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DK3256468T3 - Tricykliske forbindelser og anvendelser deraf i lægemidler - Google Patents

Tricykliske forbindelser og anvendelser deraf i lægemidler Download PDF

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Publication number
DK3256468T3
DK3256468T3 DK16748725.5T DK16748725T DK3256468T3 DK 3256468 T3 DK3256468 T3 DK 3256468T3 DK 16748725 T DK16748725 T DK 16748725T DK 3256468 T3 DK3256468 T3 DK 3256468T3
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Prior art keywords
pharmaceuticals
tricyclic compounds
tricyclic
compounds
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DK16748725.5T
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English (en)
Inventor
Xiaojun Wang
Xinye Yang
Shengqiang Pan
Rui Guo
Junwen Wu
Yingjun Zhang
Changchung Cheng
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Sunshine Lake Pharma Co Ltd
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    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a chain containing hetero atoms as chain links
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
    • A61K31/4155—1,2-Diazoles non condensed and containing further heterocyclic rings
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/4192—1,2,3-Triazoles
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    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/42—Oxazoles
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    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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TWI698430B (zh) 2020-07-11
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US10183917B2 (en) 2019-01-22
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