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LV11182A - Jauni eritromicina atvasinajumi to iegusanas metode un to izmantosana medicina - Google Patents

Jauni eritromicina atvasinajumi to iegusanas metode un to izmantosana medicina

Info

Publication number
LV11182A
LV11182A LV950363A LV950363A LV11182A LV 11182 A LV11182 A LV 11182A LV 950363 A LV950363 A LV 950363A LV 950363 A LV950363 A LV 950363A LV 11182 A LV11182 A LV 11182A
Authority
LV
Latvia
Prior art keywords
medicine
obtaining
erythromycin derivatives
new erythromycin
new
Prior art date
Application number
LV950363A
Other languages
English (en)
Other versions
LV11182B (en
Inventor
Constantin Agouridas
Yannick Benedetti
Jean-Francois Chantot
Alexis Denis
Odile Le Martret
Original Assignee
Roussel Uclaf
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Roussel Uclaf filed Critical Roussel Uclaf
Publication of LV11182A publication Critical patent/LV11182A/lv
Publication of LV11182B publication Critical patent/LV11182B/lv

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08Hetero rings containing eight or more ring members, e.g. erythromycins
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07HSUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Biotechnology (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Communicable Diseases (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
LVP-95-363A 1994-04-08 1995-01-05 Novel erythromycin derivates, method for preparing same and use thereof as drugs LV11182B (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9404154A FR2718450B1 (fr) 1994-04-08 1994-04-08 Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
PCT/FR1995/000441 WO1995027720A1 (fr) 1994-04-08 1995-04-06 Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments

Publications (2)

Publication Number Publication Date
LV11182A true LV11182A (lv) 1996-04-20
LV11182B LV11182B (en) 1997-04-20

Family

ID=9461886

Family Applications (1)

Application Number Title Priority Date Filing Date
LVP-95-363A LV11182B (en) 1994-04-08 1995-01-05 Novel erythromycin derivates, method for preparing same and use thereof as drugs

Country Status (49)

Country Link
US (2) US5656607A (lv)
EP (1) EP0676409B1 (lv)
JP (1) JP3000023B2 (lv)
KR (1) KR100317148B1 (lv)
CN (1) CN1059445C (lv)
AP (1) AP587A (lv)
AT (1) ATE234853T1 (lv)
AU (1) AU684939B2 (lv)
BG (1) BG61916B1 (lv)
BR (1) BR9506147A (lv)
CA (1) CA2164638C (lv)
CO (1) CO4370097A1 (lv)
CZ (1) CZ296005B6 (lv)
DE (1) DE69529934T2 (lv)
DK (1) DK0676409T3 (lv)
DZ (1) DZ1869A1 (lv)
EE (1) EE04498B1 (lv)
ES (1) ES2189820T3 (lv)
FI (1) FI111264B (lv)
FR (1) FR2718450B1 (lv)
GB (1) GB2288174A (lv)
GE (1) GEP19991836B (lv)
HR (1) HRP950217B1 (lv)
HU (1) HU215396B (lv)
IL (1) IL112954A (lv)
IS (1) IS1865B (lv)
JO (1) JO1850B1 (lv)
LV (1) LV11182B (lv)
MA (1) MA23501A1 (lv)
MD (1) MD663G2 (lv)
MY (1) MY114672A (lv)
NO (1) NO308361B1 (lv)
NZ (1) NZ284498A (lv)
OA (1) OA10200A (lv)
PE (1) PE2896A1 (lv)
PL (1) PL180837B1 (lv)
PT (1) PT676409E (lv)
RO (1) RO115634B1 (lv)
RU (1) RU2141965C1 (lv)
SA (1) SA97170757A (lv)
SI (1) SI0676409T1 (lv)
SK (1) SK284079B6 (lv)
SV (1) SV1995000018A (lv)
TN (1) TNSN95026A1 (lv)
TW (1) TW316908B (lv)
UA (1) UA44705C2 (lv)
WO (1) WO1995027720A1 (lv)
YU (1) YU49221B (lv)
ZA (1) ZA952059B (lv)

Families Citing this family (50)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2732023B1 (fr) * 1995-03-22 1997-04-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2742757B1 (fr) * 1995-12-22 1998-01-30 Roussel Uclaf Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2745289B1 (fr) * 1996-02-28 1998-05-29 Roussel Uclaf Nouveaux derives de l'acide 1(2h) quinoleine carboxylique, leur procede de preparation et leur application a la synthese de produits doues de proprietes antibiotiques
US5750510A (en) * 1997-04-04 1998-05-12 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
AU710532B2 (en) * 1996-05-07 1999-09-23 Abbott Laboratories 3-descladinose-2,3-anhydroerythromycin derivatives
FR2748746B1 (fr) * 1996-05-14 1998-08-14 Hoechst Marion Roussel Inc Nouveau procede d'isomerisation du radical methyle en 10 de derives de l'erythromycine
FR2751656B1 (fr) * 1996-07-24 1998-10-16 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
UA51730C2 (uk) * 1996-09-04 2002-12-16 Ебботт Лабораторіз 6-o-заміщені кетоліди з антибактеріальною активністю, спосіб їх одержання (варіанти), фармацевтична композиція та спосіб регулювання бактеріальної інфекції у ссавців
DE69733723T2 (de) * 1996-09-04 2006-04-20 Abbott Laboratories, Abbott Park 6-o-Substituierte Ketoliden mit antibakteriellen Wirkung
FR2757168B1 (fr) * 1996-12-12 1999-06-11 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
FR2760017B1 (fr) * 1997-02-27 1999-04-30 Hoechst Marion Roussel Inc Nouveaux derives de l'erytromycine, leur procede de preparation et leur application comme medicaments
US6165986A (en) * 1997-03-10 2000-12-26 Taisho Pharmaceutical Co., Ltd. Erythromycin a derivatives
US6140479A (en) * 1997-03-24 2000-10-31 Taisho Pharmaceuticals Co., Ltd. Erythromycin a derivatives
WO1998051696A1 (en) * 1997-05-09 1998-11-19 Pfizer Products Inc. Erythromycin derivatives
US5922683A (en) * 1997-05-29 1999-07-13 Abbott Laboratories Multicyclic erythromycin derivatives
TR199902995T2 (xx) * 1997-06-11 2000-02-21 Pfizer Products Inc. 9-Oksim eritromisin t�revleri
FR2771008B1 (fr) * 1997-11-17 2000-04-28 Hoechst Marion Roussel Inc Utilisation des ketolides pour la preparation de compositions pharmaceutiques destinees a prevenir les complications thrombotiques arterielles liees a l'atherosclerose
AP1060A (en) * 1998-01-02 2002-04-23 Pfizer Prod Inc Novel erythromycin derivatives.
HRP980189B1 (en) * 1998-04-06 2004-04-30 Pliva Pharm & Chem Works Novel 15-membered lactams ketolides
ES2243066T3 (es) 1998-09-22 2005-11-16 Pfizer Products Inc. Antibioticos de carbamato y carbazato cetolida.
FR2786188B1 (fr) * 1998-11-24 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
WO2000034297A1 (en) 1998-12-10 2000-06-15 Pfizer Products Inc. Carbamate and carbazate ketolide antibiotics
EP1749832A3 (en) * 1998-12-10 2008-03-26 Pfizer Products Incorporated Carbamate and carbazate ketolide antibiotics
EP1298138B1 (en) * 1998-12-10 2006-11-02 Pfizer Products Inc. Carbamate and Carbazate Ketolide Antibiotics
FR2789392B1 (fr) 1999-02-04 2001-10-05 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur application comme medicaments
US6054435A (en) * 1999-03-19 2000-04-25 Abbott Laboratories 6-O-substituted macrolides having antibacterial activity
KR20020007374A (ko) * 1999-04-16 2002-01-26 추후제출 매크롤라이드 항감염제
US6590083B1 (en) 1999-04-16 2003-07-08 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
US6399582B1 (en) 1999-04-16 2002-06-04 Ortho-Mcneil Pharmaceutical, Inc. Ketolide antibacterials
IL145739A0 (en) * 1999-05-24 2002-07-25 Pfizer Prod Inc 13-methyl-erythromycin derivatives
EP1404693A2 (en) * 2001-07-03 2004-04-07 Chiron Corporation C12 modified erythromycin macrolides and ketolides having antibacterial activity
MXPA04012978A (es) 2002-07-01 2005-09-12 Arkion Life Sciences Llc D B A Proceso y material para la produccion de glucosamina y n-acetilglucosamina.
EP3738591A3 (en) 2003-03-10 2021-03-24 Merck Sharp & Dohme Corp. Novel antibacterial agents
EP1618120A2 (en) * 2003-04-25 2006-01-25 Chiron Corporation Novel ketolide derivatives
EP1618119A2 (en) * 2003-04-25 2006-01-25 Chiron Corporation Pyridyl substituted ketolide antibiotics
AU2008316830B2 (en) 2007-10-25 2016-03-17 Cempra Pharmaceuticals, Inc. Process for the preparation of macrolide antibacterial agents
US9072759B2 (en) 2008-10-24 2015-07-07 Cempra Pharmaceuticals, Inc. Biodefenses using triazole-containing macrolides
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
ES2608285T3 (es) 2009-09-10 2017-04-07 Cempra Pharmaceuticals, Inc. Procedimientos para el tratamiento de paludismo, tuberculosis y enfermedades por MAC
ES2564097T3 (es) 2010-03-22 2016-03-17 Cempra Pharmaceuticals, Inc. Formas cristalinas de un macrólido, y usos de las mismas
ES2636948T3 (es) 2010-05-20 2017-10-10 Cempra Pharmaceuticals, Inc. Procesos para preparar macrólidos y cetólidos e intermediarios para los mismos
WO2012034058A1 (en) 2010-09-10 2012-03-15 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
IN2014DN08939A (lv) 2012-03-27 2015-05-22 Cempra Pharmaceuticals Inc
CN105163785A (zh) 2013-03-14 2015-12-16 森普拉制药公司 用于治疗呼吸道疾病的方法及其制剂
RU2015138797A (ru) 2013-03-15 2017-04-24 Семпра Фармасьютикалс, Инк. Конвергентные способы получения макролидных антибактериальных агентов
MX377459B (es) 2013-04-04 2025-03-10 Harvard College Macrolidos y metodos para su preparacion y uso.
WO2016057798A1 (en) 2014-10-08 2016-04-14 President And Fellows Of Harvard College 14-membered ketolides and methods of their preparation and use
CN107530365A (zh) 2015-03-25 2018-01-02 哈佛大学的校长及成员们 具有修饰的脱氧糖胺糖的大环内酯及其用途
MD1222Z (ro) * 2017-05-31 2018-08-31 ИНСТИТУТ ЭЛЕКТРОННОЙ ИНЖЕНЕРИИ И НАНОТЕХНОЛОГИЙ "D. Ghitu" АНМ Procedeu de tratare a materialului săditor al florilor înainte de plantare
JP7199722B2 (ja) 2019-12-25 2023-01-06 旭精工株式会社 硬貨搬送振分機構及びそれを備えた硬貨識別搬送装置

Family Cites Families (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3868414A (en) * 1973-01-22 1975-02-25 Merck & Co Inc Tetrahydrofluorene carboxylic acids and related compounds
AT342770B (de) * 1975-04-07 1978-04-25 Thomae Gmbh Dr K Verfahren zur herstellung neuer erythromycinderivate
DE2842759A1 (de) * 1978-09-30 1980-04-10 Merck Patent Gmbh Basische aether, diese enthaltende pharmazeutische zubereitungen und verfahren zu ihrer herstellung
IL114589A (en) * 1990-11-21 1999-12-22 Roussel Uclaf Intermediates for the preparation of erythromycin derivatives
FR2692579B1 (fr) * 1992-06-19 1995-06-02 Roussel Uclaf Nouveaux dérivés de la picromycine, leur procédé de préparation et leur application comme médicaments.
FR2697524B1 (fr) * 1992-11-05 1994-12-23 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
HRP930014A2 (en) * 1993-01-08 1994-08-31 Pliva Pharm & Chem Works 9-deoxo-9a-aza-11-deoxy-9a-homoeritromycin a 9a, 11-cyclic carbamates
FR2702480B1 (fr) * 1993-03-09 1995-04-28 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
AU2310795A (en) 1995-10-30
AU684939B2 (en) 1998-01-08
FI955913A0 (fi) 1995-12-08
DK0676409T3 (da) 2003-06-23
US5760233A (en) 1998-06-02
RO115634B1 (ro) 2000-04-28
US5656607A (en) 1997-08-12
TW316908B (lv) 1997-10-01
CA2164638A1 (fr) 1995-10-19
DE69529934D1 (de) 2003-04-24
MA23501A1 (fr) 1995-12-31
JP3000023B2 (ja) 2000-01-17
CZ296005B6 (cs) 2005-12-14
FI111264B (fi) 2003-06-30
OA10200A (fr) 1996-12-18
LV11182B (en) 1997-04-20
BR9506147A (pt) 1996-04-16
SA97170757A (ar) 2005-12-03
SV1995000018A (es) 1997-10-24
EP0676409B1 (fr) 2003-03-19
JO1850B1 (en) 1995-12-27
RU2141965C1 (ru) 1999-11-27
CO4370097A1 (es) 1996-10-07
GEP19991836B (en) 1999-11-05
PL180837B1 (pl) 2001-04-30
CN1126997A (zh) 1996-07-17
FI955913A7 (fi) 1995-12-08
CN1059445C (zh) 2000-12-13
MD663G2 (ro) 1997-07-31
MY114672A (en) 2002-12-31
EP0676409A1 (fr) 1995-10-11
EE9500080A (et) 1996-12-16
GB9506856D0 (en) 1995-05-24
NO954942D0 (no) 1995-12-06
GB2288174A (en) 1995-10-11
WO1995027720A1 (fr) 1995-10-19
IL112954A (en) 2000-07-16
HRP950217B1 (en) 2004-06-30
NO954942L (no) 1996-02-07
IL112954A0 (en) 1995-06-29
YU21695A (sh) 1997-12-05
UA44705C2 (uk) 2002-03-15
FR2718450B1 (fr) 1997-01-10
SI0676409T1 (en) 2003-06-30
CA2164638C (fr) 2003-12-30
HU9503505D0 (en) 1996-02-28
IS1865B (is) 2003-05-02
ES2189820T3 (es) 2003-07-16
DZ1869A1 (fr) 2002-02-17
SK154695A3 (en) 1996-10-02
PL311871A1 (en) 1996-03-18
HRP950217A2 (en) 1997-08-31
NO308361B1 (no) 2000-09-04
JPH07278177A (ja) 1995-10-24
SK284079B6 (sk) 2004-09-08
KR100317148B1 (ko) 2002-06-22
CZ322395A3 (en) 1996-08-14
IS4309A (is) 1995-11-17
NZ284498A (en) 1997-07-27
AP9500743A0 (en) 1995-07-31
BG61916B1 (bg) 1998-09-30
HU215396B (hu) 1998-12-28
YU49221B (sh) 2004-11-25
ZA952059B (en) 1996-03-13
ATE234853T1 (de) 2003-04-15
HUT73772A (en) 1996-09-30
TNSN95026A1 (fr) 1996-02-06
PT676409E (pt) 2003-08-29
PE2896A1 (es) 1996-02-12
BG100150A (bg) 1996-06-28
MD663F1 (ro) 1997-01-31
FR2718450A1 (fr) 1995-10-13
EE04498B1 (et) 2005-06-15
AP587A (en) 1997-04-29
DE69529934T2 (de) 2003-09-04

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