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RU2006119294A - Фармацевтические составы с улучшенными фармацевтическими свойствами, содержащие вкусовые вещества - Google Patents

Фармацевтические составы с улучшенными фармацевтическими свойствами, содержащие вкусовые вещества Download PDF

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Publication number
RU2006119294A
RU2006119294A RU2006119294/15A RU2006119294A RU2006119294A RU 2006119294 A RU2006119294 A RU 2006119294A RU 2006119294/15 A RU2006119294/15 A RU 2006119294/15A RU 2006119294 A RU2006119294 A RU 2006119294A RU 2006119294 A RU2006119294 A RU 2006119294A
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RU
Russia
Prior art keywords
pharmaceutical composition
pharmaceutical
salt
pradofloxacin
enrofloxacin
Prior art date
Application number
RU2006119294/15A
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English (en)
Other versions
RU2377018C2 (ru
Inventor
Патрик БОШЕ (DE)
Патрик Боше
Сабине БОНГЕРТС (DE)
Сабине БОНГЕРТС
Венката-Рангарао КАНИКАНТИ (DE)
Венката-Рангарао КАНИКАНТИ
Original Assignee
Байер ХельсКер АГ (DE)
Байер ХельсКер АГ
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Байер ХельсКер АГ (DE), Байер ХельсКер АГ filed Critical Байер ХельсКер АГ (DE)
Publication of RU2006119294A publication Critical patent/RU2006119294A/ru
Application granted granted Critical
Publication of RU2377018C2 publication Critical patent/RU2377018C2/ru

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K33/00—Medicinal preparations containing inorganic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2059—Starch, including chemically or physically modified derivatives; Amylose; Amylopectin; Dextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2068—Compounds of unknown constitution, e.g. material from plants or animals
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2013—Organic compounds, e.g. phospholipids, fats
    • A61K9/2018—Sugars, or sugar alcohols, e.g. lactose, mannitol; Derivatives thereof, e.g. polysorbates

Landscapes

  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Chemistry (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Zoology (AREA)
  • Nutrition Science (AREA)
  • Physiology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Oncology (AREA)
  • General Chemical & Material Sciences (AREA)
  • Communicable Diseases (AREA)
  • Organic Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Molecular Biology (AREA)
  • Biophysics (AREA)
  • Botany (AREA)
  • Inorganic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Quinoline Compounds (AREA)

Claims (4)

1. Твердый фармацевтический состав, содержащий фармацевтическое действующее вещество, ароматическое вещество и по меньшей мере 1,5 мас.% высокодисперсного диоксида кремния в пересчете на общую массу готового фармацевтического состава.
2. Твердый фармацевтический состав по п.1, содержащий в качестве фармацевтического действующего вещества энрофлоксацин, соль энрофлоксацина или гидрат энрофлоксацина или его соль.
3. Твердый фармацевтический состав по п.1, содержащий в качестве фармацевтического действующего вещества прадофлоксацин, соль прадофлоксацина или гидрат прадофлоксацина или его соль.
4. Способ получения твердого фармацевтического состава по п.1, состоящий в том, что вкусовое вещество гранулируют с высокодисперсным оксидом кремния, а также одним или несколькими действующими веществами и обычными фармацевтическими добавками и/или вспомогательными веществами.
RU2006119294/15A 2003-11-04 2004-10-30 Фармацевтические составы с улучшенными фармацевтическими свойствами, содержащие вкусовые вещества RU2377018C2 (ru)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10351448.1 2003-11-04
DE10351448A DE10351448A1 (de) 2003-11-04 2003-11-04 Geschmackstoffhaltige Arzneimittelformulierungen mit verbesserten pharmazeutischen Eigenschaften

Publications (2)

Publication Number Publication Date
RU2006119294A true RU2006119294A (ru) 2007-12-27
RU2377018C2 RU2377018C2 (ru) 2009-12-27

Family

ID=34559323

Family Applications (1)

Application Number Title Priority Date Filing Date
RU2006119294/15A RU2377018C2 (ru) 2003-11-04 2004-10-30 Фармацевтические составы с улучшенными фармацевтическими свойствами, содержащие вкусовые вещества

Country Status (30)

Country Link
US (2) US7858120B2 (ru)
EP (2) EP2080515A1 (ru)
JP (1) JP4892351B2 (ru)
KR (2) KR101325146B1 (ru)
CN (2) CN102335117A (ru)
AR (2) AR046226A1 (ru)
AT (1) ATE454891T1 (ru)
AU (1) AU2004286785B2 (ru)
BR (1) BRPI0416188A (ru)
CA (1) CA2544344C (ru)
CR (1) CR8371A (ru)
CY (2) CY1110541T1 (ru)
DE (2) DE10351448A1 (ru)
DK (1) DK1682144T3 (ru)
ES (1) ES2337793T3 (ru)
HR (1) HRP20100189T1 (ru)
IL (1) IL175147A (ru)
LU (1) LU91882I2 (ru)
MY (1) MY149864A (ru)
NO (1) NO339326B1 (ru)
NZ (1) NZ546921A (ru)
PE (1) PE20050575A1 (ru)
PL (1) PL1682144T3 (ru)
PT (1) PT1682144E (ru)
RU (1) RU2377018C2 (ru)
SI (1) SI1682144T1 (ru)
TW (1) TWI343819B (ru)
UA (1) UA85691C2 (ru)
WO (1) WO2005044271A1 (ru)
ZA (1) ZA200603451B (ru)

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Also Published As

Publication number Publication date
IL175147A0 (en) 2008-04-13
CY2011017I1 (el) 2016-12-14
SI1682144T1 (sl) 2010-05-31
CA2544344C (en) 2013-10-15
ATE454891T1 (de) 2010-01-15
HRP20100189T1 (hr) 2010-05-31
NZ546921A (en) 2009-08-28
RU2377018C2 (ru) 2009-12-27
JP4892351B2 (ja) 2012-03-07
JP2007510001A (ja) 2007-04-19
TW200517144A (en) 2005-06-01
CN102335117A (zh) 2012-02-01
WO2005044271A1 (de) 2005-05-19
NO339326B1 (no) 2016-11-28
AU2004286785B2 (en) 2010-08-12
DE10351448A1 (de) 2005-06-09
PT1682144E (pt) 2010-03-09
AR108594A2 (es) 2018-09-05
ES2337793T3 (es) 2010-04-29
IL175147A (en) 2014-04-30
US20110065719A1 (en) 2011-03-17
PL1682144T3 (pl) 2010-06-30
CR8371A (es) 2006-10-10
KR101325146B1 (ko) 2013-11-07
KR20060109910A (ko) 2006-10-23
CY1110541T1 (el) 2015-04-29
EP1682144B1 (de) 2010-01-13
HK1107008A1 (en) 2008-03-28
DE502004010644D1 (de) 2010-03-04
US20070196466A1 (en) 2007-08-23
ZA200603451B (en) 2007-07-25
UA85691C2 (ru) 2009-02-25
AU2004286785A8 (en) 2009-08-13
EP2080515A1 (de) 2009-07-22
MY149864A (en) 2013-10-31
CY2011017I2 (el) 2016-12-14
CA2544344A1 (en) 2005-05-19
DK1682144T3 (da) 2010-05-17
NO20062605L (no) 2006-07-25
LU91882I2 (fr) 2013-04-12
AR046226A1 (es) 2005-11-30
KR20120093299A (ko) 2012-08-22
AU2004286785A1 (en) 2005-05-19
EP1682144A1 (de) 2006-07-26
PE20050575A1 (es) 2005-10-27
US7858120B2 (en) 2010-12-28
CN1972687A (zh) 2007-05-30
TWI343819B (en) 2011-06-21
CN1972687B (zh) 2013-01-23
BRPI0416188A (pt) 2007-01-23

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