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CU20110136A7 - Régimen de dosificación para un agonista de los receptores de s1p - Google Patents

Régimen de dosificación para un agonista de los receptores de s1p

Info

Publication number
CU20110136A7
CU20110136A7 CU20110136A CU20110136A CU20110136A7 CU 20110136 A7 CU20110136 A7 CU 20110136A7 CU 20110136 A CU20110136 A CU 20110136A CU 20110136 A CU20110136 A CU 20110136A CU 20110136 A7 CU20110136 A7 CU 20110136A7
Authority
CU
Cuba
Prior art keywords
dosage regime
receiver agonist
agonist
receiver
dosage
Prior art date
Application number
CU20110136A
Other languages
English (en)
Inventor
Michael Looby
Olivier David
Thomas Dumortier
Robert Schmouder
Original Assignee
Novartis Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=41667217&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=CU20110136(A7) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Novartis Ag filed Critical Novartis Ag
Publication of CU20110136A7 publication Critical patent/CU20110136A7/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/137Arylalkylamines, e.g. amphetamine, epinephrine, salbutamol, ephedrine or methadone
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/13Amines
    • A61K31/135Amines having aromatic rings, e.g. ketamine, nortriptyline
    • A61K31/138Aryloxyalkylamines, e.g. propranolol, tamoxifen, phenoxybenzamine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/66Phosphorus compounds
    • A61K31/661Phosphorus acids or esters thereof not having P—C bonds, e.g. fosfosal, dichlorvos, malathion or mevinphos
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • A61P37/02Immunomodulators
    • A61P37/06Immunosuppressants, e.g. drugs for graft rejection
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07FACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02Phosphorus compounds
    • C07F9/06Phosphorus compounds without P—C bonds
    • C07F9/08Esters of oxyacids of phosphorus
    • C07F9/09Esters of phosphoric acids
    • C07F9/10Phosphatides, e.g. lecithin

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Immunology (AREA)
  • Organic Chemistry (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Emergency Medicine (AREA)
  • Transplantation (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Los moduladores o agonistas de los receptores de S1P se administran siguiendo un régimen de dosificación en donde, durante los días iniciales del tratamiento, la dosificación diaria es más baja que la dosificación diaria convencional.
CU20110136A 2008-12-22 2011-06-22 Régimen de dosificación para un agonista de los receptores de s1p CU20110136A7 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US13967208P 2008-12-22 2008-12-22
US21853009P 2009-06-19 2009-06-19
US24671509P 2009-09-29 2009-09-29

Publications (1)

Publication Number Publication Date
CU20110136A7 true CU20110136A7 (es) 2012-01-31

Family

ID=41667217

Family Applications (1)

Application Number Title Priority Date Filing Date
CU20110136A CU20110136A7 (es) 2008-12-22 2011-06-22 Régimen de dosificación para un agonista de los receptores de s1p

Country Status (43)

Country Link
US (12) US20100160259A1 (es)
EP (7) EP3120844A1 (es)
JP (7) JP2012513401A (es)
KR (1) KR101347919B1 (es)
CN (1) CN102264359A (es)
AR (1) AR074826A1 (es)
AU (1) AU2009330176C9 (es)
BR (1) BRPI0923500A2 (es)
CA (1) CA2747802C (es)
CL (2) CL2011001529A1 (es)
CO (1) CO6390117A2 (es)
CR (1) CR20110274A (es)
CU (1) CU20110136A7 (es)
CY (4) CY1116990T1 (es)
DK (4) DK3409274T3 (es)
EA (1) EA201100978A1 (es)
EC (1) ECSP11011222A (es)
ES (4) ES3017254T3 (es)
FI (2) FI4098256T3 (es)
FR (2) FR20C1060I1 (es)
HN (1) HN2011001759A (es)
HR (4) HRP20151190T1 (es)
HU (6) HUE048717T4 (es)
IL (3) IL213170A0 (es)
LT (5) LT3453387T (es)
LU (1) LUC00183I2 (es)
MA (1) MA32981B1 (es)
ME (2) ME03594B (es)
MX (3) MX2011006623A (es)
NO (1) NO2020038I1 (es)
NZ (1) NZ593065A (es)
PE (1) PE20120337A1 (es)
PL (4) PL3453387T3 (es)
PT (4) PT3453387T (es)
RS (3) RS66784B9 (es)
SG (1) SG171404A1 (es)
SI (4) SI3409274T1 (es)
SM (2) SMT202000441T1 (es)
TN (1) TN2011000272A1 (es)
TW (1) TW201028143A (es)
UY (1) UY32352A (es)
WO (1) WO2010075239A1 (es)
ZA (2) ZA201103863B (es)

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WO2016091996A1 (en) 2014-12-11 2016-06-16 Actelion Pharmaceuticals Ltd Dosing regimen for a selective s1p1 receptor agonist
MA41139A (fr) 2014-12-11 2017-10-17 Actelion Pharmaceuticals Ltd Combinaison pharmaceutique comportant un agoniste sélectif du récepteur sip1
ES2995737T3 (en) * 2015-01-06 2025-02-11 Arena Pharm Inc Compound for use in treating conditions related to the s1p1 receptor
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MA42807A (fr) 2015-06-22 2018-07-25 Arena Pharm Inc Sel l-arginine cristallin d'acide (r)-2-(7-(4-cyclopentyl-3-(trifluorométhyl)benzyloxy)-1,2,3,4-tétrahydrocyclo-penta[b]indol-3-yl)acétique (composé 1) pour une utilisation dans des troubles associés au récepteur de s1p1
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ES2552823T3 (es) 2015-12-02
RS60666B1 (sr) 2020-09-30
HUE052048T2 (hu) 2021-04-28
MX385959B (es) 2025-03-18
CL2013001558A1 (es) 2013-10-25
JP2016135752A (ja) 2016-07-28
FIC20253002I1 (fi) 2025-05-23
LTPA2025520I1 (es) 2025-06-25
CR20110274A (es) 2011-07-19
CA2747802C (en) 2021-02-09
HN2011001759A (es) 2013-11-26
EP3409274B1 (en) 2019-11-20
JP2014144970A (ja) 2014-08-14
PE20120337A1 (es) 2012-04-24
ME03594B (me) 2020-07-20
SI4098256T1 (sl) 2025-06-30
CN102264359A (zh) 2011-11-30
ZA201103863B (en) 2012-10-31
CY2020036I1 (el) 2021-03-12
AU2009330176A1 (en) 2011-07-07
EP3409274A1 (en) 2018-12-05
SG171404A1 (en) 2011-07-28
PL2379067T3 (pl) 2016-02-29
JP2019167360A (ja) 2019-10-03
EP3120844A1 (en) 2017-01-25
PL3453387T3 (pl) 2020-11-02
ME03802B (me) 2021-04-20
US20170189353A1 (en) 2017-07-06
AU2009330176C9 (en) 2017-01-05
EP3677260A1 (en) 2020-07-08
RS59857B1 (sr) 2020-02-28
HRP20151190T1 (hr) 2016-01-01
LT3453387T (lt) 2020-08-25
EP2907511A1 (en) 2015-08-19
JP2022103194A (ja) 2022-07-07
US20100160259A1 (en) 2010-06-24
US20160081949A1 (en) 2016-03-24
CL2011001529A1 (es) 2012-02-24
SMT202000054T1 (it) 2020-03-13
EP4098256A1 (en) 2022-12-07
MA32981B1 (fr) 2012-01-02
JP2012513401A (ja) 2012-06-14
PT3409274T (pt) 2019-12-17
EP3453387B1 (en) 2020-06-03
JP7329965B2 (ja) 2023-08-21
TW201028143A (en) 2010-08-01
PL3409274T3 (pl) 2020-06-01
HUS2000046I1 (hu) 2020-12-28
KR101347919B1 (ko) 2014-01-07
HRP20192175T1 (hr) 2020-03-20
JP2024129030A (ja) 2024-09-26
LT4098256T (lt) 2025-06-10
US20140066657A1 (en) 2014-03-06
SI2379067T1 (sl) 2016-01-29
EP4098256B1 (en) 2025-02-26
HUE071189T2 (hu) 2025-08-28
IL274756A (en) 2020-07-30
NO2020038I1 (no) 2020-11-18
AU2009330176C1 (en) 2016-12-08
US20110257133A1 (en) 2011-10-20
KR20110096175A (ko) 2011-08-29
LUC00183I2 (es) 2024-07-01
ZA201205942B (en) 2013-03-27
ES3017254T3 (en) 2025-05-12
SI3453387T1 (sl) 2020-10-30
US20190091180A1 (en) 2019-03-28
PL4098256T3 (pl) 2025-06-09
US20140148415A1 (en) 2014-05-29
AU2009330176B2 (en) 2014-03-06
DK3453387T3 (da) 2020-08-10
DK4098256T3 (da) 2025-04-22
FR20C1060I1 (fr) 2020-12-25
EP2379067B1 (en) 2015-09-02
CA2747802A1 (en) 2010-07-01
SMT202000441T1 (it) 2020-09-10
EP2379067A1 (en) 2011-10-26
DK3409274T3 (da) 2019-12-16
IL278914A (en) 2021-01-31
ES2810823T3 (es) 2021-03-09
FR25C1012I1 (fr) 2025-06-13
PT3453387T (pt) 2020-08-11
CY2020036I2 (el) 2021-06-25
TN2011000272A1 (en) 2012-12-17
FI4098256T3 (fi) 2025-03-31
MX2021010759A (es) 2022-07-19
PT2379067E (pt) 2015-12-23
WO2010075239A1 (en) 2010-07-01
HRP20250568T1 (hr) 2025-07-04
EP4098256B9 (en) 2025-06-18
HUE026869T2 (en) 2016-08-29
ECSP11011222A (es) 2011-08-31
PT4098256T (pt) 2025-04-10
CY1123255T1 (el) 2021-10-29
US20250262171A1 (en) 2025-08-21
HUE048717T2 (hu) 2020-08-28
SI3409274T1 (sl) 2020-03-31
ES2760607T3 (es) 2020-05-14
DK2379067T3 (en) 2015-12-07
MX2011006623A (es) 2011-07-12
RS66784B9 (sr) 2025-08-29
CY1122812T1 (el) 2021-05-05
HRP20201167T1 (hr) 2020-12-11
LT3409274T (lt) 2020-02-10
US20220142949A1 (en) 2022-05-12
JP2017141238A (ja) 2017-08-17
CO6390117A2 (es) 2012-02-29
IL213170A0 (en) 2011-07-31
DK4098256T5 (da) 2025-07-21
HUE048717T4 (hu) 2022-02-28
US20180289638A1 (en) 2018-10-11
US20200330407A1 (en) 2020-10-22
BRPI0923500A2 (pt) 2018-05-29
US20160263061A1 (en) 2016-09-15
CY1116990T1 (el) 2017-04-05
EA201100978A1 (ru) 2012-01-30
LTPA2020005I1 (lt) 2020-12-10
UY32352A (es) 2010-07-30
NZ593065A (en) 2012-11-30
EP3453387A1 (en) 2019-03-13
AR074826A1 (es) 2011-02-16
HUS2500026I1 (hu) 2025-07-28
RS66784B1 (sr) 2025-06-30

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