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SI0922040T1 - Process for preparing intermediates to florfenicol - Google Patents

Process for preparing intermediates to florfenicol

Info

Publication number
SI0922040T1
SI0922040T1 SI9730688T SI9730688T SI0922040T1 SI 0922040 T1 SI0922040 T1 SI 0922040T1 SI 9730688 T SI9730688 T SI 9730688T SI 9730688 T SI9730688 T SI 9730688T SI 0922040 T1 SI0922040 T1 SI 0922040T1
Authority
SI
Slovenia
Prior art keywords
florfenicol
preparing intermediates
intermediates
preparing
Prior art date
Application number
SI9730688T
Other languages
English (en)
Slovenian (sl)
Inventor
James C. Towson
Dhiru B. Vashi
Original Assignee
Schering Corporation
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=24808601&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=SI0922040(T1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Schering Corporation filed Critical Schering Corporation
Publication of SI0922040T1 publication Critical patent/SI0922040T1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
    • C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
    • C07D263/08—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D263/16—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D263/28—Nitrogen atoms not forming part of a nitro radical

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
SI9730688T 1996-08-19 1997-08-18 Process for preparing intermediates to florfenicol SI0922040T1 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US08/699,271 US5663361A (en) 1996-08-19 1996-08-19 Process for preparing intermediates to florfenicol
PCT/US1997/014205 WO1998007709A1 (fr) 1996-08-19 1997-08-18 Procede de preparation d'intermediaires du florfenicol
EP97938263.7A EP0922040B2 (fr) 1996-08-19 1997-08-18 Procede de preparation d'intermediaires du florfenicol

Publications (1)

Publication Number Publication Date
SI0922040T1 true SI0922040T1 (en) 2005-02-28

Family

ID=24808601

Family Applications (1)

Application Number Title Priority Date Filing Date
SI9730688T SI0922040T1 (en) 1996-08-19 1997-08-18 Process for preparing intermediates to florfenicol

Country Status (30)

Country Link
US (1) US5663361A (fr)
EP (1) EP0922040B2 (fr)
JP (1) JP3274868B2 (fr)
KR (1) KR100286851B1 (fr)
CN (1) CN1097583C (fr)
AR (1) AR008298A1 (fr)
AT (1) ATE283847T1 (fr)
AU (1) AU714495B2 (fr)
BR (1) BR9711318B1 (fr)
CA (1) CA2264116C (fr)
CO (1) CO4560550A1 (fr)
CZ (1) CZ297915B6 (fr)
DE (1) DE69731835T3 (fr)
DK (1) DK0922040T3 (fr)
ES (1) ES2234026T5 (fr)
HU (1) HU229610B1 (fr)
ID (1) ID18047A (fr)
IL (1) IL128574A (fr)
MY (1) MY115679A (fr)
NO (1) NO312962B1 (fr)
NZ (1) NZ334111A (fr)
PE (1) PE99798A1 (fr)
PL (2) PL196454B1 (fr)
PT (1) PT922040E (fr)
SI (1) SI0922040T1 (fr)
SK (1) SK286124B6 (fr)
TR (2) TR199900354T2 (fr)
TW (1) TW381075B (fr)
WO (1) WO1998007709A1 (fr)
ZA (1) ZA977406B (fr)

Families Citing this family (40)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CN1173933C (zh) * 2001-06-01 2004-11-03 中国科学院上海有机化学研究所 一种从l型取代苯丝氨酸酯制备d－（－）－苏式1－r－取代苯基－2－二氯乙酰氨基－3－氟－1－丙醇的方法
KR20040091698A (ko) * 2002-03-08 2004-10-28 쉐링-플라우 리미티드. 신규한 플로르페니콜형 항생제
PE20050386A1 (es) 2003-05-29 2005-06-23 Schering Plough Ltd Composiciones farmaceuticas de florfenicol
US7439268B2 (en) * 2003-07-18 2008-10-21 Idexx Laboratories Compositions containing prodrugs of florfenicol and methods of use
US20050049210A1 (en) * 2003-08-27 2005-03-03 Idexx Laboratories, Inc. Methods for the controlled delivery of pharmacologically active compounds
US7126005B2 (en) * 2003-10-06 2006-10-24 Aurobindo Pharma Limited Process for preparing florfenicol
CA2576589C (fr) * 2004-08-13 2013-11-12 Schering-Plough Ltd. Formulation pharmaceutique comprenant un antibiotique, un triazole et un corticosteroide
AR054981A1 (es) 2004-09-23 2007-08-01 Schering Plough Ltd Control de parasitos en animales mediante el uso de nuevos derivados de trifluorometansulfonanilida oxima eter
DE602005017419D1 (de) * 2004-11-19 2009-12-10 Schering Plough Ltd Kontrolle von parasiten bei tieren mittels verwendung von parasitiziden 2-phenyl-3-(1h-pyrrol-2-yl) acrylonitril-derivaten
ES2315942T3 (es) * 2004-12-21 2009-04-01 Intervet International Bv Composicion veterinaria inyectable que contiene florfenicol.
CA2609574A1 (fr) * 2005-06-09 2006-12-21 Schering-Plough Ltd. Controle de parasites chez des animaux a l'aide de derives de n-[(phenyloxy)phenyl]-1,1,1-trifluoromethanesulfonamide et de n-[(phenylsulfanyl)phenyl]-1,1,1-trifluoromethanesulfonamide
EP1928820B1 (fr) * 2005-09-07 2014-01-29 Intervet International BV Procede de preparation de composes d'ester oxazolidine et leur conversion en florfenicol
US8119667B2 (en) * 2005-12-29 2012-02-21 Schering-Plough Animal Health Corporation Carbonates of fenicol antibiotics
US7518017B2 (en) 2006-02-17 2009-04-14 Idexx Laboratories Fenicol compounds and methods synthesizing 2-trifluoroacetamido-3-substituted propiophenone compounds
US20070238700A1 (en) * 2006-04-10 2007-10-11 Winzenberg Kevin N N-phenyl-1,1,1-trifluoromethanesulfonamide hydrazone derivative compounds and their usage in controlling parasites
WO2008076259A1 (fr) * 2006-12-13 2008-06-26 Schering-Plough Ltd. Promédicaments de florfenicol solubles dans l'eau et analogues
MX2009006467A (es) * 2006-12-13 2009-08-21 Schering Plough Ltd Profarmacos solubles en agua de cloranfenicol, tiamfenicol y analogos de los mismos.
JP2010525059A (ja) * 2007-04-27 2010-07-22 シェーリング−プラウ・リミテッド シクロデキストリンを用いてフロルフェニコールおよび構造的に関連する抗生物質の溶解度を高めるための化合物および方法
MX2009013016A (es) * 2007-05-30 2010-02-17 Schering Plough Ltd Un procedimiento para preparar compuestos de aminodiol oxazolina-protegidos utiles como intermediarios para florfenicol.
TWI430995B (zh) 2007-06-26 2014-03-21 Du Pont 萘異唑啉無脊椎有害動物控制劑
JP6006471B2 (ja) 2007-06-27 2016-10-12 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニーＥ．Ｉ．Ｄｕ Ｐｏｎｔ Ｄｅ Ｎｅｍｏｕｒｓ Ａｎｄ Ｃｏｍｐａｎｙ 動物有害生物の防除方法
WO2009015111A2 (fr) * 2007-07-25 2009-01-29 Intervet Intermatonal B.V. Procédé pour préparer des aminodiols d'oxazolidine et d'oxazolidinone
US7550625B2 (en) * 2007-10-19 2009-06-23 Idexx Laboratories Esters of florfenicol
CA2705063C (fr) * 2007-11-09 2013-02-05 Intervet International B.V. Formulation solide a liberation rapide, sa preparation et son utilisation
TWI468407B (zh) 2008-02-06 2015-01-11 Du Pont 中離子農藥
CA2732017A1 (fr) * 2008-07-30 2010-02-04 Intervet International B.V. Procede de preparation de composes aminodiol d'oxazoline proteges  utiles comme produits intermediaires dans la production de florfenicol
JP2013501059A (ja) 2009-08-05 2013-01-10 イー・アイ・デュポン・ドウ・ヌムール・アンド・カンパニー メソイオン性殺虫剤
UA107804C2 (en) 2009-08-05 2015-02-25 Du Pont Mixtures of pesticides mezoionnyh
UA110924C2 (uk) 2009-08-05 2016-03-10 Е. І. Дю Пон Де Немур Енд Компані Мезоіонні пестициди
BR112012002524A2 (pt) 2009-08-05 2019-09-24 Du Pont "composto de fórmula, composição, composição para proteger um animal de uma praga parasítica de invertebrados, métodos para controlar uma praga invertebrada e semente tratada"
BRPI1002023A2 (pt) 2010-03-01 2011-10-25 Nanocore Biotecnologia S A forma farmacêutica sólida de dissolução rápida para tratamento de infecções bacterianas
KR20130124458A (ko) 2010-05-27 2013-11-14 이 아이 듀폰 디 네모아 앤드 캄파니 4-[5-[3-클로로-5-(트라이플루오로메틸)페닐]-4,5-다이하이드로-5-(트라이플루오로메틸)-3-아이속사졸릴]-n-[2-옥소-2-[(2,2,2-트라이플루오로에틸)아미노]에틸]-1-나프탈렌카르복스아미드의 결정 형태
WO2012087630A1 (fr) 2010-12-20 2012-06-28 E.I. Du Pont De Nemours And Company Composés de pyridine et de pyrimidine utilisés pour lutter contre des nuisibles invertébrés
WO2013158422A1 (fr) 2012-04-17 2013-10-24 E. I. Du Pont De Nemours And Company Composés hétérocycliques pour la lutte contre des animaux nuisibles invertébrés
CN102911133B (zh) * 2012-10-31 2014-07-02 绍兴民生医药有限公司 (4r,5r)-2-二氯甲基-4,5-二氢-5-(4-甲砜基苯基)-4-恶唑甲醇的纯化方法
CN103254147B (zh) * 2013-04-19 2016-04-06 浙江科技学院 一种d-苏式-2-(二氯甲基)-4,5-二氢-5-[对-（甲砜基）苯基]-4-噁唑甲醇的制备方法
CN106278964B (zh) * 2016-07-31 2018-01-16 浙江润康药业有限公司 氟苯尼考的制备方法
CN106631872A (zh) * 2016-12-13 2017-05-10 浙江普洛家园药业有限公司 一种氟苯尼考类似物中间体的合成方法
CN110272856B (zh) * 2019-05-08 2022-05-03 江南大学 一种表达d-苏氨酸醛缩酶的重组菌及其构建方法与应用
CN117466787B (zh) * 2023-12-28 2024-03-22 山东国邦药业有限公司 一种氟苯尼考中间体的制备方法

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US2759001A (en) * 1952-03-01 1956-08-14 Parke Davis & Co Process for the production of delta2-oxazolines
US4361557A (en) * 1980-01-28 1982-11-30 Schering Corporation 1-Aryl-2-acylamido-3-fluoro-1-propanol acylates, methods for their use as anti-bacterial agents and compositions useful therefor
EP0678506A3 (fr) * 1983-06-02 1996-07-24 Zambon Spa Intermédiaires pour la préparation des dérivés de 1-phényl-1-hydroxy-2-amino-3-fluoropropane.
US4876352A (en) * 1988-09-14 1989-10-24 Schering Corporation Pressurized fluorination of hydroxy alkyl groups
WO1990014434A1 (fr) † 1989-05-15 1990-11-29 Schering Corporation Procede de preparation de composes antibacteriens et intermediaires
ES2067958T3 (es) * 1990-10-25 1995-04-01 Schering Corp Procedimiento para preparar florfenicol, sus analogos y productos intermedios de la oxazolina para dicho procedimiento.

Also Published As

Publication number Publication date
HK1017890A1 (en) 1999-12-03
AU714495B2 (en) 2000-01-06
CA2264116A1 (fr) 1998-02-26
CZ54099A3 (cs) 1999-07-14
SK286124B6 (sk) 2008-04-07
MY115679A (en) 2003-08-30
PL196454B1 (pl) 2008-01-31
US5663361A (en) 1997-09-02
AR008298A1 (es) 1999-12-29
BR9711318A (pt) 1999-08-17
KR20000068178A (ko) 2000-11-25
DK0922040T3 (da) 2005-04-04
PL331644A1 (en) 1999-08-02
DE69731835D1 (de) 2005-01-05
SK19999A3 (en) 2000-02-14
ES2234026T3 (es) 2005-06-16
TR199900354T2 (xx) 1999-05-21
PL198553B1 (pl) 2008-06-30
NO312962B1 (no) 2002-07-22
WO1998007709A1 (fr) 1998-02-26
ZA977406B (en) 1998-02-18
JP2000501424A (ja) 2000-02-08
NO990756L (no) 1999-02-18
DE69731835T3 (de) 2013-12-05
BR9711318B1 (pt) 2009-01-13
CN1233244A (zh) 1999-10-27
EP0922040A1 (fr) 1999-06-16
NZ334111A (en) 1999-10-28
JP3274868B2 (ja) 2002-04-15
ATE283847T1 (de) 2004-12-15
ID18047A (id) 1998-02-19
CO4560550A1 (es) 1998-02-10
HUP9904166A2 (hu) 2000-05-28
PE99798A1 (es) 1998-12-28
EP0922040B2 (fr) 2013-07-17
CA2264116C (fr) 2002-07-02
NO990756D0 (no) 1999-02-18
AU4063897A (en) 1998-03-06
TR200800474T2 (tr) 2008-04-21
HU229610B1 (en) 2014-03-28
DE69731835T2 (de) 2005-07-21
EP0922040B1 (fr) 2004-12-01
KR100286851B1 (ko) 2001-04-16
CN1097583C (zh) 2003-01-01
PT922040E (pt) 2005-02-28
IL128574A (en) 2002-04-21
HUP9904166A3 (en) 2001-11-28
ES2234026T5 (es) 2013-11-12
IL128574A0 (en) 2000-01-31
CZ297915B6 (cs) 2007-04-25
TW381075B (en) 2000-02-01

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