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SI3409274T1 - Režim odmerjanja za S1P receptor agonist - Google Patents

Režim odmerjanja za S1P receptor agonist

Info

Publication number
SI3409274T1
SI3409274T1 SI200932015T SI200932015T SI3409274T1 SI 3409274 T1 SI3409274 T1 SI 3409274T1 SI 200932015 T SI200932015 T SI 200932015T SI 200932015 T SI200932015 T SI 200932015T SI 3409274 T1 SI3409274 T1 SI 3409274T1
Authority
SI
Slovenia
Prior art keywords
receptor agonist
dosage regimen
regimen
dosage
agonist
Prior art date
Application number
SI200932015T
Other languages
English (en)
Inventor
Robert Schmouder
Thomas Dumortier
Olivier David
Michael Looby
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41667217&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI3409274(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of SI3409274T1 publication Critical patent/SI3409274T1/sl

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/661Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/10Phosphatides, e.g. lecithin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
SI200932015T 2008-12-22 2009-12-21 Režim odmerjanja za S1P receptor agonist SI3409274T1 (sl)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US13967208P 2008-12-22 2008-12-22
US21853009P 2009-06-19 2009-06-19
US24671509P 2009-09-29 2009-09-29
EP18179301.9A EP3409274B1 (en) 2008-12-22 2009-12-21 Dosage regimen for a s1p receptor agonist

Publications (1)

Publication Number Publication Date
SI3409274T1 true SI3409274T1 (sl) 2020-03-31

Family

ID=41667217

Family Applications (4)

Application Number Title Priority Date Filing Date
SI200932015T SI3409274T1 (sl) 2008-12-22 2009-12-21 Režim odmerjanja za S1P receptor agonist
SI200931311T SI2379067T1 (sl) 2008-12-22 2009-12-21 Režim odmerjanja fingolimoda za zdravljenje multiple skleroze
SI200932211T SI4098256T1 (sl) 2008-12-22 2009-12-21 Režim odmerjanja za agonist receptorja s1p
SI200932080T SI3453387T1 (sl) 2008-12-22 2009-12-21 Režim odmerjanja za agonist receptorja S1P

Family Applications After (3)

Application Number Title Priority Date Filing Date
SI200931311T SI2379067T1 (sl) 2008-12-22 2009-12-21 Režim odmerjanja fingolimoda za zdravljenje multiple skleroze
SI200932211T SI4098256T1 (sl) 2008-12-22 2009-12-21 Režim odmerjanja za agonist receptorja s1p
SI200932080T SI3453387T1 (sl) 2008-12-22 2009-12-21 Režim odmerjanja za agonist receptorja S1P

Country Status (43)

Country Link
US (12) US20100160259A1 (sl)
EP (7) EP3120844A1 (sl)
JP (7) JP2012513401A (sl)
KR (1) KR101347919B1 (sl)
CN (1) CN102264359A (sl)
AR (1) AR074826A1 (sl)
AU (1) AU2009330176C9 (sl)
BR (1) BRPI0923500A2 (sl)
CA (1) CA2747802C (sl)
CL (2) CL2011001529A1 (sl)
CO (1) CO6390117A2 (sl)
CR (1) CR20110274A (sl)
CU (1) CU20110136A7 (sl)
CY (4) CY1116990T1 (sl)
DK (4) DK3409274T3 (sl)
EA (1) EA201100978A1 (sl)
EC (1) ECSP11011222A (sl)
ES (4) ES3017254T3 (sl)
FI (2) FI4098256T3 (sl)
FR (2) FR20C1060I1 (sl)
HN (1) HN2011001759A (sl)
HR (4) HRP20151190T1 (sl)
HU (6) HUE048717T4 (sl)
IL (3) IL213170A0 (sl)
LT (5) LT3453387T (sl)
LU (1) LUC00183I2 (sl)
MA (1) MA32981B1 (sl)
ME (2) ME03594B (sl)
MX (3) MX2011006623A (sl)
NO (1) NO2020038I1 (sl)
NZ (1) NZ593065A (sl)
PE (1) PE20120337A1 (sl)
PL (4) PL3453387T3 (sl)
PT (4) PT3453387T (sl)
RS (3) RS66784B9 (sl)
SG (1) SG171404A1 (sl)
SI (4) SI3409274T1 (sl)
SM (2) SMT202000441T1 (sl)
TN (1) TN2011000272A1 (sl)
TW (1) TW201028143A (sl)
UY (1) UY32352A (sl)
WO (1) WO2010075239A1 (sl)
ZA (2) ZA201103863B (sl)

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HRP20151190T1 (hr) 2008-12-22 2016-01-01 Novartis Ag Režim doziranja za fingolimod u lijeäśenju multiple skleroze
US20120264719A1 (en) 2009-09-29 2012-10-18 Craig Boulton Dosage regimen of an s1p receptor modulator
US20110124605A1 (en) * 2009-11-20 2011-05-26 Shreeram Aradhye Use of an S1P Receptor Agonist
SG10201500639TA (en) 2010-01-27 2015-03-30 Arena Pharm Inc Processes for the preparation of (r)-2-(7-(4-cyclopentyl-3-(trifluoromethyl)benzyloxy)-1,2,3,4-tetrahydrocyclopenta[b]indol-3-yl)acetic acid and salts thereof
EP2566473B1 (en) * 2010-05-06 2016-01-06 Novartis AG Dosage regimen of diaryl sulfide derivatives
EP2455080A1 (en) * 2010-11-23 2012-05-23 Almirall, S.A. S1P1 receptor agonists for use in the treatment of multiple sclerosis
FR2968556B1 (fr) 2010-12-13 2013-12-27 Centre Nat Rech Scient Inhibiteurs des infections a vih et leurs utilisations
BR112013017302B1 (pt) 2011-01-07 2021-12-07 Novartis Ag Composição farmacêutica em fase sólida
JP6133790B2 (ja) 2011-02-18 2017-05-24 ザ スクリプス リサーチ インスティテュート ミエリン形成細胞運命へのオリゴデンドロサイト前駆細胞の定方向分化
JO3177B1 (ar) 2011-04-01 2018-03-08 Novartis Ag تركيبات تتالف من 2-أمينو-2- [ 2- ( 4- أكتيل فينيل ) إثيل ] بروبان - 3, 1- ديول
US9592268B2 (en) 2011-05-23 2017-03-14 Cornell University Endothelium protective materials and methods of use
TW201320994A (zh) 2011-10-11 2013-06-01 Novartis Ag 投藥療程
SI2885266T1 (sl) 2012-08-17 2020-10-30 Actelion Pharmaceuticals Ltd Postopek za pripravo (2Z,5Z)-5-(3-kloro-4-((R)-2,3-dihidroksipropoksi) benziliden)-2-(propilimino)-3-(O-tolil)tiazolidin-4-on in v omenjenem postopku uporabljena vmesna spojina
EP2964249A1 (en) * 2013-03-06 2016-01-13 Acorda Therapeutics, Inc. Therapeutic dosing of a neuregulin or a fragment thereof for treatment or prophylaxis of heart failure
US10675254B2 (en) 2013-10-11 2020-06-09 Teikoku Seiyaku Co., Ltd. Sphingosine-1-phosphate receptor agonist iontophoretic devices and methods of using the same
WO2015053878A1 (en) 2013-10-11 2015-04-16 Teikoku Pharma Usa, Inc. Topical sphingosine-1-phosphate receptor agonist formulations and methods of using the same
US20170027907A1 (en) * 2014-04-10 2017-02-02 Eric Legangneux Sip modulator immediate release dosage regimen
WO2016091996A1 (en) 2014-12-11 2016-06-16 Actelion Pharmaceuticals Ltd Dosing regimen for a selective s1p1 receptor agonist
MA41139A (fr) 2014-12-11 2017-10-17 Actelion Pharmaceuticals Ltd Combinaison pharmaceutique comportant un agoniste sélectif du récepteur sip1
ES2995737T3 (en) * 2015-01-06 2025-02-11 Arena Pharm Inc Compound for use in treating conditions related to the s1p1 receptor
US20180042895A1 (en) 2015-02-26 2018-02-15 Novartis Ag Treatment of autoimmune disease in a patient receiving additionally a beta-blocker
MA42807A (fr) 2015-06-22 2018-07-25 Arena Pharm Inc Sel l-arginine cristallin d'acide (r)-2-(7-(4-cyclopentyl-3-(trifluorométhyl)benzyloxy)-1,2,3,4-tétrahydrocyclo-penta[b]indol-3-yl)acétique (composé 1) pour une utilisation dans des troubles associés au récepteur de s1p1
WO2018151873A1 (en) 2017-02-16 2018-08-23 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of primary biliary cholangitis
CA3053416A1 (en) 2017-02-16 2018-08-23 Arena Pharmaceuticals, Inc. Compounds and methods for treatment of inflammatory bowel disease with extra-intestinal manifestations
EP3801459B1 (en) 2018-06-06 2024-08-07 Arena Pharmaceuticals, Inc. Methods of treating conditions related to the s1p1 receptor
PH12022551043A1 (en) 2019-10-31 2023-05-03 Idorsia Pharmaceuticals Ltd Combination of a cxcr7 antagonist with an s1p1 receptor modulator
US11135197B2 (en) 2020-02-07 2021-10-05 Argentum Pharmaceuticals Llc Dosage regimen of an S1P receptor modulator
WO2021158848A1 (en) * 2020-02-07 2021-08-12 Argentum Pharmaceuticals Llc Dosage regimen of an s1p receptor agonist
JP2023515612A (ja) * 2020-02-28 2023-04-13 アカール・ファーマ・プロプライエタリー・リミテッド S1p受容体調節物質
CN113332435B (zh) * 2021-06-18 2022-10-18 广州中医药大学(广州中医药研究院) 鞘氨醇-1-磷酸4受体激动剂及其与真武汤联合在制备治疗慢性肾小球肾炎药物中的应用

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KR101718639B1 (ko) 2008-03-17 2017-03-21 액테리온 파마슈티칼 리미티드 선별적 s1p₁ 수용체 작동약에 대한 투약 섭생
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JP5657565B2 (ja) 2008-12-22 2015-01-21 ノバルティス アーゲー S1p受容体アゴニストの投与レジメン

Also Published As

Publication number Publication date
ES2552823T3 (es) 2015-12-02
RS60666B1 (sr) 2020-09-30
HUE052048T2 (hu) 2021-04-28
MX385959B (es) 2025-03-18
CL2013001558A1 (es) 2013-10-25
JP2016135752A (ja) 2016-07-28
FIC20253002I1 (fi) 2025-05-23
LTPA2025520I1 (sl) 2025-06-25
CR20110274A (es) 2011-07-19
CA2747802C (en) 2021-02-09
HN2011001759A (es) 2013-11-26
EP3409274B1 (en) 2019-11-20
JP2014144970A (ja) 2014-08-14
PE20120337A1 (es) 2012-04-24
ME03594B (me) 2020-07-20
SI4098256T1 (sl) 2025-06-30
CN102264359A (zh) 2011-11-30
ZA201103863B (en) 2012-10-31
CY2020036I1 (el) 2021-03-12
AU2009330176A1 (en) 2011-07-07
EP3409274A1 (en) 2018-12-05
SG171404A1 (en) 2011-07-28
PL2379067T3 (pl) 2016-02-29
JP2019167360A (ja) 2019-10-03
EP3120844A1 (en) 2017-01-25
PL3453387T3 (pl) 2020-11-02
ME03802B (me) 2021-04-20
US20170189353A1 (en) 2017-07-06
AU2009330176C9 (en) 2017-01-05
EP3677260A1 (en) 2020-07-08
RS59857B1 (sr) 2020-02-28
HRP20151190T1 (hr) 2016-01-01
LT3453387T (lt) 2020-08-25
EP2907511A1 (en) 2015-08-19
JP2022103194A (ja) 2022-07-07
US20100160259A1 (en) 2010-06-24
US20160081949A1 (en) 2016-03-24
CL2011001529A1 (es) 2012-02-24
SMT202000054T1 (it) 2020-03-13
EP4098256A1 (en) 2022-12-07
MA32981B1 (fr) 2012-01-02
JP2012513401A (ja) 2012-06-14
PT3409274T (pt) 2019-12-17
EP3453387B1 (en) 2020-06-03
JP7329965B2 (ja) 2023-08-21
TW201028143A (en) 2010-08-01
PL3409274T3 (pl) 2020-06-01
HUS2000046I1 (hu) 2020-12-28
KR101347919B1 (ko) 2014-01-07
HRP20192175T1 (hr) 2020-03-20
JP2024129030A (ja) 2024-09-26
LT4098256T (lt) 2025-06-10
US20140066657A1 (en) 2014-03-06
SI2379067T1 (sl) 2016-01-29
EP4098256B1 (en) 2025-02-26
HUE071189T2 (hu) 2025-08-28
IL274756A (en) 2020-07-30
NO2020038I1 (no) 2020-11-18
AU2009330176C1 (en) 2016-12-08
US20110257133A1 (en) 2011-10-20
KR20110096175A (ko) 2011-08-29
LUC00183I2 (sl) 2024-07-01
ZA201205942B (en) 2013-03-27
ES3017254T3 (en) 2025-05-12
SI3453387T1 (sl) 2020-10-30
US20190091180A1 (en) 2019-03-28
PL4098256T3 (pl) 2025-06-09
US20140148415A1 (en) 2014-05-29
AU2009330176B2 (en) 2014-03-06
DK3453387T3 (da) 2020-08-10
DK4098256T3 (da) 2025-04-22
FR20C1060I1 (fr) 2020-12-25
EP2379067B1 (en) 2015-09-02
CA2747802A1 (en) 2010-07-01
SMT202000441T1 (it) 2020-09-10
EP2379067A1 (en) 2011-10-26
DK3409274T3 (da) 2019-12-16
IL278914A (en) 2021-01-31
ES2810823T3 (es) 2021-03-09
FR25C1012I1 (fr) 2025-06-13
PT3453387T (pt) 2020-08-11
CY2020036I2 (el) 2021-06-25
TN2011000272A1 (en) 2012-12-17
FI4098256T3 (fi) 2025-03-31
MX2021010759A (es) 2022-07-19
PT2379067E (pt) 2015-12-23
WO2010075239A1 (en) 2010-07-01
HRP20250568T1 (hr) 2025-07-04
EP4098256B9 (en) 2025-06-18
HUE026869T2 (en) 2016-08-29
ECSP11011222A (es) 2011-08-31
PT4098256T (pt) 2025-04-10
CY1123255T1 (el) 2021-10-29
US20250262171A1 (en) 2025-08-21
CU20110136A7 (es) 2012-01-31
HUE048717T2 (hu) 2020-08-28
ES2760607T3 (es) 2020-05-14
DK2379067T3 (en) 2015-12-07
MX2011006623A (es) 2011-07-12
RS66784B9 (sr) 2025-08-29
CY1122812T1 (el) 2021-05-05
HRP20201167T1 (hr) 2020-12-11
LT3409274T (lt) 2020-02-10
US20220142949A1 (en) 2022-05-12
JP2017141238A (ja) 2017-08-17
CO6390117A2 (es) 2012-02-29
IL213170A0 (en) 2011-07-31
DK4098256T5 (da) 2025-07-21
HUE048717T4 (hu) 2022-02-28
US20180289638A1 (en) 2018-10-11
US20200330407A1 (en) 2020-10-22
BRPI0923500A2 (pt) 2018-05-29
US20160263061A1 (en) 2016-09-15
CY1116990T1 (el) 2017-04-05
EA201100978A1 (ru) 2012-01-30
LTPA2020005I1 (lt) 2020-12-10
UY32352A (es) 2010-07-30
NZ593065A (en) 2012-11-30
EP3453387A1 (en) 2019-03-13
AR074826A1 (es) 2011-02-16
HUS2500026I1 (hu) 2025-07-28
RS66784B1 (sr) 2025-06-30

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