EE03099B1 - Tsüklilised iminoderivaadid, neid ühendeid sisaldavad ravimid ja meetodid nende saamiseks - Google Patents

Tsüklilised iminoderivaadid, neid ühendeid sisaldavad ravimid ja meetodid nende saamiseks

Info

Publication number: EE03099B1
Authority: EE; Estonia
Prior art keywords: compounds; preparation; drugs containing; cyclic imino; methods
Prior art date: 1990-11-02

Application number

EE9400438A

Other languages

English (en)

Estonian (et)

Inventor

Himmelsbach Frank

Austel Volkhard

Pieper Helmut

Eisert Wolfgang

Mller Thomas

Weisenberger Johannes

Linz G�nter

Kr�ger Gerd

Original Assignee

Dr. Karl Thomae Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1990-11-02

Filing date

1994-11-23

Publication date

1998-06-15

1994-11-23 Application filed by Dr. Karl Thomae Gmbh filed Critical Dr. Karl Thomae Gmbh

1998-06-15 Publication of EE03099B1 publication Critical patent/EE03099B1/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/08—Vasodilators for multiple indications
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- C07D207/273—2-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
- C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
- C07D207/24—Oxygen or sulfur atoms
- C07D207/26—2-Pyrrolidones
- C07D207/273—2-Pyrrolidones with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to other ring carbon atoms
- C07D207/277—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
- C07F9/572—Five-membered rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
General Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Engineering & Computer Science (AREA)
Animal Behavior & Ethology (AREA)
Bioinformatics & Cheminformatics (AREA)
Biochemistry (AREA)
Diabetes (AREA)
Cardiology (AREA)
Heart & Thoracic Surgery (AREA)
Molecular Biology (AREA)
Hematology (AREA)
Vascular Medicine (AREA)
Pulmonology (AREA)
Urology & Nephrology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
Hydrogenated Pyridines (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Nitrogen Condensed Heterocyclic Rings (AREA)
Pyrrole Compounds (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Other In-Based Heterocyclic Compounds (AREA)
Indole Compounds (AREA)
Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
Detergent Compositions (AREA)

EE9400438A 1990-11-02 1994-11-23 Tsüklilised iminoderivaadid, neid ühendeid sisaldavad ravimid ja meetodid nende saamiseks EE03099B1 (et)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
DE4035961A DE4035961A1 (de)	1990-11-02	1990-11-02	Cyclische iminoderivate, diese verbindungen enthaltende arzneimittel und verfahren zu ihrer herstellung

Publications (1)

Publication Number	Publication Date
EE03099B1 true EE03099B1 (et)	1998-06-15

Family

ID=6418111

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EE9400438A EE03099B1 (et)	1990-11-02	1994-11-23	Tsüklilised iminoderivaadid, neid ühendeid sisaldavad ravimid ja meetodid nende saamiseks

Country Status (25)

Country	Link
US (2)	US5541343A (xx)
EP (1)	EP0483667B1 (xx)
JP (1)	JP2937589B2 (xx)
KR (1)	KR100223135B1 (xx)
AT (1)	ATE163008T1 (xx)
BG (1)	BG62025B2 (xx)
BR (1)	BR1100445A (xx)
CA (1)	CA2054850C (xx)
DE (2)	DE4035961A1 (xx)
DK (1)	DK0483667T3 (xx)
EE (1)	EE03099B1 (xx)
ES (1)	ES2113867T3 (xx)
FI (1)	FI107606B (xx)
GR (1)	GR3026508T3 (xx)
HK (1)	HK1008742A1 (xx)
HU (2)	HUT67288A (xx)
IE (1)	IE913822A1 (xx)
IL (1)	IL99926A (xx)
MX (1)	MX9203677A (xx)
NO (1)	NO174806B (xx)
NZ (1)	NZ240463A (xx)
PT (1)	PT99402B (xx)
RU (1)	RU2040519C1 (xx)
SG (1)	SG81852A1 (xx)
ZA (1)	ZA918734B (xx)

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EP3071541B1 (en)	2013-11-21	2023-06-07	Marquette University	Substituted (4'-hydroxyphenyl)cycloalkane compounds and uses thereof as selective agonists of the estrogen receptor beta isoform
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US4247466A (en) *	1979-07-05	1981-01-27	American Cyanamid Company	Lactone metabolites of 3-(4-biphenylylcarbonyl)propionic acid
EP0194548A3 (de) *	1985-03-12	1988-08-17	Dr. Karl Thomae GmbH	Neue Sulfonylaminoäthylverbindungen, diese Verbindungen enthaltende Arzneimittel und Verfahren zu ihrer Herstellung
PT82200B (pt) *	1985-03-16	1990-02-08	Wellcome Found	Processo para a preparacao de novos derivados do acido hidroxamico e de composicoes farmaceuticas que os contem
DE3823299A1 (de) *	1988-07-07	1990-01-11	Schering Ag	Substituierte phenyl-pyrrolidin-2-one, -oxazolidin-2-one und -imidazolidin-2-one, ihre herstellung sowie verwendung in arzneimitteln

1990
- 1990-11-02 DE DE4035961A patent/DE4035961A1/de not_active Ceased
1991
- 1991-10-24 DK DK91118148T patent/DK0483667T3/da active
- 1991-10-24 DE DE59108930T patent/DE59108930D1/de not_active Expired - Lifetime
- 1991-10-24 EP EP91118148A patent/EP0483667B1/de not_active Expired - Lifetime
- 1991-10-24 AT AT91118148T patent/ATE163008T1/de not_active IP Right Cessation
- 1991-10-24 SG SG9601241A patent/SG81852A1/en unknown
- 1991-10-24 ES ES91118148T patent/ES2113867T3/es not_active Expired - Lifetime
- 1991-10-31 FI FI915136A patent/FI107606B/fi not_active IP Right Cessation
- 1991-10-31 PT PT99402A patent/PT99402B/pt not_active IP Right Cessation
- 1991-11-01 CA CA002054850A patent/CA2054850C/en not_active Expired - Lifetime
- 1991-11-01 IL IL9992691A patent/IL99926A/en not_active IP Right Cessation
- 1991-11-01 IE IE382291A patent/IE913822A1/en not_active IP Right Cessation
- 1991-11-01 HU HU913455A patent/HUT67288A/hu unknown
- 1991-11-01 NO NO914294A patent/NO174806B/no not_active IP Right Cessation
- 1991-11-01 JP JP3313154A patent/JP2937589B2/ja not_active Expired - Lifetime
- 1991-11-01 RU SU915001905A patent/RU2040519C1/ru active
- 1991-11-02 KR KR1019910019458A patent/KR100223135B1/ko not_active Expired - Lifetime
- 1991-11-04 ZA ZA918734A patent/ZA918734B/xx unknown
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1992
- 1992-06-29 MX MX9203677A patent/MX9203677A/es unknown
1994
- 1994-01-25 BG BG098416A patent/BG62025B2/bg unknown
- 1994-11-23 EE EE9400438A patent/EE03099B1/xx not_active IP Right Cessation
- 1994-12-28 US US08/365,336 patent/US5541343A/en not_active Expired - Lifetime
1995
- 1995-06-01 US US08/458,096 patent/US5591769A/en not_active Expired - Lifetime
- 1995-06-02 HU HU95P/P00156P patent/HU211563A9/hu unknown
1997
- 1997-05-06 BR BR1100445-2A patent/BR1100445A/pt active IP Right Grant
1998
- 1998-04-03 GR GR980400691T patent/GR3026508T3/el unknown
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Also Published As

Publication number	Publication date
IL99926A (en)	1996-06-18
KR920009793A (ko)	1992-06-25
DK0483667T3 (da)	1998-09-23
PT99402B (pt)	1999-04-30
FI915136A0 (fi)	1991-10-31
CA2054850C (en)	2001-01-02
ES2113867T3 (es)	1998-05-16
ZA918734B (en)	1993-05-04
NO174806C (xx)	1994-07-13
EP0483667B1 (de)	1998-02-04
EP0483667A2 (de)	1992-05-06
US5591769A (en)	1997-01-07
GR3026508T3 (en)	1998-07-31
CA2054850A1 (en)	1992-05-03
RU2040519C1 (ru)	1995-07-25
HUT67288A (en)	1995-03-28
HU913455D0 (en)	1992-01-28
NZ240463A (en)	1997-04-24
NO174806B (no)	1994-04-05
DE59108930D1 (de)	1998-03-12
MX9203677A (es)	1992-07-01
BG62025B2 (bg)	1998-12-30
JP2937589B2 (ja)	1999-08-23
EP0483667A3 (en)	1992-09-16
AU8692691A (en)	1992-05-07
FI915136L (fi)	1992-05-03
IL99926A0 (en)	1992-08-18
ATE163008T1 (de)	1998-02-15
DE4035961A1 (de)	1992-05-07
HU211563A9 (en)	1995-12-28
FI107606B (fi)	2001-09-14
BR1100445A (pt)	2000-07-18
AU650488B2 (en)	1994-06-23
NO914294L (no)	1992-05-04
HK1008742A1 (en)	1999-05-14
PT99402A (pt)	1992-09-30
US5541343A (en)	1996-07-30
SG81852A1 (en)	2001-07-24
KR100223135B1 (ko)	1999-10-15
IE913822A1 (en)	1992-05-22
JPH04264068A (ja)	1992-09-18
NO914294D0 (no)	1991-11-01

Publication	Publication Date	Title
EE03099B1 (et)	1998-06-15	Tsüklilised iminoderivaadid, neid ühendeid sisaldavad ravimid ja meetodid nende saamiseks
FI923691A0 (fi)	1992-08-18	Cykliska iminoderivat, dessa foereningar innehaollande farmaceutiska blandningar och foerfarande foer deras framstaellning.
NO180045C (no)	1997-02-05	Cykliske iminoderivater, og legemiddelpreparater inneholdende dem
NO177852C (no)	1995-12-06	Bifenylderivater, legemidler inneholdende disse, og anvendelse av dem for fremstilling av legemidler
NO920957L (no)	1992-09-14	Cykliske urinstoffderivater og legemidler inneholdende disse forbindelser
NO923466L (no)	1993-03-08	Heterocykliske forbindelser med 5 ledd, fremgangsmaate forfremstilling, samt legemidler som inneholder disse forbindelser
MA20369A1 (fr)	1985-10-01	Compositions a base de derives de la piperidine ,nouveaux derives de la piperidine et leurs procedes de preparation
MX9803556A (es)	1998-09-30	Derivados de aminoacidos, medicamentos que contienen tales compuestos y metodos para producirlos.

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