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CY1107574T1 - Παρασκευασματα αντιβιοτικων κατηγοριας κινολονης βραδειας απελευθερωσης και μεθοδος για την παραγωγη αυτων - Google Patents

Παρασκευασματα αντιβιοτικων κατηγοριας κινολονης βραδειας απελευθερωσης και μεθοδος για την παραγωγη αυτων

Info

Publication number
CY1107574T1
CY1107574T1 CY20071100478T CY071100478T CY1107574T1 CY 1107574 T1 CY1107574 T1 CY 1107574T1 CY 20071100478 T CY20071100478 T CY 20071100478T CY 071100478 T CY071100478 T CY 071100478T CY 1107574 T1 CY1107574 T1 CY 1107574T1
Authority
CY
Cyprus
Prior art keywords
preparations
antibiotic
lettle
liberty
clinic
Prior art date
Application number
CY20071100478T
Other languages
English (en)
Inventor
Venkata-Rangarao Kanikanti
Roland Rupp
Wolfgang Weber
Peter Deuringer
Jan-Olav Henck
Heino Stass
Takaaki Nishioka
Yoshifumi Katakawa
Chika Taniguchi
Hitoshi Ichihashi
Original Assignee
Bayer Healthcare Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Healthcare Ag filed Critical Bayer Healthcare Ag
Publication of CY1107574T1 publication Critical patent/CY1107574T1/el

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/205—Polysaccharides, e.g. alginate, gums; Cyclodextrin
    • A61K9/2054—Cellulose; Cellulose derivatives, e.g. hydroxypropyl methylcellulose
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2072—Pills, tablets, discs, rods characterised by shape, structure or size; Tablets with holes, special break lines or identification marks; Partially coated tablets; Disintegrating flat shaped forms
    • A61K9/2086—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat
    • A61K9/209—Layered tablets, e.g. bilayer tablets; Tablets of the type inert core-active coat containing drug in at least two layers or in the core and in at least one outer layer
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2004—Excipients; Inactive ingredients
    • A61K9/2022—Organic macromolecular compounds
    • A61K9/2027—Organic macromolecular compounds obtained by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyvinyl pyrrolidone, poly(meth)acrylates

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Epidemiology (AREA)
  • Organic Chemistry (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)

Abstract

Η παρούσα εφεύρεση αναφέρεται σε παρασκευάσματα στοματικώς χορηγήσιμα τα οποία περιέχουν κάποιο αντιβιοτικό κατηγορίας κινολόνης, και τα οποία απελευθερώνουν τη δραστική ουσία βραδέως. Μία προτιμώμενη διαμόρφωση αναφέρεται σε παρασκευάσματα τα οποία ως δραστική ουσία περιέχουν το μείγμα κάποιας ελεύθερης βάσης κινολόνης και άλατος αυτής. Προτιμούνται ιδιαιτέρως μείγματα υδροχλωρικής κιπροφλοξακίνης και βεταΐνης κιπροφλοξακίνης.
CY20071100478T 2000-06-26 2007-04-04 Παρασκευασματα αντιβιοτικων κατηγοριας κινολονης βραδειας απελευθερωσης και μεθοδος για την παραγωγη αυτων CY1107574T1 (el)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE10031043A DE10031043A1 (de) 2000-06-26 2000-06-26 Retardzubereitungen von Chinolonantibiotika und Verfahren zu ihrer Herstellung
EP01949412A EP1296685B1 (de) 2000-06-26 2001-06-13 Retard-zubereitungen von chinolon-antibiotika und verfahren zu ihrer herstellung

Publications (1)

Publication Number Publication Date
CY1107574T1 true CY1107574T1 (el) 2013-03-13

Family

ID=7646816

Family Applications (1)

Application Number Title Priority Date Filing Date
CY20071100478T CY1107574T1 (el) 2000-06-26 2007-04-04 Παρασκευασματα αντιβιοτικων κατηγοριας κινολονης βραδειας απελευθερωσης και μεθοδος για την παραγωγη αυτων

Country Status (40)

Country Link
US (3) US7709022B2 (el)
EP (1) EP1296685B1 (el)
JP (1) JP4958373B2 (el)
KR (1) KR100939617B1 (el)
CN (1) CN1273138C (el)
AR (1) AR029688A1 (el)
AT (1) ATE355062T1 (el)
AU (1) AU2001270573A1 (el)
BG (1) BG65914B1 (el)
BR (1) BRPI0111911B8 (el)
CA (1) CA2414271C (el)
CU (1) CU23264B7 (el)
CY (1) CY1107574T1 (el)
CZ (1) CZ301812B6 (el)
DE (2) DE10031043A1 (el)
DK (1) DK1296685T3 (el)
DO (1) DOP2001000199A (el)
EE (1) EE04992B1 (el)
ES (1) ES2282270T3 (el)
GT (1) GT200100126A (el)
HN (1) HN2001000132A (el)
HR (1) HRP20030050B1 (el)
HU (1) HU229806B1 (el)
IL (2) IL153333A0 (el)
MA (1) MA25761A1 (el)
MX (1) MXPA02012727A (el)
MY (1) MY140994A (el)
NO (1) NO325415B1 (el)
NZ (1) NZ523352A (el)
PE (1) PE20020207A1 (el)
PL (1) PL203710B1 (el)
PT (1) PT1296685E (el)
RU (1) RU2332204C2 (el)
SI (1) SI1296685T1 (el)
SK (1) SK287384B6 (el)
SV (1) SV2002000505A (el)
TW (1) TWI279232B (el)
UA (1) UA83616C2 (el)
WO (1) WO2002000219A1 (el)
ZA (1) ZA200210350B (el)

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Also Published As

Publication number Publication date
BR0111911A (pt) 2003-05-13
SK18212002A3 (sk) 2003-04-01
US20070065509A1 (en) 2007-03-22
DE10031043A1 (de) 2002-02-14
DK1296685T3 (da) 2007-05-07
CZ20024216A3 (cs) 2003-04-16
DE50112123D1 (de) 2007-04-12
CN1273138C (zh) 2006-09-06
TWI279232B (en) 2007-04-21
BG107372A (bg) 2003-09-30
WO2002000219A1 (de) 2002-01-03
IL153333A (en) 2010-05-31
HU229806B1 (en) 2014-07-28
RU2332204C2 (ru) 2008-08-27
ES2282270T3 (es) 2007-10-16
HRP20030050B1 (en) 2011-07-31
ATE355062T1 (de) 2006-03-15
HN2001000132A (es) 2001-09-11
JP2004504278A (ja) 2004-02-12
NO20026160D0 (no) 2002-12-20
NO20026160L (no) 2002-12-20
NZ523352A (en) 2004-08-27
US8187632B2 (en) 2012-05-29
IL153333A0 (en) 2003-07-06
PL360632A1 (en) 2004-09-20
US20070237824A1 (en) 2007-10-11
MY140994A (en) 2010-02-12
PE20020207A1 (es) 2002-04-27
EE200200707A (et) 2004-08-16
CN1438889A (zh) 2003-08-27
NO325415B1 (no) 2008-04-21
SV2002000505A (es) 2002-12-02
ZA200210350B (en) 2004-02-10
US7780986B2 (en) 2010-08-24
SK287384B6 (sk) 2010-08-09
HK1058479A1 (en) 2004-05-21
US7709022B2 (en) 2010-05-04
SI1296685T1 (sl) 2007-06-30
EP1296685A1 (de) 2003-04-02
EP1296685B1 (de) 2007-02-28
HUP0300953A2 (hu) 2003-08-28
CU23264B7 (es) 2008-03-14
BRPI0111911B1 (pt) 2015-08-25
PL203710B1 (pl) 2009-11-30
GT200100126A (es) 2002-01-31
AU2001270573A1 (en) 2002-01-08
PT1296685E (pt) 2007-05-31
UA83616C2 (uk) 2008-08-11
MXPA02012727A (es) 2003-05-14
BRPI0111911B8 (pt) 2021-05-25
BG65914B1 (bg) 2010-05-31
AR029688A1 (es) 2003-07-10
HUP0300953A3 (en) 2009-04-28
KR20030023883A (ko) 2003-03-20
EE04992B1 (et) 2008-04-15
HRP20030050A2 (en) 2004-06-30
US20040024018A1 (en) 2004-02-05
JP4958373B2 (ja) 2012-06-20
KR100939617B1 (ko) 2010-02-01
CA2414271C (en) 2005-09-27
DOP2001000199A (es) 2002-05-15
CA2414271A1 (en) 2002-12-23
MA25761A1 (fr) 2003-04-01
CZ301812B6 (cs) 2010-06-30

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