NO20081686L - Fremgangsmate for fremstilling av esteroksazolidinforbindelser, og deres omdannelse til Florfnicol - Google Patents

Fremgangsmate for fremstilling av esteroksazolidinforbindelser, og deres omdannelse til Florfnicol

Info

Publication number: NO20081686L
Authority: NO; Norway
Prior art keywords: preparation; florfnicol; conversion; oxazolidine compounds; ester oxazolidine
Prior art date: 2005-09-07

Application number

NO20081686A

Other languages

English (en)

Norwegian (no)

Inventor

James C Towson

Original Assignee

Schering Plough Ltd

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2005-09-07

Filing date

2008-04-04

Publication date

2008-06-05

2008-04-04 Application filed by Schering Plough Ltd filed Critical Schering Plough Ltd

2008-06-05 Publication of NO20081686L publication Critical patent/NO20081686L/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C317/00—Sulfones; Sulfoxides
- C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
- C07C317/48—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C07C315/04—Preparation of sulfones; Preparation of sulfoxides by reactions not involving the formation of sulfone or sulfoxide groups
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
- C07C315/00—Preparation of sulfones; Preparation of sulfoxides
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D263/00—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings
- C07D263/02—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings
- C07D263/04—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
- C07D263/06—Heterocyclic compounds containing 1,3-oxazole or hydrogenated 1,3-oxazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by oxygen atoms, attached to ring carbon atoms

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Chemical Kinetics & Catalysis (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)

NO20081686A 2005-09-07 2008-04-04 Fremgangsmate for fremstilling av esteroksazolidinforbindelser, og deres omdannelse til Florfnicol NO20081686L (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
US71468505P	2005-09-07	2005-09-07
PCT/US2006/034370 WO2007030405A2 (fr)	2005-09-07	2006-08-31	Procede de preparation de composes d'ester oxazolidine et leur conversion en florfenicol

Publications (1)

Publication Number	Publication Date
NO20081686L true NO20081686L (no)	2008-06-05

Family

ID=37684114

Family Applications (3)

Application Number	Title	Priority Date	Filing Date
NO20081686A NO20081686L (no)	2005-09-07	2008-04-04	Fremgangsmate for fremstilling av esteroksazolidinforbindelser, og deres omdannelse til Florfnicol
NO20081685A NO20081685L (no)	2005-09-07	2008-04-04	Fremgangsmate for fremstilling oksazolidin-beskyttelse aminodolforbindelser anvendbare som mellomprodukter for Florfenicol
NO20081684A NO20081684L (no)	2005-09-07	2008-04-04	En forbedret fremgangsmate for fremstilling av okazolidin-beskyttende aminodiolforbindelser anvendbare som mellomprodukter for Florfenicol

Family Applications After (2)

Application Number	Title	Priority Date	Filing Date
NO20081685A NO20081685L (no)	2005-09-07	2008-04-04	Fremgangsmate for fremstilling oksazolidin-beskyttelse aminodolforbindelser anvendbare som mellomprodukter for Florfenicol
NO20081684A NO20081684L (no)	2005-09-07	2008-04-04	En forbedret fremgangsmate for fremstilling av okazolidin-beskyttende aminodiolforbindelser anvendbare som mellomprodukter for Florfenicol

Country Status (19)

Country	Link
US (3)	US7786329B2 (fr)
EP (3)	EP1928820B1 (fr)
JP (3)	JP2009507074A (fr)
KR (3)	KR20080049040A (fr)
CN (3)	CN101300238A (fr)
AU (3)	AU2006287696A1 (fr)
BR (3)	BRPI0615767A2 (fr)
CA (3)	CA2621971A1 (fr)
EC (3)	ECSP088266A (fr)
ES (1)	ES2459205T3 (fr)
IL (3)	IL189828A0 (fr)
MX (3)	MX2008003188A (fr)
NO (3)	NO20081686L (fr)
RU (3)	RU2008112950A (fr)
SI (1)	SI1928820T1 (fr)
TW (3)	TWI331139B (fr)
UA (1)	UA93212C2 (fr)
WO (3)	WO2007030386A2 (fr)
ZA (3)	ZA200802047B (fr)

Families Citing this family (16)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
PE20050386A1 (es)	2003-05-29	2005-06-23	Schering Plough Ltd	Composiciones farmaceuticas de florfenicol
EP1785414A1 (fr) *	2005-11-09	2007-05-16	KRKA, tovarna zdravil, d.d., Novo mesto	Procédé pour la synthèse des intermédiaires du chloramphenicol ou de ses analogues
MX2009006467A (es) *	2006-12-13	2009-08-21	Schering Plough Ltd	Profarmacos solubles en agua de cloranfenicol, tiamfenicol y analogos de los mismos.
WO2009015111A2 (fr) *	2007-07-25	2009-01-29	Intervet Intermatonal B.V.	Procédé pour préparer des aminodiols d'oxazolidine et d'oxazolidinone
PE20091171A1 (es) *	2007-12-14	2009-08-03	Schering Plough Ltd	Proceso para recuperar florfenicol y analogos de florfenicol
CA2732017A1 (fr) *	2008-07-30	2010-02-04	Intervet International B.V.	Procede de preparation de composes aminodiol d'oxazoline proteges utiles comme produits intermediaires dans la production de florfenicol
CN101941927B (zh) *	2010-09-28	2012-10-03	湖北美天生物科技有限公司	氟苯尼考中间体(1r,2r)-2-氨基-1–(4-(甲砜基)苯基)-1,3-丙二醇的合成方法
EP2705044A1 (fr)	2011-05-02	2014-03-12	Zoetis Llc	Nouvelles céphalosporines utiles en tant qu'agents antibactériens
CN103254103A (zh) *	2013-06-05	2013-08-21	南通金利油脂工业有限公司	氟化剂在制备氟苯尼考工艺中的应用
CN103965085B (zh) *	2014-04-17	2016-02-24	上海恒晟药业有限公司	一种取代1,2-氨基醇药物的制备方法
CN106278964B (zh) *	2016-07-31	2018-01-16	浙江润康药业有限公司	氟苯尼考的制备方法
CN111500652B (zh) *	2019-01-30	2024-03-26	苏州引航生物科技有限公司	一种制备氟苯尼考的方法
CN110302163A (zh) *	2019-07-23	2019-10-08	东莞正大康地饲料有限公司	一种氟苯尼考可溶性粉及其制备方法
CN110773207A (zh) *	2019-09-25	2020-02-11	陈红菊	一种在室温且无光条件下可完全分解甲醛的冷触媒材料及其制备方法
CN111423391A (zh) *	2020-03-18	2020-07-17	浙江康牧药业有限公司	一种氟苯尼考中间体的制备方法
CN113402475A (zh) *	2021-06-07	2021-09-17	山东国邦药业有限公司	一种氟苯尼考中间体的制备方法

Family Cites Families (8)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US4002637A (en) *	1973-07-09	1977-01-11	Rohm And Haas Company	Oxazolidine, oxazolidine-containing condensation and addition polymers and methods of producing them
EP0678506A3 (fr) *	1983-06-02	1996-07-24	Zambon Spa	Intermédiaires pour la préparation des dérivés de 1-phényl-1-hydroxy-2-amino-3-fluoropropane.
IT1237798B (it) *	1989-10-20	1993-06-17	Zambon Spa	Processo per l'inversione stereochimica di (2s,3s)-2-ammino-3-fenil-1 ,3-propandioli nei corrispondenti enantiomeri (2r,3r).
WO1994004523A1 (fr) *	1992-08-21	1994-03-03	Japan Tobacco Inc.	Compose dioxacycloalcane a activite inhibitrice de la renine
US5663361A (en) *	1996-08-19	1997-09-02	Schering Corporation	Process for preparing intermediates to florfenicol
JP2001240571A (ja) *	2000-03-01	2001-09-04	Udagawa Reiko	フッ素アルコールの製造方法
KR20040091698A (ko)	2002-03-08	2004-10-28	쉐링-플라우 리미티드.	신규한 플로르페니콜형 항생제
US7126005B2 (en) *	2003-10-06	2006-10-24	Aurobindo Pharma Limited	Process for preparing florfenicol

2006
- 2006-08-31 EP EP06824884.8A patent/EP1928820B1/fr active Active
- 2006-08-31 RU RU2008112950/04A patent/RU2008112950A/ru not_active Application Discontinuation
- 2006-08-31 UA UAA200804362A patent/UA93212C2/ru unknown
- 2006-08-31 CA CA002621971A patent/CA2621971A1/fr not_active Abandoned
- 2006-08-31 BR BRPI0615767-0A patent/BRPI0615767A2/pt not_active IP Right Cessation
- 2006-08-31 TW TW095132192A patent/TWI331139B/zh not_active IP Right Cessation
- 2006-08-31 SI SI200631769T patent/SI1928820T1/sl unknown
- 2006-08-31 MX MX2008003188A patent/MX2008003188A/es unknown
- 2006-08-31 WO PCT/US2006/034219 patent/WO2007030386A2/fr not_active Ceased
- 2006-08-31 KR KR1020087005954A patent/KR20080049040A/ko not_active Withdrawn
- 2006-08-31 KR KR1020087005920A patent/KR101408596B1/ko not_active Expired - Fee Related
- 2006-08-31 CA CA002621987A patent/CA2621987A1/fr not_active Abandoned
- 2006-08-31 MX MX2008003186A patent/MX2008003186A/es unknown
- 2006-08-31 AU AU2006287696A patent/AU2006287696A1/en not_active Abandoned
- 2006-08-31 RU RU2008112946/04A patent/RU2008112946A/ru not_active Application Discontinuation
- 2006-08-31 CN CNA2006800412359A patent/CN101300238A/zh active Pending
- 2006-08-31 JP JP2008530112A patent/JP2009507074A/ja not_active Withdrawn
- 2006-08-31 ES ES06824884.8T patent/ES2459205T3/es active Active
- 2006-08-31 JP JP2008530125A patent/JP5113754B2/ja not_active Expired - Fee Related
- 2006-08-31 WO PCT/US2006/034217 patent/WO2007030385A2/fr not_active Ceased
- 2006-08-31 CN CNA2006800410847A patent/CN101300237A/zh active Pending
- 2006-08-31 CA CA002621961A patent/CA2621961A1/fr not_active Abandoned
- 2006-08-31 US US11/515,135 patent/US7786329B2/en active Active
- 2006-08-31 AU AU2006287716A patent/AU2006287716A1/en not_active Abandoned
- 2006-08-31 BR BRPI0615565-0A patent/BRPI0615565A2/pt not_active IP Right Cessation
- 2006-08-31 CN CN2006800411958A patent/CN101300227B/zh active Active
- 2006-08-31 JP JP2008530111A patent/JP2009507842A/ja active Pending
- 2006-08-31 RU RU2008112952/04A patent/RU2008112952A/ru unknown
- 2006-08-31 EP EP06802794A patent/EP1934189A2/fr not_active Withdrawn
- 2006-08-31 BR BRPI0615764-5A patent/BRPI0615764A2/pt not_active IP Right Cessation
- 2006-08-31 KR KR1020087005952A patent/KR20080049039A/ko not_active Withdrawn
- 2006-08-31 MX MX2008003187A patent/MX2008003187A/es unknown
- 2006-08-31 US US11/515,278 patent/US20070055067A1/en not_active Abandoned
- 2006-08-31 WO PCT/US2006/034370 patent/WO2007030405A2/fr not_active Ceased
- 2006-08-31 TW TW095132200A patent/TW200800924A/zh unknown
- 2006-08-31 US US11/514,741 patent/US20070055066A1/en not_active Abandoned
- 2006-08-31 EP EP06802796A patent/EP1934190A2/fr not_active Withdrawn
- 2006-08-31 TW TW095132185A patent/TW200804253A/zh unknown
- 2006-08-31 AU AU2006287697A patent/AU2006287697A1/en not_active Abandoned
2008
- 2008-02-28 IL IL189828A patent/IL189828A0/en unknown
- 2008-02-28 IL IL189830A patent/IL189830A0/en unknown
- 2008-02-28 IL IL189829A patent/IL189829A0/en unknown
- 2008-03-04 ZA ZA200802047A patent/ZA200802047B/xx unknown
- 2008-03-04 ZA ZA200802048A patent/ZA200802048B/xx unknown
- 2008-03-04 ZA ZA200802046A patent/ZA200802046B/xx unknown
- 2008-03-13 EC EC2008008266A patent/ECSP088266A/es unknown
- 2008-03-13 EC EC2008008267A patent/ECSP088267A/es unknown
- 2008-03-13 EC EC2008008268A patent/ECSP088268A/es unknown
- 2008-04-04 NO NO20081686A patent/NO20081686L/no not_active Application Discontinuation
- 2008-04-04 NO NO20081685A patent/NO20081685L/no not_active Application Discontinuation
- 2008-04-04 NO NO20081684A patent/NO20081684L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
EP1928820B1 (fr)	2014-01-29
NO20081684L (no)	2008-06-05
EP1934190A2 (fr)	2008-06-25
TWI331139B (en)	2010-10-01
US20070055080A1 (en)	2007-03-08
KR20080041699A (ko)	2008-05-13
WO2007030385A2 (fr)	2007-03-15
MX2008003188A (es)	2008-03-18
ZA200802046B (en)	2008-12-31
RU2008112946A (ru)	2009-10-20
ECSP088266A (es)	2008-04-28
TW200800924A (en)	2008-01-01
EP1928820A2 (fr)	2008-06-11
JP2009507842A (ja)	2009-02-26
CN101300237A (zh)	2008-11-05
SI1928820T1 (sl)	2014-08-29
RU2008112952A (ru)	2009-10-20
CN101300227B (zh)	2013-07-03
IL189828A0 (en)	2008-11-03
CA2621961A1 (fr)	2007-03-15
JP2009507074A (ja)	2009-02-19
WO2007030386A2 (fr)	2007-03-15
US20070055066A1 (en)	2007-03-08
BRPI0615764A2 (pt)	2011-05-24
TW200804254A (en)	2008-01-16
JP5113754B2 (ja)	2013-01-09
UA93212C2 (ru)	2011-01-25
KR20080049039A (ko)	2008-06-03
KR101408596B1 (ko)	2014-06-17
NO20081685L (no)	2008-06-05
US7786329B2 (en)	2010-08-31
ZA200802048B (en)	2008-11-26
BRPI0615565A2 (pt)	2011-05-24
KR20080049040A (ko)	2008-06-03
US20070055067A1 (en)	2007-03-08
WO2007030386A3 (fr)	2007-05-24
BRPI0615767A2 (pt)	2011-05-24
AU2006287697A1 (en)	2007-03-15
CA2621971A1 (fr)	2007-03-15
EP1934189A2 (fr)	2008-06-25
IL189830A0 (en)	2008-11-03
WO2007030405A2 (fr)	2007-03-15
CA2621987A1 (fr)	2007-03-15
ZA200802047B (en)	2008-12-31
ECSP088267A (es)	2008-04-28
WO2007030385A3 (fr)	2007-05-24
MX2008003186A (es)	2008-03-18
CN101300238A (zh)	2008-11-05
WO2007030405A3 (fr)	2007-05-18
RU2008112950A (ru)	2009-10-20
AU2006287716A1 (en)	2007-03-15
ES2459205T3 (es)	2014-05-08
MX2008003187A (es)	2008-03-18
TW200804253A (en)	2008-01-16
CN101300227A (zh)	2008-11-05
JP2009507075A (ja)	2009-02-19
AU2006287696A1 (en)	2007-03-15
ECSP088268A (es)	2008-04-28
IL189829A0 (en)	2008-11-03

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Legal Events

Date	Code	Title	Description
2012-03-26	FC2A	Withdrawal, rejection or dismissal of laid open patent application