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NO996108L - 9-oksinerytromycinderivater - Google Patents

9-oksinerytromycinderivater

Info

Publication number
NO996108L
NO996108L NO996108A NO996108A NO996108L NO 996108 L NO996108 L NO 996108L NO 996108 A NO996108 A NO 996108A NO 996108 A NO996108 A NO 996108A NO 996108 L NO996108 L NO 996108L
Authority
NO
Norway
Prior art keywords
compounds
formula
disclosed
methods
oksinerytromycinderivater
Prior art date
Application number
NO996108A
Other languages
English (en)
Norwegian (no)
Other versions
NO996108D0 (no
Inventor
Yong-Jin Wu
Original Assignee
Pfizer Prod Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer Prod Inc filed Critical Pfizer Prod Inc
Publication of NO996108D0 publication Critical patent/NO996108D0/no
Publication of NO996108L publication Critical patent/NO996108L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/70—Carbohydrates; Sugars; Derivatives thereof
    • A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
    • A61K31/7048—Compounds having saccharide radicals and heterocyclic rings having oxygen as a ring hetero atom, e.g. leucoglucosan, hesperidin, erythromycin, nystatin, digitoxin or digoxin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Molecular Biology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biochemistry (AREA)
  • Biotechnology (AREA)
  • Genetics & Genomics (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Communicable Diseases (AREA)
  • Oncology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
NO996108A 1997-06-11 1999-12-10 9-oksinerytromycinderivater NO996108L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US4934997P 1997-06-11 1997-06-11
PCT/IB1998/000741 WO1998056800A1 (fr) 1997-06-11 1998-05-15 Derives de 9-oxime erythromycine

Publications (2)

Publication Number Publication Date
NO996108D0 NO996108D0 (no) 1999-12-10
NO996108L true NO996108L (no) 2000-02-10

Family

ID=21959341

Family Applications (1)

Application Number Title Priority Date Filing Date
NO996108A NO996108L (no) 1997-06-11 1999-12-10 9-oksinerytromycinderivater

Country Status (31)

Country Link
EP (1) EP0988308A1 (fr)
JP (1) JP2000513026A (fr)
KR (1) KR20010013660A (fr)
CN (1) CN1259135A (fr)
AP (1) AP9801253A0 (fr)
AR (1) AR012244A1 (fr)
AU (1) AU7226798A (fr)
BG (1) BG103947A (fr)
BR (1) BR9810021A (fr)
CA (1) CA2293335A1 (fr)
CO (1) CO4940506A1 (fr)
CZ (1) CZ9904388A3 (fr)
EA (1) EA199901016A1 (fr)
GT (1) GT199800074A (fr)
HN (1) HN1998000073A (fr)
HR (1) HRP980316A2 (fr)
HU (1) HUP0002252A3 (fr)
ID (1) ID24529A (fr)
IL (1) IL132767A0 (fr)
IS (1) IS5251A (fr)
MA (1) MA26505A1 (fr)
NO (1) NO996108L (fr)
OA (1) OA11225A (fr)
PA (1) PA8451801A1 (fr)
PE (1) PE79899A1 (fr)
PL (1) PL337606A1 (fr)
TN (1) TNSN98083A1 (fr)
TR (1) TR199902995T2 (fr)
TW (1) TW448174B (fr)
WO (1) WO1998056800A1 (fr)
ZA (1) ZA985018B (fr)

Families Citing this family (29)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HN1998000159A (es) * 1997-10-29 1999-02-09 Monsanto Co Derivados de 9- amino - 3 ceto eritromicina
DE69926005T2 (de) 1998-09-22 2006-05-18 Pfizer Products Inc., Groton Carbamat- und carbazatketolidantibiotika
FR2786188B1 (fr) * 1998-11-24 2002-10-31 Hoechst Marion Roussel Inc Nouveaux derives de l'erythromycine, leur procede de preparation et leur applicaion comme medicaments
US6258785B1 (en) 1998-12-02 2001-07-10 Pfizer Inc. Crystalline 9-E-(O-methyl)oxime of 11, 12-dideoxy-3-de(2,6-dideoxy-3-C-methyl-3-O-methyl-α-L-ribohexopyranosyloxy)-6-O-methyl-12,11-(iminocarbonyl-(2-(3-(4-(3-pyridinyl)1H-imadazol-1-yl)propyl)hydrazono))-3-oxoerythromycin
EP1298138B1 (fr) * 1998-12-10 2006-11-02 Pfizer Products Inc. Dérivés anitiobiotiques de Carbamate et de Carbazate Kètolides
US6284732B1 (en) * 1998-12-18 2001-09-04 Bio-Rad Laboratories, Inc. Peptides and peptide analogues designed from HFE protein and their uses in the treatment of iron overload diseases
NZ515027A (en) * 1999-04-16 2004-01-30 Kosan Biosciences Inc Erythromycin derivatives as antibiotics
OA11945A (en) 1999-05-24 2006-04-13 Pfizer Prod Inc 13-Methyl erythromycin derivatives.
JP2003501439A (ja) * 1999-06-07 2003-01-14 アボット・ラボラトリーズ ６−ｏ−カルバメートケトライド誘導体
ID27331A (id) * 1999-09-29 2001-03-29 Pfizer Prod Inc Pembuatan antibiotik-antibiotik ketolida karbamat
EP1114826A3 (fr) * 1999-12-29 2001-10-31 Pfizer Products Inc. Macrolides antibactériennes et prokinétiques
EP1439186A3 (fr) * 1999-12-29 2004-11-03 Pfizer Products Inc. Intermédiaires pour macrolides antibactérielles et procinétiques
US6946446B2 (en) 2000-02-24 2005-09-20 Abbott Laboratories Anti-infective agents useful against multidrug-resistant strains of bacteria
US6403776B1 (en) 2000-07-05 2002-06-11 Pfizer Inc. Synthesis of carbamate ketolide antibiotics
WO2003090761A1 (fr) * 2002-04-25 2003-11-06 Abbott Laboratories Antibacteriens 9-oxime macrolide
AR043050A1 (es) 2002-09-26 2005-07-13 Rib X Pharmaceuticals Inc Compuestos heterociclicos bifuncionales y metodos para preparar y usar los mismos
EP1638549A4 (fr) 2003-03-10 2011-06-15 Optimer Pharmaceuticals Inc Nouveaux agents antibacteriens
EP1723159B1 (fr) 2004-02-27 2019-06-12 Melinta Therapeutics, Inc. Composes macrocycliques et leurs procedes de fabrication et d'utilisation
CA2703475A1 (fr) 2007-10-25 2009-04-30 Cempra Pharmaceuticals, Inc. Procede pour la preparation d'agents antibacteriens macrolides
EP2358379B1 (fr) 2008-10-24 2015-12-16 Cempra Pharmaceuticals, Inc. Biodéfenses utilisant des macrolides contenant du triazole
US9937194B1 (en) 2009-06-12 2018-04-10 Cempra Pharmaceuticals, Inc. Compounds and methods for treating inflammatory diseases
ES2608285T3 (es) 2009-09-10 2017-04-07 Cempra Pharmaceuticals, Inc. Procedimientos para el tratamiento de paludismo, tuberculosis y enfermedades por MAC
CN102146085B (zh) * 2010-02-09 2014-03-26 北京理工大学 一种9-肟醚酮内酯衍生物、制备方法及其药物组合物
MX361413B (es) 2010-03-22 2018-12-05 Cempra Pharmaceuticals Inc Star Formas cristalinas de un macrólido y usos para las mismas.
KR101945324B1 (ko) 2010-05-20 2019-02-07 셈프라 파마슈티컬스, 인크. 매크로라이드들 및 케톨라이드들과 이의 중간체들을 제조하는 공정들
US9815863B2 (en) 2010-09-10 2017-11-14 Cempra Pharmaceuticals, Inc. Hydrogen bond forming fluoro ketolides for treating diseases
KR20140139083A (ko) 2012-03-27 2014-12-04 셈프라 파마슈티컬스, 인크. 마크롤라이드계 항생제를 투여하기 위한 비경구 제제
RU2015138796A (ru) 2013-03-14 2017-04-19 Семпра Фармасьютикалс, Инк. Способы и составы для лечения респираторных заболеваний
JP6675973B2 (ja) 2013-03-15 2020-04-08 センプラ ファーマシューティカルズ，インコーポレイテッド マクロライド抗菌薬を調製するための集束的な方法

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them
US5527780A (en) * 1992-11-05 1996-06-18 Roussel Uclaf Erythromycin derivatives
FR2718450B1 (fr) * 1994-04-08 1997-01-10 Roussel Uclaf Nouveaux dérivés de l'érythromycine, leur procédé de préparation et leur application comme médicaments.

Also Published As

Publication number Publication date
MA26505A1 (fr) 2004-12-20
TNSN98083A1 (fr) 2005-03-15
KR20010013660A (ko) 2001-02-26
CA2293335A1 (fr) 1998-12-17
CZ9904388A3 (cs) 2002-10-16
AP9801253A0 (en) 1999-12-04
TW448174B (en) 2001-08-01
NO996108D0 (no) 1999-12-10
PE79899A1 (es) 1999-08-25
ZA985018B (en) 1999-12-10
OA11225A (en) 2003-07-17
HRP980316A2 (en) 1999-04-30
BG103947A (en) 2000-07-31
HUP0002252A3 (en) 2002-01-28
PA8451801A1 (es) 2000-05-24
IS5251A (is) 1999-11-16
ID24529A (id) 2000-07-20
HN1998000073A (es) 1999-01-08
AU7226798A (en) 1998-12-30
AR012244A1 (es) 2000-09-27
JP2000513026A (ja) 2000-10-03
PL337606A1 (en) 2000-08-28
IL132767A0 (en) 2001-03-19
CN1259135A (zh) 2000-07-05
EA199901016A1 (ru) 2000-06-26
TR199902995T2 (xx) 2000-02-21
HUP0002252A2 (hu) 2000-12-28
GT199800074A (es) 1999-11-27
WO1998056800A1 (fr) 1998-12-17
CO4940506A1 (es) 2000-07-24
BR9810021A (pt) 2000-09-19
EP0988308A1 (fr) 2000-03-29

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Legal Events

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FC2A Withdrawal, rejection or dismissal of laid open patent application