-11-24	Tibotec Pharmaceuticals, Ltd.	Broadspecturm 2-amino-benzoxazole sulfonamide HIV protease inhibitors
WO2002100407A1 (en) *	2001-06-12	2002-12-19	Smartrix Technologies Inc.	Itraconazole granulations: pharmaceutical formulations for oral administration and method of preparing same
US8071133B2 (en)	2001-08-20	2011-12-06	Stiefel Laboratories, Inc.	Oral dosage forms of water insoluble drugs and methods of making the same
CA2470964C (en)	2001-12-21	2013-07-02	Tibotec Pharmaceuticals Ltd.	Broadspectrum heterocyclic substituted phenyl containing sulfonamide hiv protease inhibitors
MY142238A (en)	2002-03-12	2010-11-15	Tibotec Pharm Ltd	Broadspectrum substituted benzimidazole sulfonamide hiv protease inhibitors
IL165043A0 (en)	2002-05-17	2005-12-18	Tibotec Pharm Ltd	broadspectrum substituted benzisoxazole sulfonamide hiv protease inhibitors
AP2126A (en)	2002-08-14	2010-06-03	Tibotec Pharm Ltd	Broadspectrum substituted oxindole sulfonamide HIVprotease inhibitors
KR100557680B1 (ko) *	2002-11-23	2006-03-07	한국유나이티드제약 주식회사	이트라코나졸의 용해도 개선을 위한 펠렛제제 및 그제조방법
PT1438961E (pt) *	2003-01-14	2007-05-31	Cimex Pharma Ag	Composição bioquivalente de itraconazol disperso num polímero hidrofílico.
DK1438960T4 (da) *	2003-01-14	2013-03-25	Cimex Pharma Ag	Sammensætning af itraconazol dispergeret i en hydrofil polymer med forhøjet biotilgængelighed
EP1651192A1 (en)	2003-08-06	2006-05-03	Nirmal Mulye	Pharmaceutical composition containing water soluble drug
SG145742A1 (en)	2003-09-11	2008-09-29	Tibotec Pharm Ltd	Entry inhibitors of the hiv virus
EP1568369A1 (en)	2004-02-23	2005-08-31	Boehringer Ingelheim Vetmedica Gmbh	Use of meloxicam for the treatment of respiratory diseases in pigs
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1998
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Also Published As

Publication number	Publication date
BR9806174A (pt)	1999-10-19
NZ335364A (en)	2000-08-25
HK1022840A1 (en)	2000-08-25
RU2218153C2 (ru)	2003-12-10
ID21477A (id)	1999-06-17
IL129575A0 (en)	2000-02-29
HU224217B1 (hu)	2005-06-28
BG103356A (en)	2000-03-31
NO992114L (no)	1999-08-26
PT969821E (pt)	2003-10-31
EP0969821A1 (en)	2000-01-12
AU734248B2 (en)	2001-06-07
WO1998042318A1 (en)	1998-10-01
AU7210798A (en)	1998-10-20
CN1244796A (zh)	2000-02-16
CY2384B1 (en)	2004-06-04
IL129575A (en)	2004-06-20
EE03904B1 (et)	2002-12-16
TR199900990T2 (xx)	1999-10-21
UA60318C2 (uk)	2003-10-15
CN1206984C (zh)	2005-06-22
SI0969821T1 (en)	2003-10-31
DE69815316D1 (de)	2003-07-10
CA2269501A1 (en)	1998-10-01
CZ295502B6 (cs)	2005-08-17
KR20000052971A (ko)	2000-08-25
JP2001520663A (ja)	2001-10-30
BG64434B1 (en)	2005-02-28
DE69815316T2 (de)	2004-04-29
EP0969821B1 (en)	2003-06-04
CA2269501C (en)	2005-11-08
PL190566B1 (pl)	2005-12-30
OA11162A (en)	2003-04-16
AP9901516A0 (en)	1999-06-30
JP3608800B2 (ja)	2005-01-12
KR100520936B1 (ko)	2005-10-17
NO992114D0 (no)	1999-04-30
EE9900453A (et)	2000-04-17
NO325102B1 (no)	2008-02-04
HUP0002056A3 (en)	2001-01-29
ATE241969T1 (de)	2003-06-15
HUP0002056A2 (hu)	2000-12-28
CZ139899A3 (cs)	1999-10-13
PL335542A1 (en)	2000-04-25
DK0969821T3 (da)	2003-09-15
AP1227A (en)	2003-11-24
SK54499A3 (en)	2000-01-18
ES2201485T3 (es)	2004-03-16

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RU2219909C2 (ru)	2003-12-27	Гранулы, имеющие ядро, покрытое противогрибковым препаратом и полимером
CZ293841B6 (cs)	2004-08-18	Částice s obsahem itrakonazolu
HU220614B1 (hu)	2002-03-28	Gombaellenes szerrel és polimerrel bevont magot tartalmazó mikrorészecskék, eljárás előállításukra és az azokat tartalmazó gyógyszerkészítmények
CN104010632B (zh)	2016-08-24	双层片剂形式的贝那普利和匹莫苯的固定剂量组合
SK15252000A3 (sk)	2001-10-08	Peleta, ktorej jadro je obalené činidlom znižujúcim lipidy a polymérom
MXPA99004411A (en)	1999-09-01	Pellets having a core coated with an antifungal and a polymer
HK1022840B (en)	2003-09-05	Pellets having a core coated with an antifungal and a polymer
MXPA00008322A (en)	2001-07-09	Pellets having a core coated with an antifungal and a polymer
MXPA00010649A (en)	2001-07-31	Pellets having a core coated with a lipid lowering agent and a polymer
CZ20003753A3 (cs)	2001-01-17	Peleta, jejíž jádro je potaženo činidlem snižujícím lipidy a polymerem

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