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RU2019108189A3 - - Google Patents

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Publication number
RU2019108189A3
RU2019108189A3 RU2019108189A RU2019108189A RU2019108189A3 RU 2019108189 A3 RU2019108189 A3 RU 2019108189A3 RU 2019108189 A RU2019108189 A RU 2019108189A RU 2019108189 A RU2019108189 A RU 2019108189A RU 2019108189 A3 RU2019108189 A3 RU 2019108189A3
Authority
RU
Russia
Application number
RU2019108189A
Other versions
RU2743126C2 (ru
RU2743126C9 (ru
RU2019108189A (ru
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed filed Critical
Publication of RU2019108189A3 publication Critical patent/RU2019108189A3/ru
Publication of RU2019108189A publication Critical patent/RU2019108189A/ru
Publication of RU2743126C2 publication Critical patent/RU2743126C2/ru
Application granted granted Critical
Publication of RU2743126C9 publication Critical patent/RU2743126C9/ru

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Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D498/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D498/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and oxygen atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D498/04Ortho-condensed systems

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Plural Heterocyclic Compounds (AREA)
RU2019108189A 2016-08-22 2017-08-22 Ингибитор pde4 RU2743126C9 (ru)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
CN201610700714 2016-08-22
CN201610700714.2 2016-08-22
PCT/CN2017/098461 WO2018036469A1 (zh) 2016-08-22 2017-08-22 Pde4抑制剂

Publications (4)

Publication Number Publication Date
RU2019108189A3 true RU2019108189A3 (ru) 2020-09-22
RU2019108189A RU2019108189A (ru) 2020-09-22
RU2743126C2 RU2743126C2 (ru) 2021-02-15
RU2743126C9 RU2743126C9 (ru) 2021-04-27

Family

ID=61246401

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2019108189A RU2743126C9 (ru) 2016-08-22 2017-08-22 Ингибитор pde4

Country Status (9)

Country Link
US (1) US10662189B2 (ru)
EP (1) EP3502111B1 (ru)
JP (1) JP7029444B2 (ru)
CN (1) CN109661395B (ru)
AU (1) AU2017317123B9 (ru)
CA (1) CA3034785C (ru)
RU (1) RU2743126C9 (ru)
WO (1) WO2018036469A1 (ru)
ZA (1) ZA201901773B (ru)

Families Citing this family (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP3747884B1 (en) * 2018-01-29 2022-11-02 Medshine Discovery Inc. Crystal form of 1h-imidazo[4,5-b]pyridine-2(3h)-one compound and preparation method therefor
BR112021004730A2 (pt) * 2018-09-13 2021-06-01 Kissei Pharmaceutical Co., Ltd. composto de imidazopiridinona
CN115397819A (zh) * 2020-02-24 2022-11-25 苏州隆博泰药业有限公司 Pde4抑制剂化合物及其医药用途
JP7504822B2 (ja) * 2020-03-12 2024-06-24 キッセイ薬品工業株式会社 イミダゾピリジノン化合物を含む医薬組成物
CN112876403B (zh) * 2021-01-27 2022-10-21 成都摩尔生物医药有限公司 一种阿普斯特杂质的制备方法
EP4326713A4 (en) * 2021-04-12 2025-03-19 Impact Therapeutics (Shanghai), Inc. Substituted fused bicyclic compounds as parp inhibitors and the use thereof
CN119161297A (zh) * 2024-09-18 2024-12-20 浙江工业大学 一种4-溴-6-氯烟酸甲酯的制备方法

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US6667316B1 (en) * 1999-11-12 2003-12-23 Celgene Corporation Pharmaceutically active isoindoline derivatives
BRPI0519030A2 (pt) 2004-12-13 2008-12-23 Celgene Corp mÉtodos de tratamento, prevenÇço, ou controle de inflamaÇço das vias aÉreas e de uma doenÇa ou distérbio das vias aÉreas ou pulmonar, e, composiÇço farmacÊutica
ES2347172T3 (es) 2005-02-16 2010-10-26 Astrazeneca Ab Compuestos quimicos.
CN101119996A (zh) * 2005-02-16 2008-02-06 阿斯利康(瑞典)有限公司 化学化合物
GB0525143D0 (en) * 2005-12-09 2006-01-18 Novartis Ag Organic compounds
MX2009004077A (es) 2006-10-19 2009-05-05 Signal Pharm Llc Compuestos de heteroarilo, composiciones de los mismos, y su uso como inhibidores de proteina cinasas.
JP5662319B2 (ja) * 2008-09-09 2015-01-28 ベーリンガー インゲルハイム インターナショナル ゲゼルシャフト ミット ベシュレンクテル ハフツング アザ−ベンゾイミダゾロンキマーゼ阻害剤
WO2011021678A1 (ja) 2009-08-21 2011-02-24 武田薬品工業株式会社 縮合複素環化合物
WO2015175956A1 (en) * 2014-05-16 2015-11-19 Celgene Corporation Compositions and methods for the treatment of atherosclerotic cardiovascular diseases with pde4 modulators

Also Published As

Publication number Publication date
EP3502111B1 (en) 2022-07-27
EP3502111A1 (en) 2019-06-26
US10662189B2 (en) 2020-05-26
ZA201901773B (en) 2021-08-25
JP7029444B2 (ja) 2022-04-07
AU2017317123B9 (en) 2021-11-25
AU2017317123A1 (en) 2019-04-11
CN109661395B (zh) 2020-09-01
EP3502111A4 (en) 2020-05-20
WO2018036469A1 (zh) 2018-03-01
CA3034785C (en) 2022-11-15
AU2017317123B2 (en) 2021-07-29
CA3034785A1 (en) 2018-03-01
RU2743126C2 (ru) 2021-02-15
US20190177318A1 (en) 2019-06-13
RU2743126C9 (ru) 2021-04-27
RU2019108189A (ru) 2020-09-22
JP2019528298A (ja) 2019-10-10
CN109661395A (zh) 2019-04-19

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Legal Events

Date Code Title Description
TH4A Reissue of patent specification
PC41 Official registration of the transfer of exclusive right

Effective date: 20210830