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PE20070950A1 - Sales de adicion de acido de n-{3-[4-(2-metoxifenil)-1-piperazinil]-propil}-7-oxo-5-trifluormetil-7h-tieno[3,2-b]piran-3-carboxamida - Google Patents

Sales de adicion de acido de n-{3-[4-(2-metoxifenil)-1-piperazinil]-propil}-7-oxo-5-trifluormetil-7h-tieno[3,2-b]piran-3-carboxamida

Info

Publication number
PE20070950A1
PE20070950A1 PE2007000119A PE2007000119A PE20070950A1 PE 20070950 A1 PE20070950 A1 PE 20070950A1 PE 2007000119 A PE2007000119 A PE 2007000119A PE 2007000119 A PE2007000119 A PE 2007000119A PE 20070950 A1 PE20070950 A1 PE 20070950A1
Authority
PE
Peru
Prior art keywords
metoxifenil
piperazinil
oxo
propyl
salts
Prior art date
Application number
PE2007000119A
Other languages
English (en)
Inventor
Amedeo Leonardi
Gianni Motta
Original Assignee
Recordati Ireland Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Recordati Ireland Ltd filed Critical Recordati Ireland Ltd
Publication of PE20070950A1 publication Critical patent/PE20070950A1/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/02—Drugs for disorders of the urinary system of urine or of the urinary tract, e.g. urine acidifiers
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00—Drugs for disorders of the urinary system
    • A61P13/08—Drugs for disorders of the urinary system of the prostate
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/06—Antianaemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system

Landscapes

  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Urology & Nephrology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

SE REFIERE A SALES DE ADICION DE N-{3-[4-(2-METOXIFENIL)-1-PIPERAZINIL]-PROPIL}-7-OXO-5-TRIFLUORMETIL-7H-TIENO[3,2-b]PIRAN-3-CARBOXAMIDA (COMPUESTO A) CON ACIDOS INORGANICOS TAL COMO EL ACIDO CLORHIDRICO O BROMHIDRICO, ACIDOS SULFONICOS TAL COMO EL ACIDO METANSULFONICO, BENCENSULFONICO, TOLUENSULFONICO O NAFTALEN-1,5-DISULFONICO, O ACIDO CARBOXILICO. SIENDO UNA SAL PREFERIDA LA FORMA CRISTALINA DEL MESILATO DE N-{3-[4-(2-METOXIFENIL)-1-PIPERAZINIL]-PROPIL}-7-OXO-5-TRIFLUORMETIL-7H-TIENO[3,2-b]PIRAN-3-CARBOXAMIDA CUYOS PICOS DEL PATRON DE DIFRACCION DE POLVO DE RAYOS X EXPRESADO EN GRADOS 2 SON 10,97; 14,67; 15,73; 16,49; 18,75; 20,76; 22,07; 22,73; 24,35; 26,65 Y 27,74. SE REFIERE TAMBIEN A UNA COMPOSICION FARMACEUTICA. DICHAS SALES DE ADICION DEL COMPUESTO A SON UTILES PARA EL TRATAMIENTO DE SINDROMES OBSTRUCTIVOS DEL TRACTO URINARIO INFERIOR TAL COMO HIPERTROFIA PROSTATICA BENIGNA
PE2007000119A 2006-02-03 2007-02-02 Sales de adicion de acido de n-{3-[4-(2-metoxifenil)-1-piperazinil]-propil}-7-oxo-5-trifluormetil-7h-tieno[3,2-b]piran-3-carboxamida PE20070950A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76482406P 2006-02-03 2006-02-03

Publications (1)

Publication Number Publication Date
PE20070950A1 true PE20070950A1 (es) 2007-09-10

Family

ID=37983328

Family Applications (1)

Application Number Title Priority Date Filing Date
PE2007000119A PE20070950A1 (es) 2006-02-03 2007-02-02 Sales de adicion de acido de n-{3-[4-(2-metoxifenil)-1-piperazinil]-propil}-7-oxo-5-trifluormetil-7h-tieno[3,2-b]piran-3-carboxamida

Country Status (6)

Country Link
US (1) US20070185129A1 (es)
AR (1) AR059302A1 (es)
PE (1) PE20070950A1 (es)
TW (1) TW200804395A (es)
UY (1) UY30111A1 (es)
WO (1) WO2007088063A1 (es)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8557807B2 (en) * 2008-01-24 2013-10-15 Signal Rx Pharmaceuticals, Inc. Thienopyranones as kinase inhibitors

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1313581B1 (it) * 1999-07-30 2002-09-09 Recordati Chem Pharm Derivati tienopirancarbossamidici.
US6387909B1 (en) * 1999-07-30 2002-05-14 Recordati S.A. Chemical And Pharmaceutical Company Thienopyranecarboxamide derivatives
US6306861B1 (en) * 1999-07-30 2001-10-23 Recordati S.A. Chemical And Pharmaceutical Company Thienopyrancecarboxamide derivatives
TWI265925B (en) * 1999-10-11 2006-11-11 Pfizer Pyrazolo[4,3-d]pyrimidin-7-ones useful in inhibiting type 5 cyclic guanosine 3',5'-monophosphate phosphodiesterases(cGMP PDE5), process and intermediates for their preparation, their uses and composition comprising them
ITMI20010164A1 (it) * 2001-01-30 2002-07-30 Recordati Chem Pharm Alfa 1 antagonisti selettivi a + d
US6992192B2 (en) * 2001-06-05 2006-01-31 Lilly Icos Llc. Carboline derivatives as PDE5 inhibitors

Also Published As

Publication number Publication date
US20070185129A1 (en) 2007-08-09
AR059302A1 (es) 2008-03-26
UY30111A1 (es) 2007-04-30
TW200804395A (en) 2008-01-16
WO2007088063A1 (en) 2007-08-09

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