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DK0668851T3 - Hidtil ukendt arylpropionsyrederivat, fremgangsmåde til fremstilling heraf og anvendelse heraf som analgetisk middel - Google Patents

Hidtil ukendt arylpropionsyrederivat, fremgangsmåde til fremstilling heraf og anvendelse heraf som analgetisk middel

Info

Publication number
DK0668851T3
DK0668851T3 DK93924604.7T DK93924604T DK0668851T3 DK 0668851 T3 DK0668851 T3 DK 0668851T3 DK 93924604 T DK93924604 T DK 93924604T DK 0668851 T3 DK0668851 T3 DK 0668851T3
Authority
DK
Denmark
Prior art keywords
analgesic
preparation
propionic acid
acid derivative
hitherto unknown
Prior art date
Application number
DK93924604.7T
Other languages
English (en)
Inventor
Germano Carganico
Casellas David Mauleon
Perez M Luisa Garcia
Original Assignee
Menarini Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8278730&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DK0668851(T3) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Menarini Lab filed Critical Menarini Lab
Application granted granted Critical
Publication of DK0668851T3 publication Critical patent/DK0668851T3/da

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C215/00Compounds containing amino and hydroxy groups bound to the same carbon skeleton
    • C07C215/02Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton
    • C07C215/04Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated
    • C07C215/06Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic
    • C07C215/10Compounds containing amino and hydroxy groups bound to the same carbon skeleton having hydroxy groups and amino groups bound to acyclic carbon atoms of the same carbon skeleton the carbon skeleton being saturated and acyclic with one amino group and at least two hydroxy groups bound to the carbon skeleton
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P21/00Drugs for disorders of the muscular or neuromuscular system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07CACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40Unsaturated compounds
    • C07C59/76Unsaturated compounds containing keto groups
    • C07C59/84Unsaturated compounds containing keto groups containing six membered aromatic rings

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Neurology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
DK93924604.7T 1992-11-10 1993-11-09 Hidtil ukendt arylpropionsyrederivat, fremgangsmåde til fremstilling heraf og anvendelse heraf som analgetisk middel DK0668851T3 (da)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
ES09202260A ES2058024B1 (es) 1992-11-10 1992-11-10 Nuevo derivado arilpropionico, procedimiento de fabricacion del mismo y su utilizacion como analgesico.

Publications (1)

Publication Number Publication Date
DK0668851T3 true DK0668851T3 (da) 1997-12-22

Family

ID=8278730

Family Applications (1)

Application Number Title Priority Date Filing Date
DK93924604.7T DK0668851T3 (da) 1992-11-10 1993-11-09 Hidtil ukendt arylpropionsyrederivat, fremgangsmåde til fremstilling heraf og anvendelse heraf som analgetisk middel

Country Status (27)

Country Link
US (1) US5554789A (da)
EP (1) EP0668851B1 (da)
JP (1) JP3778516B2 (da)
KR (1) KR100284838B1 (da)
AT (1) ATE153649T1 (da)
AU (1) AU674040B2 (da)
BG (1) BG61723B1 (da)
BR (1) BR9307408A (da)
CA (1) CA2149013C (da)
CZ (1) CZ286621B6 (da)
DE (2) DE69311130T2 (da)
DK (1) DK0668851T3 (da)
ES (2) ES2058024B1 (da)
FI (1) FI108637B (da)
GR (2) GR960300012T1 (da)
HK (1) HK1006306A1 (da)
HU (2) HU217973B (da)
MD (1) MD921G2 (da)
NO (2) NO304306B1 (da)
NZ (1) NZ257557A (da)
PL (1) PL175265B1 (da)
RO (1) RO118712B1 (da)
RU (1) RU2128160C1 (da)
SK (1) SK280550B6 (da)
UA (1) UA44233C2 (da)
UY (1) UY24179A1 (da)
WO (1) WO1994011332A1 (da)

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US20080051411A1 (en) * 2002-12-17 2008-02-28 Cink Russell D Salts of Fenofibric Acid and Pharmaceutical Formulations Thereof
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EP1739072A1 (en) * 2005-06-15 2007-01-03 Laboratorios Menarini S.A. Polymorphic forms of dexketoprofen trometamol, preparation and pharmaceutical compositions thereof
CN101594878A (zh) 2006-09-18 2009-12-02 雷普特药品公司 通过给予受体相关蛋白(rap)-缀合物对肝病症的治疗
TWI364413B (en) * 2008-07-25 2012-05-21 Univ Nat Central Racemic ibuprofen amine salt and synthesis method thereof
NZ592378A (en) * 2008-10-31 2012-09-28 C A I R Biosciences Gmbh Choline and tromethamine salt of licofelone
DK3395372T3 (da) 2009-02-20 2022-04-19 Enhanx Biopharm Inc System til afgivelse af glutathion-baseret medikament
CN110075069A (zh) 2009-05-06 2019-08-02 实验室护肤股份有限公司 包含活性剂-磷酸钙颗粒复合物的皮肤递送组合物及其应用
ES2350670B1 (es) * 2009-06-10 2011-12-07 Polichem, S.L. Composicion veterinaria de ketoprofeno
CN101928214B (zh) * 2009-06-19 2012-12-19 黄石世星药业有限责任公司 右旋酮洛芬氨丁三醇的一种合成方法
WO2011001213A1 (en) * 2009-06-30 2011-01-06 Abdi Ibrahim Ilac Sanayi Ve Ticaret Anonim Sirketi A process for preparing dexketoprofen trometamol form a and form b crystals
US20120077778A1 (en) 2010-09-29 2012-03-29 Andrea Bourdelais Ladder-Frame Polyether Conjugates
CN102557976B (zh) * 2010-12-15 2015-06-10 辽宁盛京制药有限公司 溴芬酸有机盐及其制备方法、其组合物及用途
TR201104864A2 (tr) 2011-05-18 2012-12-21 B�Lg�� Mahmut Deksketoprofen içeren suda çözünebilir formülasyonlar.
TR201205317A2 (tr) 2011-05-18 2012-12-21 B�Lg�� Mahmut Deksketoprofen içeren efervesan formülasyonlar.
CN102381986A (zh) * 2011-07-25 2012-03-21 南京特丰药业股份有限公司 一种右旋布洛芬氨丁三醇盐及其口服溶液的制备方法
WO2013022410A2 (en) 2011-08-08 2013-02-14 Mahmut Bilgic Production method for effervescent formulations comprising dexketoprofen
WO2013095315A1 (en) 2011-12-19 2013-06-27 Mahmut Bilgic Formulations comprising dexketoprofen (particle size 300-2500 micrometer)
WO2013100877A1 (en) 2011-12-27 2013-07-04 Mahmut Bilgic Dexketoprofen formulations
ES2501415T3 (es) 2012-06-06 2016-02-22 Galenicum Health S.L. Composiciones farmacéuticas estables de acción rápida
EP2759293A1 (en) 2013-01-25 2014-07-30 Laboratorios Lesvi, S.L. Pharmaceutical compositions of (+)-(s)-2-(3-benzoylphenyl)propionic acid tromethamine salt
ES2512497T1 (es) 2013-02-06 2014-10-24 Galenicum Health S.L. Proceso para preparar una composición farmacéutica estable que comprende dexketoprofeno trometamol
ITMI20130210A1 (it) 2013-02-14 2014-08-15 Menarini Lab Composizioni farmaceutiche contenenti dexketoprofene e tramadolo
TR201616365A1 (tr) 2016-11-14 2018-05-21 Sanovel Ilac Sanayi Ve Ticaret Anonim Sirketi Deksketoprofen ve eletri̇ptanin oral farmasöti̇k kompozi̇syonlari
US10927067B2 (en) 2016-11-28 2021-02-23 Sarin Parayil Organic crystalline salt of haloacetic acid
TR201618765A2 (tr) 2016-12-16 2018-07-23 Imuneks Farma Ilac Sanayi Ve Ticaret Anonim Sirketi Ağrı ve enflamasyonun tedavisi için steroid olmayan anti-enflamatuvar ilaçlar ve H2 reseptörü antagonisti kombinasyonları.
KR102552315B1 (ko) * 2020-11-11 2023-07-06 대원제약주식회사 펠루비프로펜 신규 염을 주성분으로 하며 위장장애 부작용이 저감된 약학적 조성물
KR102462607B1 (ko) * 2020-11-11 2022-11-03 대원제약주식회사 펠루비프로펜 신규 염을 주성분으로 하는 안정성이 증가된 약학적 조성물
US20250214968A1 (en) * 2022-03-25 2025-07-03 Ildong Pharmaceutical Co., Ltd. Novel Salt of GLP-1 Receptor Agonist Compound, Preparation Method Thereof and Pharmaceutical Composition Comprising Thereof

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Also Published As

Publication number Publication date
UY24179A1 (es) 1996-09-03
HU217973B (hu) 2000-05-28
NO951790D0 (no) 1995-05-08
CZ114995A3 (en) 1995-10-18
JPH08503203A (ja) 1996-04-09
NO951790L (no) 1995-07-06
EP0668851A1 (en) 1995-08-30
MD921G2 (ro) 1998-10-31
HU9802850D0 (en) 1999-02-01
KR100284838B1 (ko) 2001-04-02
CA2149013C (en) 2004-08-10
ES2081780T3 (es) 1997-07-01
HK1006306A1 (en) 1999-02-19
CZ286621B6 (cs) 2000-05-17
FI952230L (fi) 1995-05-09
ES2058024A1 (es) 1994-10-16
EP0668851B1 (en) 1997-05-28
PL175265B1 (pl) 1998-12-31
US5554789A (en) 1996-09-10
FI108637B (fi) 2002-02-28
UA44233C2 (uk) 2002-02-15
HU9501375D0 (en) 1995-06-28
DE69311130D1 (de) 1997-07-03
HU219975B (hu) 2001-10-28
BG99609A (bg) 1996-01-31
NO2006007I1 (no) 2006-08-14
GR3024344T3 (en) 1997-10-31
CA2149013A1 (en) 1994-05-26
WO1994011332A1 (en) 1994-05-26
ATE153649T1 (de) 1997-06-15
JP3778516B2 (ja) 2006-05-24
ES2081780T1 (es) 1996-03-16
HUT71903A (en) 1996-02-28
DE69311130T2 (de) 1997-09-18
GR960300012T1 (en) 1996-03-31
SK280550B6 (sk) 2000-03-13
DE668851T1 (de) 1996-10-10
AU674040B2 (en) 1996-12-05
BR9307408A (pt) 1999-08-24
NO304306B1 (no) 1998-11-30
RU95112575A (ru) 1997-06-20
NZ257557A (en) 1996-01-26
AU5421094A (en) 1994-06-08
RU2128160C1 (ru) 1999-03-27
RO118712B1 (ro) 2003-09-30
ES2058024B1 (es) 1995-05-01
SK60395A3 (en) 1995-09-13
FI952230A0 (fi) 1995-05-09
BG61723B1 (bg) 1998-04-30
PL308466A1 (en) 1995-07-24

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