FI116197B - Menetelmä farmaseuttisten koostumusten valmistamiseksi vaikeasti liukenevia aktiiviaineita varten - Google Patents

Menetelmä farmaseuttisten koostumusten valmistamiseksi vaikeasti liukenevia aktiiviaineita varten Download PDF

Info

Publication number: FI116197B
Authority: FI; Finland
Prior art keywords: component; fatty acid; polyglyceryl; carrier composition; weight
Prior art date: 1993-07-08

Application number

FI960032A

Other languages

English (en)

Finnish (fi)

Swedish (sv)

Other versions

FI960032L (fi

FI960032A0 (fi

Inventor

Ulrich Posanski

Original Assignee

Novartis Ag

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1993-07-08

Filing date

1996-01-03

Publication date

2005-10-14

Family has litigation

First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=6492300&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=FI116197(B) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.

1996-01-03 Application filed by Novartis Ag filed Critical Novartis Ag

1996-01-03 Publication of FI960032A0 publication Critical patent/FI960032A0/fi

1996-02-09 Publication of FI960032L publication Critical patent/FI960032L/fi

2005-10-14 Application granted granted Critical

2005-10-14 Publication of FI116197B publication Critical patent/FI116197B/fi

Links

238000000034 method Methods 0.000 title claims description 16
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238000002360 preparation method Methods 0.000 title description 20
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235000014113 dietary fatty acids Nutrition 0.000 claims abstract description 32
239000000194 fatty acid Substances 0.000 claims abstract description 32
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UIAGMCDKSXEBJQ-IBGZPJMESA-N 3-o-(2-methoxyethyl) 5-o-propan-2-yl (4s)-2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3,5-dicarboxylate Chemical compound COCCOC(=O)C1=C(C)NC(C)=C(C(=O)OC(C)C)[C@H]1C1=CC=CC([N+]([O-])=O)=C1 UIAGMCDKSXEBJQ-IBGZPJMESA-N 0.000 claims abstract description 5
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QUEDXNHFTDJVIY-UHFFFAOYSA-N γ-tocopherol Chemical class OC1=C(C)C(C)=C2OC(CCCC(C)CCCC(C)CCCC(C)C)(C)CCC2=C1 QUEDXNHFTDJVIY-UHFFFAOYSA-N 0.000 description 1

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K38/00—Medicinal preparations containing peptides
- A61K38/04—Peptides having up to 20 amino acids in a fully defined sequence; Derivatives thereof
- A61K38/12—Cyclic peptides, e.g. bacitracins; Polymyxins; Gramicidins S, C; Tyrocidins A, B or C
- A61K38/13—Cyclosporins
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/08—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite containing oxygen, e.g. ethers, acetals, ketones, quinones, aldehydes, peroxides
- A61K47/14—Esters of carboxylic acids, e.g. fatty acid monoglycerides, medium-chain triglycerides, parabens or PEG fatty acid esters
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/06—Organic compounds, e.g. natural or synthetic hydrocarbons, polyolefins, mineral oil, petrolatum or ozokerite
- A61K47/26—Carbohydrates, e.g. sugar alcohols, amino sugars, nucleic acids, mono-, di- or oligo-saccharides; Derivatives thereof, e.g. polysorbates, sorbitan fatty acid esters or glycyrrhizin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
- A61K47/44—Oils, fats or waxes according to two or more groups of A61K47/02-A61K47/42; Natural or modified natural oils, fats or waxes, e.g. castor oil, polyethoxylated castor oil, montan wax, lignite, shellac, rosin, beeswax or lanolin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/48—Preparations in capsules, e.g. of gelatin, of chocolate
- A61K9/4841—Filling excipients; Inactive ingredients
- A61K9/4858—Organic compounds
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A61P37/02—Immunomodulators
- A61P37/06—Immunosuppressants, e.g. drugs for graft rejection

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Medicinal Chemistry (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Epidemiology (AREA)
Immunology (AREA)
General Chemical & Material Sciences (AREA)
Bioinformatics & Cheminformatics (AREA)
Oil, Petroleum & Natural Gas (AREA)
Chemical Kinetics & Catalysis (AREA)
Biochemistry (AREA)
Gastroenterology & Hepatology (AREA)
Proteomics, Peptides & Aminoacids (AREA)
Transplantation (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Organic Chemistry (AREA)
Molecular Biology (AREA)
Medicinal Preparation (AREA)
Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
Medicines Containing Material From Animals Or Micro-Organisms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)

FI960032A 1993-07-08 1996-01-03 Menetelmä farmaseuttisten koostumusten valmistamiseksi vaikeasti liukenevia aktiiviaineita varten FI116197B (fi)

Applications Claiming Priority (4)

Application Number	Priority Date	Filing Date	Title
DE4322826		1993-07-08
DE4322826A DE4322826A1 (de)	1993-07-08	1993-07-08	Pharmazeutisches Präparat
EP9402248		1994-07-08
PCT/EP1994/002248 WO1995001786A1 (de)	1993-07-08	1994-07-08	Pharmazeutische präparate für schwerlösliche wirkstoffe

Publications (3)

Publication Number	Publication Date
FI960032A0 FI960032A0 (fi)	1996-01-03
FI960032L FI960032L (fi)	1996-02-09
FI116197B true FI116197B (fi)	2005-10-14

Family

ID=6492300

Family Applications (2)

Application Number	Title	Priority Date	Filing Date
FI960032A FI116197B (fi)	1993-07-08	1996-01-03	Menetelmä farmaseuttisten koostumusten valmistamiseksi vaikeasti liukenevia aktiiviaineita varten
FI960042A FI116714B (fi)	1993-07-08	1996-01-04	Menetelmä valmistaa farmaseuttisia valmisteita, jotka on tarkoitettu niukkaliukoisille aktiivisille aineille

Family Applications After (1)

Application Number	Title	Priority Date	Filing Date
FI960042A FI116714B (fi)	1993-07-08	1996-01-04	Menetelmä valmistaa farmaseuttisia valmisteita, jotka on tarkoitettu niukkaliukoisille aktiivisille aineille

Country Status (24)

Country	Link
EP (3)	EP0710103B1 (el)
JP (4)	JPH08512303A (el)
KR (2)	KR100359044B1 (el)
CN (2)	CN1313154C (el)
AT (3)	ATE201985T1 (el)
AU (2)	AU7385094A (el)
BR (1)	BR9407002A (el)
CA (2)	CA2166204C (el)
CY (2)	CY2308B1 (el)
CZ (1)	CZ291401B6 (el)
DE (6)	DE4322826A1 (el)
DK (3)	DK0710104T3 (el)
ES (3)	ES2124420T3 (el)
FI (2)	FI116197B (el)
GR (1)	GR3036571T3 (el)
HU (2)	HU228127B1 (el)
NO (2)	NO306763B1 (el)
NZ (2)	NZ269552A (el)
PL (1)	PL179717B1 (el)
PT (2)	PT1092429E (el)
RU (1)	RU2140291C1 (el)
SI (1)	SI1092429T1 (el)
SK (1)	SK280615B6 (el)
WO (2)	WO1995001785A1 (el)

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1993
- 1993-07-08 DE DE4322826A patent/DE4322826A1/de not_active Withdrawn
1994
- 1994-07-08 EP EP94922269A patent/EP0710103B1/de not_active Expired - Lifetime
- 1994-07-08 ES ES94923715T patent/ES2124420T3/es not_active Expired - Lifetime
- 1994-07-08 NZ NZ269552A patent/NZ269552A/xx not_active IP Right Cessation
- 1994-07-08 EP EP94923715A patent/EP0710104B1/de not_active Expired - Lifetime
- 1994-07-08 DK DK94923715T patent/DK0710104T3/da active
- 1994-07-08 PL PL94312255A patent/PL179717B1/pl unknown
- 1994-07-08 DE DE59410365T patent/DE59410365D1/de not_active Expired - Lifetime
- 1994-07-08 PT PT00122248T patent/PT1092429E/pt unknown
- 1994-07-08 CN CNB031522890A patent/CN1313154C/zh not_active Expired - Lifetime
- 1994-07-08 NZ NZ269808A patent/NZ269808A/xx not_active IP Right Cessation
- 1994-07-08 DE DE59407239T patent/DE59407239D1/de not_active Expired - Fee Related
- 1994-07-08 AU AU73850/94A patent/AU7385094A/en not_active Abandoned
- 1994-07-08 AT AT94922269T patent/ATE201985T1/de active
- 1994-07-08 EP EP00122248A patent/EP1092429B1/de not_active Expired - Lifetime
- 1994-07-08 ES ES00122248T patent/ES2218046T3/es not_active Expired - Lifetime
- 1994-07-08 DE DE4494851T patent/DE4494851D2/de not_active Expired - Fee Related
- 1994-07-08 DK DK00122248T patent/DK1092429T3/da active
- 1994-07-08 PT PT94922269T patent/PT710103E/pt unknown
- 1994-07-08 ES ES94922269T patent/ES2159564T3/es not_active Expired - Lifetime
- 1994-07-08 HU HU9503965A patent/HU228127B1/hu not_active IP Right Cessation
- 1994-07-08 DE DE4494850T patent/DE4494850D2/de not_active Expired - Fee Related
- 1994-07-08 JP JP7503833A patent/JPH08512303A/ja active Pending
- 1994-07-08 DK DK94922269T patent/DK0710103T3/da active
- 1994-07-08 JP JP7503830A patent/JPH08512301A/ja active Pending
- 1994-07-08 CA CA002166204A patent/CA2166204C/en not_active Expired - Fee Related
- 1994-07-08 SK SK19-96A patent/SK280615B6/sk not_active IP Right Cessation
- 1994-07-08 BR BR9407002A patent/BR9407002A/pt not_active Application Discontinuation
- 1994-07-08 WO PCT/EP1994/002238 patent/WO1995001785A1/de not_active Ceased
- 1994-07-08 KR KR1019960700042A patent/KR100359044B1/ko not_active Expired - Fee Related
- 1994-07-08 CZ CZ199645A patent/CZ291401B6/cs not_active IP Right Cessation
- 1994-07-08 CA CA002164100A patent/CA2164100A1/en not_active Abandoned
- 1994-07-08 AU AU73457/94A patent/AU689486B2/en not_active Expired
- 1994-07-08 SI SI9430465T patent/SI1092429T1/xx unknown
- 1994-07-08 WO PCT/EP1994/002248 patent/WO1995001786A1/de not_active Ceased
- 1994-07-08 AT AT94923715T patent/ATE172876T1/de not_active IP Right Cessation
- 1994-07-08 CN CN94192714A patent/CN1121853C/zh not_active Expired - Lifetime
- 1994-07-08 DE DE59409787T patent/DE59409787D1/de not_active Expired - Lifetime
- 1994-07-08 RU RU96102012A patent/RU2140291C1/ru active
- 1994-07-08 AT AT00122248T patent/ATE261720T1/de active
- 1994-07-08 KR KR1019960700026A patent/KR100386533B1/ko not_active Expired - Lifetime
- 1994-07-08 HU HU9503868A patent/HU223073B1/hu active IP Right Grant
1996
- 1996-01-03 FI FI960032A patent/FI116197B/fi active IP Right Grant
- 1996-01-04 FI FI960042A patent/FI116714B/fi not_active IP Right Cessation
- 1996-01-05 NO NO960069A patent/NO306763B1/no not_active IP Right Cessation
- 1996-01-05 NO NO960062A patent/NO306929B1/no not_active IP Right Cessation
2001
- 2001-09-10 GR GR20010401428T patent/GR3036571T3/el unknown
2002
- 2002-12-12 CY CY0200068A patent/CY2308B1/xx unknown
2005
- 2005-09-08 CY CY0500049A patent/CY2604B2/el unknown
2009
- 2009-02-04 JP JP2009023837A patent/JP2009138008A/ja not_active Withdrawn
2011
- 2011-03-24 JP JP2011066324A patent/JP2011153150A/ja active Pending

Also Published As

Publication number	Publication date
EP0710103B1 (de)	2001-06-13
BR9407002A (pt)	1996-09-03
SK280615B6 (sk)	2000-05-16
CN1313154C (zh)	2007-05-02
DE4494851D2 (de)	1996-12-19
RU2140291C1 (ru)	1999-10-27
CN1121853C (zh)	2003-09-24
DE59407239D1 (de)	1998-12-10
HU228127B1 (en)	2012-12-28
SI1092429T1 (en)	2004-08-31
DK1092429T3 (da)	2004-07-19
EP0710103A1 (de)	1996-05-08
DK0710104T3 (da)	1999-07-19
ATE261720T1 (de)	2004-04-15
NO960062D0 (no)	1996-01-05
ATE172876T1 (de)	1998-11-15
FI960042A0 (fi)	1996-01-04
CY2604B2 (el)	2010-04-28
NO306763B1 (no)	1999-12-20
JPH08512301A (ja)	1996-12-24
ES2159564T3 (es)	2001-10-16
JPH08512303A (ja)	1996-12-24
ATE201985T1 (de)	2001-06-15
PT1092429E (pt)	2004-08-31
CZ4596A3 (en)	1996-04-17
NO306929B1 (no)	2000-01-17
SK1996A3 (en)	1997-04-09
CA2164100A1 (en)	1995-01-19
FI960042L (fi)	1996-01-04
PT710103E (pt)	2001-11-30
DE4494850D2 (de)	1996-08-22
ES2124420T3 (es)	1999-02-01
WO1995001785A1 (de)	1995-01-19
DK0710103T3 (da)	2001-09-24
FI960032L (fi)	1996-02-09
FI960032A0 (fi)	1996-01-03
EP1092429A1 (de)	2001-04-18
DE59410365D1 (de)	2004-04-22
ES2218046T3 (es)	2004-11-16
FI116714B (fi)	2006-02-15
HU9503868D0 (en)	1996-02-28
HU223073B1 (hu)	2004-03-01
CN1496743A (zh)	2004-05-19
KR100359044B1 (ko)	2003-02-05
EP0710104B1 (de)	1998-11-04
CA2166204A1 (en)	1995-01-19
AU7385094A (en)	1995-02-06
PL312255A1 (en)	1996-04-01
GR3036571T3 (en)	2001-12-31
NZ269552A (en)	1996-07-26
JP2011153150A (ja)	2011-08-11
HU9503965D0 (en)	1996-03-28
NZ269808A (en)	1996-07-26
DE59409787D1 (de)	2001-07-19
CZ291401B6 (cs)	2003-03-12
CN1128495A (zh)	1996-08-07
DE4322826A1 (de)	1995-01-12
CY2308B1 (en)	2003-11-14
WO1995001786A1 (de)	1995-01-19
KR100386533B1 (ko)	2003-08-21
HUT73661A (en)	1996-09-30
HUT73427A (en)	1996-07-29
PL179717B1 (pl)	2000-10-31
AU689486B2 (en)	1998-04-02
AU7345794A (en)	1995-02-06
NO960062L (no)	1996-01-05
NO960069D0 (no)	1996-01-05
CA2166204C (en)	2009-04-14
EP0710104A1 (de)	1996-05-08
EP1092429B1 (de)	2004-03-17
NO960069L (no)	1996-01-05
JP2009138008A (ja)	2009-06-25

Publication	Publication Date	Title
FI116197B (fi)	2005-10-14	Menetelmä farmaseuttisten koostumusten valmistamiseksi vaikeasti liukenevia aktiiviaineita varten
US20050048087A1 (en)	2005-03-03	Pharmaceutical compositions for sparingly soluble therapeutic agents
AU2002333098B2 (en)	2006-03-16	Novel cyclosporin analog microemulsion preconcentrates
EP0711550A1 (en)	1996-05-15	Cyclosporin-containing soft capsule compositions
US6187747B1 (en)	2001-02-13	Pharmaceutical composition comprising cyclosporin
US20020049158A1 (en)	2002-04-25	Oral drug composition containing a verapamil derivative as a drug-absorption promotor
EP0985412B1 (en)	2004-10-27	Cyclosporin compositions
MXPA05001351A (es)	2005-10-05	Composiciones farmaceuticas orales que comprenden ciclosporina.
EP1151755B1 (en)	2005-03-16	Pharmaceutical compositions comprising cyclosporin as active ingredient
AU762963B2 (en)	2003-07-10	Cyclosporin solution
AU741923B2 (en)	2001-12-13	Pharmaceutical compositions

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Date	Code	Title	Description
1997-08-12	GB	Transfer or assigment of application	Owner name: NOVARTIS AG
2005-10-14	FG	Patent granted	Ref document number: 116197 Country of ref document: FI

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