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FI882836L - Menetelmä terapeuttisesti käyttökelpoisen (E)-2-(p-fluorifenetyyli)-3-fluoriallyyliamiinin valmistamiseksi - Google Patents

Menetelmä terapeuttisesti käyttökelpoisen (E)-2-(p-fluorifenetyyli)-3-fluoriallyyliamiinin valmistamiseksi Download PDF

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Publication number
FI882836L
FI882836L FI882836A FI882836A FI882836L FI 882836 L FI882836 L FI 882836L FI 882836 A FI882836 A FI 882836A FI 882836 A FI882836 A FI 882836A FI 882836 L FI882836 L FI 882836L
Authority
FI
Finland
Prior art keywords
fluoroallylamine
fluorophenethyl
therapeutically useful
preparing therapeutically
preparing
Prior art date
Application number
FI882836A
Other languages
English (en)
Swedish (sv)
Other versions
FI882836A0 (fi
FI90658C (fi
FI90658B (fi
Inventor
Ian A Mcdonald
Michael G Palfreyman
Original Assignee
Merrell Dow Pharma
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Merrell Dow Pharma filed Critical Merrell Dow Pharma
Publication of FI882836A0 publication Critical patent/FI882836A0/fi
Publication of FI882836L publication Critical patent/FI882836L/fi
Application granted granted Critical
Publication of FI90658B publication Critical patent/FI90658B/fi
Publication of FI90658C publication Critical patent/FI90658C/fi

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/185Acids; Anhydrides, halides or salts thereof, e.g. sulfur acids, imidic, hydrazonic or hydroximic acids
    • A61K31/19Carboxylic acids, e.g. valproic acid
    • A61K31/195Carboxylic acids, e.g. valproic acid having an amino group
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C211/00Compounds containing amino groups bound to a carbon skeleton
    • C07C211/01Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms
    • C07C211/26Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring
    • C07C211/29Compounds containing amino groups bound to a carbon skeleton having amino groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing at least one six-membered aromatic ring the carbon skeleton being further substituted by halogen atoms or by nitro or nitroso groups
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Neurosurgery (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Epidemiology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
FI882836A 1987-06-16 1988-06-14 Menetelmä terapeuttisesti käyttökelpoisen (E)-2-(p-fluorifenetyyli)-3-fluoriallyyliamiinin valmistamiseksi FI90658C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US6275887A 1987-06-16 1987-06-16
US6275887 1987-06-16

Publications (4)

Publication Number Publication Date
FI882836A0 FI882836A0 (fi) 1988-06-14
FI882836L true FI882836L (fi) 1988-12-17
FI90658B FI90658B (fi) 1993-11-30
FI90658C FI90658C (fi) 1994-03-10

Family

ID=22044602

Family Applications (1)

Application Number Title Priority Date Filing Date
FI882836A FI90658C (fi) 1987-06-16 1988-06-14 Menetelmä terapeuttisesti käyttökelpoisen (E)-2-(p-fluorifenetyyli)-3-fluoriallyyliamiinin valmistamiseksi

Country Status (16)

Country Link
EP (1) EP0295604A1 (fi)
JP (1) JP2511293B2 (fi)
KR (1) KR970000142B1 (fi)
CN (1) CN1031075A (fi)
AR (1) AR243493A1 (fi)
AU (1) AU612655B2 (fi)
CA (1) CA1335897C (fi)
DK (1) DK325788A (fi)
FI (1) FI90658C (fi)
HU (1) HU202823B (fi)
IL (1) IL86746A0 (fi)
NO (1) NO167381C (fi)
NZ (1) NZ224982A (fi)
PH (1) PH24012A (fi)
PT (1) PT87732B (fi)
ZA (1) ZA884183B (fi)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
EP0639972A1 (en) * 1992-05-15 1995-03-01 University Of Saskatchewan Method for preventing endothelium damage in mammals and for alleviating pain associated with gout and arthritis
HUT72316A (en) * 1992-05-27 1996-04-29 Merrell Dow Pharma Use of (e)-2-(p-fluorophenethyl)-3-fluoroallylamine for the preparation of pharmaceutical composition against alzheimers`s disease
US5488188A (en) * 1994-09-29 1996-01-30 Merrell Dow Pharmaceuticals Inc. Process for the preparation of (E)-1-amino-2-(fluoromethylene)-4-(p-fluorophenyl)butane, novel processes for preparing an intermediate thereof, and novel intermediates thereof
US5599986A (en) * 1994-09-29 1997-02-04 Hoechst Marion Roussel Inc. Process for the preparation of alkali metal salts of diformylamide

Family Cites Families (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4454158A (en) * 1981-06-01 1984-06-12 Merrell Toraude Et Compagnie Allyl amine MAO inhibitors
ATE71933T1 (de) * 1985-12-05 1992-02-15 Merrell Dow Pharma Nichtaromatische fluoralkylamin-mao-inhibitoren.

Also Published As

Publication number Publication date
NO167381C (no) 1991-10-30
HUT51232A (en) 1990-04-28
AU1762988A (en) 1988-12-22
CN1031075A (zh) 1989-02-15
AR243493A1 (es) 1993-08-31
NO882655D0 (no) 1988-06-15
NO167381B (no) 1991-07-22
PH24012A (en) 1990-02-09
JP2511293B2 (ja) 1996-06-26
KR970000142B1 (ko) 1997-01-04
PT87732B (pt) 1992-10-30
DK325788D0 (da) 1988-06-15
PT87732A (pt) 1988-07-01
IL86746A0 (en) 1988-11-30
KR890000399A (ko) 1989-03-14
JPS6416752A (en) 1989-01-20
NZ224982A (en) 1990-08-28
EP0295604A1 (en) 1988-12-21
DK325788A (da) 1988-12-17
FI882836A0 (fi) 1988-06-14
CA1335897C (en) 1995-06-13
HU202823B (en) 1991-04-29
AU612655B2 (en) 1991-07-18
ZA884183B (en) 1989-02-22
FI90658C (fi) 1994-03-10
FI90658B (fi) 1993-11-30
NO882655L (no) 1988-12-19

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Date Code Title Description
BB Publication of examined application
MM Patent lapsed

Owner name: MERRELL DOW PHARMACEUTICALS INC.