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SG146694A1 - 1,1,1-trifluoro-4-phenyl-4-methyl-2-(1h-pyrrolo-2,3-c pyridin-2- ylmethyl)pentan-2-ol derivatives and related compounds as glucocorticoid ligands for the treatment of inflammatory diseases and diabetes - Google Patents

1,1,1-trifluoro-4-phenyl-4-methyl-2-(1h-pyrrolo-2,3-c pyridin-2- ylmethyl)pentan-2-ol derivatives and related compounds as glucocorticoid ligands for the treatment of inflammatory diseases and diabetes

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Publication number
SG146694A1
SG146694A1 SG200807363-7A SG2008073637A SG146694A1 SG 146694 A1 SG146694 A1 SG 146694A1 SG 2008073637 A SG2008073637 A SG 2008073637A SG 146694 A1 SG146694 A1 SG 146694A1
Authority
SG
Singapore
Prior art keywords
pentan
pyrrolo
ylmethyl
trifluoro
pyridin
Prior art date
Application number
SG200807363-7A
Other languages
English (en)
Inventor
Younes Bekkali
Rajashekhar Betageri
Michael J Emmanuel
Abdelhakim Hammach
Christian H J J Harcken
Thomas Martin Kirrane
Daniel Kuzmich
Thomas Wai-Ho Lee
Pingrong Liu
Usha R Patel
Hossein Razavi
Doris Riether
Hidenori Takahashi
David S Thomson
Ji Wang
Renee Zindell
John Robert Proudfoot
Original Assignee
Boehringer Ingelheim Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Pharma filed Critical Boehringer Ingelheim Pharma
Publication of SG146694A1 publication Critical patent/SG146694A1/en

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    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
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