[go: up one dir, main page]

AU2001234159A1 - Process for producing quinolonecarboxylic acids and intermediates thereof - Google Patents

Process for producing quinolonecarboxylic acids and intermediates thereof

Info

Publication number
AU2001234159A1
AU2001234159A1 AU2001234159A AU3415901A AU2001234159A1 AU 2001234159 A1 AU2001234159 A1 AU 2001234159A1 AU 2001234159 A AU2001234159 A AU 2001234159A AU 3415901 A AU3415901 A AU 3415901A AU 2001234159 A1 AU2001234159 A1 AU 2001234159A1
Authority
AU
Australia
Prior art keywords
intermediates
quinolonecarboxylic acids
producing
producing quinolonecarboxylic
acids
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Abandoned
Application number
AU2001234159A
Other languages
English (en)
Inventor
Toshifumi Akiba
Toshiaki Jouno
Tatsuru Saito
Yu-Ichiro Tani
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Daiichi Pharmaceutical Co Ltd
Original Assignee
Daiichi Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Daiichi Pharmaceutical Co Ltd filed Critical Daiichi Pharmaceutical Co Ltd
Publication of AU2001234159A1 publication Critical patent/AU2001234159A1/en
Abandoned legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/48—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen
    • C07D215/54—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3
    • C07D215/56—Carbon atoms having three bonds to hetero atoms with at the most one bond to halogen attached in position 3 with oxygen atoms in position 4
    • A—HUMAN NECESSITIES
    • A01—AGRICULTURE; FORESTRY; ANIMAL HUSBANDRY; HUNTING; TRAPPING; FISHING
    • A01N—PRESERVATION OF BODIES OF HUMANS OR ANIMALS OR PLANTS OR PARTS THEREOF; BIOCIDES, e.g. AS DISINFECTANTS, AS PESTICIDES OR AS HERBICIDES; PEST REPELLANTS OR ATTRACTANTS; PLANT GROWTH REGULATORS
    • A01N43/00—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds
    • A01N43/34—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom
    • A01N43/40—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings
    • A01N43/42—Biocides, pest repellants or attractants, or plant growth regulators containing heterocyclic compounds having rings with one nitrogen atom as the only ring hetero atom six-membered rings condensed with carbocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/47—Quinolines; Isoquinolines
    • A61K31/4709—Non-condensed quinolines and containing further heterocyclic rings
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/56—Ring systems containing three or more rings
    • C07D209/96—Spiro-condensed ring systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D215/00—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems
    • C07D215/02—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom
    • C07D215/16—Heterocyclic compounds containing quinoline or hydrogenated quinoline ring systems having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen atoms or carbon atoms directly attached to the ring nitrogen atom with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D215/18—Halogen atoms or nitro radicals
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D401/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom
    • C07D401/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings
    • C07D401/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, at least one ring being a six-membered ring with only one nitrogen atom containing two hetero rings directly linked by a ring-member-to-ring-member bond

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Wood Science & Technology (AREA)
  • Dentistry (AREA)
  • Environmental Sciences (AREA)
  • Zoology (AREA)
  • Engineering & Computer Science (AREA)
  • Agronomy & Crop Science (AREA)
  • Pest Control & Pesticides (AREA)
  • Plant Pathology (AREA)
  • Oncology (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Quinoline Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
AU2001234159A 2000-02-25 2001-02-23 Process for producing quinolonecarboxylic acids and intermediates thereof Abandoned AU2001234159A1 (en)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2000054349 2000-02-25
JP2000-54349 2000-02-25
JP2000-117208 2000-04-13
JP2000117208 2000-04-13
PCT/JP2001/001370 WO2001062734A1 (fr) 2000-02-25 2001-02-23 Procede de production d'acides quinolonecarboxyliques et de leurs intermediaires

Publications (1)

Publication Number Publication Date
AU2001234159A1 true AU2001234159A1 (en) 2001-09-03

Family

ID=26586419

Family Applications (1)

Application Number Title Priority Date Filing Date
AU2001234159A Abandoned AU2001234159A1 (en) 2000-02-25 2001-02-23 Process for producing quinolonecarboxylic acids and intermediates thereof

Country Status (10)

Country Link
EP (1) EP1258478A4 (fr)
KR (1) KR20020075447A (fr)
CN (1) CN1426399A (fr)
AU (1) AU2001234159A1 (fr)
CA (1) CA2400819A1 (fr)
HK (1) HK1048119A1 (fr)
IL (1) IL151451A0 (fr)
NO (1) NO20024046L (fr)
RU (1) RU2002122758A (fr)
WO (1) WO2001062734A1 (fr)

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RU2299205C2 (ru) * 2000-02-09 2007-05-20 Дайити Фармасьютикал Ко., Лтд. Средство против кислотоустойчивых бактерий, содержащее пиридонкарбоновые кислоты в качестве активного компонента
EP1669354B1 (fr) * 2003-09-29 2013-03-20 Daiichi Sankyo Company, Limited Derive d'acide 8-cyanoquinolone-carboxylique
CN1305849C (zh) * 2004-12-29 2007-03-21 江苏正大天晴药业股份有限公司 3－甲氨基哌啶及其盐的制备方法
CN101830815B (zh) * 2010-03-03 2014-01-29 伊泰(北京)合成技术有限公司 环状化合物及以其作为中间体制备氮杂螺环化合物的方法

Family Cites Families (10)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3420743A1 (de) * 1984-06-04 1985-12-05 Bayer Ag, 5090 Leverkusen 7-amino-1-cyclopropyl-6,8-dihalogen-1,4-dihydro-4-oxo-3-chinolincarbonsaeuren, verfahren zu ihrer herstellung sowie diese enthaltende antibakterielle mittel
DE3906365A1 (de) * 1988-07-15 1990-01-18 Bayer Ag 7-(1-pyrrolidinyl)-3-chinolon- und -naphthyridoncarbonsaeure-derivate, verfahren sowie substituierte (oxa)diazabicyclooctane und -nonane als zwischenprodukte zu ihrer herstellung, und sie enthaltende antibakterielle mittel und futterzusatzstoffe
KR950014567B1 (ko) * 1991-08-01 1995-12-08 주식회사대웅제약 신규한 퀴놀론 카르복실산 유도체
TW252107B (fr) * 1993-08-27 1995-07-21 Hokuriku Pharmacetical Co Ltd
DE4342186A1 (de) * 1993-12-10 1995-06-14 Bayer Ag Eintopfverfahren zur Herstellung von 3-Chinoloncarbonsäurederivaten
WO1996022988A1 (fr) * 1995-01-24 1996-08-01 Hokuriku Seiyaku Co., Ltd. Derives de l'acide quiloleine carboxylique
KR19990071558A (ko) * 1995-11-22 1999-09-27 스즈키 다다시 치환된 아미노시클로알킬피롤리딘 유도체
JP4148550B2 (ja) * 1997-11-26 2008-09-10 イハラケミカル工業株式会社 ５−アミノ−１−シクロプロピル−４−オキソキノリン−３−カルボン酸誘導体とその製造方法
JP2000247970A (ja) * 1999-02-26 2000-09-12 Hokuriku Seiyaku Co Ltd ５−アミノ−８−メチル−７−ピロリジニルキノリン−３−カルボン酸誘導体の製造法及びその製造中間体
JP2000319261A (ja) * 1999-05-13 2000-11-21 Dai Ichi Seiyaku Co Ltd キノロンカルボン酸類の製造方法

Also Published As

Publication number Publication date
EP1258478A1 (fr) 2002-11-20
CA2400819A1 (fr) 2001-08-30
RU2002122758A (ru) 2004-01-10
NO20024046D0 (no) 2002-08-23
KR20020075447A (ko) 2002-10-04
CN1426399A (zh) 2003-06-25
HK1048119A1 (en) 2003-03-21
NO20024046L (no) 2002-10-24
IL151451A0 (en) 2003-04-10
WO2001062734A1 (fr) 2001-08-30
EP1258478A4 (fr) 2006-03-15

Similar Documents

Publication Publication Date Title
AU2001227573A1 (en) Ceramics and process for producing
AU2001279683A1 (en) Biosensor and method for production thereof
AU2001252638A1 (en) Process for the preparation of 2-halobenzoic acids
AU2001284514A1 (en) Process for producing ester
AU2882201A (en) Sustained-release preparation and process for producing the same
AU2002234635A1 (en) Method for producing cyclohexane dicarboxylic acids and the derivatives thereof
AU2001294549A1 (en) Process and intermediates
AU2001264134A1 (en) Microconnectors and method for their production
HU9901526D0 (en) Pharmaceutical intermediates and process for producing them
AU2002312431A1 (en) Novel process for preparing rac-bicalutamide and its intermediates
AU2001230207A1 (en) Method for the production of 1-amino-3-aryl-uracils
AU2002325845A1 (en) Preparation process for atorvastatin and intermediates
AU3228301A (en) Process for producing fumaric ester
AU2002221090A1 (en) Process for production of dicarboxylic acids
AU2001272757A1 (en) Process for producing 5-fluorooxyindole and for producing intermediate therefor
AU2002210547A1 (en) Method for producing acetic acid
AU2001232342A1 (en) Processes for preparing quinoline derivatives and intermediates thereof
AU2001234159A1 (en) Process for producing quinolonecarboxylic acids and intermediates thereof
AU2001270569A1 (en) Method for producing amides or esters
AU2002221164A1 (en) (r)-hydroxycarboxylic acid producing recombinant microorganism and process for preparing (r)-hydroxycarboxylic acid using the same
AU2001267855A1 (en) Intermediate and process for producing fluorinated carboxylic acid derivative from the same
AU2001269501A1 (en) Process for producing 2-hydroxy-4-methylthiobutanoic acid
AU2002229149A1 (en) Process for producing hydrazinomonosaccharide derivatives and use thereof
AU2001274004A1 (en) Method for the production of 2- coumarone and substituted 2-coumarones
AU2001283030A1 (en) Process for making 3-hydroxyalkanenitriles and hydroxyaminoalkanes