FI882836L - Menetelmä terapeuttisesti käyttökelpoisen (E)-2-(p-fluorifenetyyli)-3-fluoriallyyliamiinin valmistamiseksi - Google Patents
Menetelmä terapeuttisesti käyttökelpoisen (E)-2-(p-fluorifenetyyli)-3-fluoriallyyliamiinin valmistamiseksi Download PDFInfo
- Publication number
- FI882836L FI882836L FI882836A FI882836A FI882836L FI 882836 L FI882836 L FI 882836L FI 882836 A FI882836 A FI 882836A FI 882836 A FI882836 A FI 882836A FI 882836 L FI882836 L FI 882836L
- Authority
- FI
- Finland
- Prior art keywords
- fluoroallylamine
- fluorophenethyl
- therapeutically useful
- preparing therapeutically
- preparing
- Prior art date
Links
- 238000004519 manufacturing process Methods 0.000 title 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/185—Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
- A61K31/19—Carboxylic acids, e.g. valproic acid
- A61K31/195—Carboxylic acids, e.g. valproic acid having an amino group
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C211/00—Compounds containing amino groups bound to a carbon skeleton
- C07C211/01—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
- C07C211/26—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
- C07C211/29—Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
Landscapes
- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Veterinary Medicine (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Neurosurgery (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Neurology (AREA)
- Biomedical Technology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Epidemiology (AREA)
- Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US6275887A | 1987-06-16 | 1987-06-16 | |
| US6275887 | 1987-06-16 |
Publications (4)
| Publication Number | Publication Date |
|---|---|
| FI882836A0 FI882836A0 (fi) | 1988-06-14 |
| FI882836L true FI882836L (fi) | 1988-12-17 |
| FI90658B FI90658B (fi) | 1993-11-30 |
| FI90658C FI90658C (fi) | 1994-03-10 |
Family
ID=22044602
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI882836A FI90658C (fi) | 1987-06-16 | 1988-06-14 | Menetelmä terapeuttisesti käyttökelpoisen (E)-2-(p-fluorifenetyyli)-3-fluoriallyyliamiinin valmistamiseksi |
Country Status (16)
| Country | Link |
|---|---|
| EP (1) | EP0295604A1 (fi) |
| JP (1) | JP2511293B2 (fi) |
| KR (1) | KR970000142B1 (fi) |
| CN (1) | CN1031075A (fi) |
| AR (1) | AR243493A1 (fi) |
| AU (1) | AU612655B2 (fi) |
| CA (1) | CA1335897C (fi) |
| DK (1) | DK325788A (fi) |
| FI (1) | FI90658C (fi) |
| HU (1) | HU202823B (fi) |
| IL (1) | IL86746A0 (fi) |
| NO (1) | NO167381C (fi) |
| NZ (1) | NZ224982A (fi) |
| PH (1) | PH24012A (fi) |
| PT (1) | PT87732B (fi) |
| ZA (1) | ZA884183B (fi) |
Families Citing this family (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0639972A1 (en) * | 1992-05-15 | 1995-03-01 | University Of Saskatchewan | Method for preventing endothelium damage in mammals and for alleviating pain associated with gout and arthritis |
| HUT72316A (en) * | 1992-05-27 | 1996-04-29 | Merrell Dow Pharma | Use of (e)-2-(p-fluorophenethyl)-3-fluoroallylamine for the preparation of pharmaceutical composition against alzheimers`s disease |
| US5488188A (en) * | 1994-09-29 | 1996-01-30 | Merrell Dow Pharmaceuticals Inc. | Process for the preparation of (E)-1-amino-2-(fluoromethylene)-4-(p-fluorophenyl)butane, novel processes for preparing an intermediate thereof, and novel intermediates thereof |
| US5599986A (en) * | 1994-09-29 | 1997-02-04 | Hoechst Marion Roussel Inc. | Process for the preparation of alkali metal salts of diformylamide |
Family Cites Families (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US4454158A (en) * | 1981-06-01 | 1984-06-12 | Merrell Toraude Et Compagnie | Allyl amine MAO inhibitors |
| ATE71933T1 (de) * | 1985-12-05 | 1992-02-15 | Merrell Dow Pharma | Nichtaromatische fluoralkylamin-mao-inhibitoren. |
-
1988
- 1988-06-10 ZA ZA884183A patent/ZA884183B/xx unknown
- 1988-06-10 AR AR88311087A patent/AR243493A1/es active
- 1988-06-10 CA CA000569205A patent/CA1335897C/en not_active Expired - Fee Related
- 1988-06-10 AU AU17629/88A patent/AU612655B2/en not_active Ceased
- 1988-06-10 NZ NZ224982A patent/NZ224982A/xx unknown
- 1988-06-13 EP EP88109375A patent/EP0295604A1/en not_active Withdrawn
- 1988-06-14 FI FI882836A patent/FI90658C/fi not_active IP Right Cessation
- 1988-06-14 PH PH37070A patent/PH24012A/en unknown
- 1988-06-14 KR KR1019880007103A patent/KR970000142B1/ko not_active Expired - Fee Related
- 1988-06-15 CN CN88103634A patent/CN1031075A/zh active Pending
- 1988-06-15 DK DK325788A patent/DK325788A/da not_active Application Discontinuation
- 1988-06-15 PT PT87732A patent/PT87732B/pt not_active IP Right Cessation
- 1988-06-15 IL IL86746A patent/IL86746A0/xx unknown
- 1988-06-15 NO NO882655A patent/NO167381C/no not_active IP Right Cessation
- 1988-06-15 HU HU883079A patent/HU202823B/hu not_active IP Right Cessation
- 1988-06-16 JP JP63147052A patent/JP2511293B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| NO167381C (no) | 1991-10-30 |
| HUT51232A (en) | 1990-04-28 |
| AU1762988A (en) | 1988-12-22 |
| CN1031075A (zh) | 1989-02-15 |
| AR243493A1 (es) | 1993-08-31 |
| NO882655D0 (no) | 1988-06-15 |
| NO167381B (no) | 1991-07-22 |
| PH24012A (en) | 1990-02-09 |
| JP2511293B2 (ja) | 1996-06-26 |
| KR970000142B1 (ko) | 1997-01-04 |
| PT87732B (pt) | 1992-10-30 |
| DK325788D0 (da) | 1988-06-15 |
| PT87732A (pt) | 1988-07-01 |
| IL86746A0 (en) | 1988-11-30 |
| KR890000399A (ko) | 1989-03-14 |
| JPS6416752A (en) | 1989-01-20 |
| NZ224982A (en) | 1990-08-28 |
| EP0295604A1 (en) | 1988-12-21 |
| DK325788A (da) | 1988-12-17 |
| FI882836A0 (fi) | 1988-06-14 |
| CA1335897C (en) | 1995-06-13 |
| HU202823B (en) | 1991-04-29 |
| AU612655B2 (en) | 1991-07-18 |
| ZA884183B (en) | 1989-02-22 |
| FI90658C (fi) | 1994-03-10 |
| FI90658B (fi) | 1993-11-30 |
| NO882655L (no) | 1988-12-19 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| BB | Publication of examined application | ||
| MM | Patent lapsed |
Owner name: MERRELL DOW PHARMACEUTICALS INC. |