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NO20054371L - Somatostatin-dopamin kimaere analoger - Google Patents

Somatostatin-dopamin kimaere analoger

Info

Publication number
NO20054371L
NO20054371L NO20054371A NO20054371A NO20054371L NO 20054371 L NO20054371 L NO 20054371L NO 20054371 A NO20054371 A NO 20054371A NO 20054371 A NO20054371 A NO 20054371A NO 20054371 L NO20054371 L NO 20054371L
Authority
NO
Norway
Prior art keywords
somatostatin
dopamine chimeric
chimeric analogs
analogs
dopamine
Prior art date
Application number
NO20054371A
Other languages
English (en)
Norwegian (no)
Other versions
NO20054371D0 (no
Inventor
Yeelana Shen
Michael Dewitt Culler
Zheng Xin Dong
Original Assignee
Sod Conseils Rech Applic
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sod Conseils Rech Applic filed Critical Sod Conseils Rech Applic
Publication of NO20054371D0 publication Critical patent/NO20054371D0/no
Publication of NO20054371L publication Critical patent/NO20054371L/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07K—PEPTIDES
    • C07K14/00—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • C07K14/435—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • C07K14/575—Hormones
    • C07K14/655—Somatostatins
    • C07K14/6555—Somatostatins at least 1 amino acid in D-form
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
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    • A61K38/16—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof
    • A61K38/17—Peptides having more than 20 amino acids; Gastrins; Somatostatins; Melanotropins; Derivatives thereof from animals; from humans
    • A61K38/22—Hormones
    • A61K38/31—Somatostatins
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D265/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one oxygen atom as the only ring hetero atoms
    • C07D265/28—1,4-Oxazines; Hydrogenated 1,4-oxazines
    • C07D265/34—1,4-Oxazines; Hydrogenated 1,4-oxazines condensed with carbocyclic rings
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • C—CHEMISTRY; METALLURGY
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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/04—Ortho-condensed systems
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    • C07D513/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04—Ortho-condensed systems
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    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00—Medicinal preparations containing peptides
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    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
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  • Health & Medical Sciences (AREA)
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  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Engineering & Computer Science (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Immunology (AREA)
  • Hematology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Obesity (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Neurosurgery (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Urology & Nephrology (AREA)
  • Biochemistry (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biophysics (AREA)
  • Zoology (AREA)
  • Cardiology (AREA)
  • Epidemiology (AREA)
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NO20054371A 2003-04-11 2005-09-21 Somatostatin-dopamin kimaere analoger NO20054371L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US46237403P 2003-04-11 2003-04-11
PCT/US2004/010891 WO2004091490A2 (fr) 2003-04-11 2004-04-08 Analogues chimeres de la somatostatine-dopamine

Publications (2)

Publication Number Publication Date
NO20054371D0 NO20054371D0 (no) 2005-09-21
NO20054371L true NO20054371L (no) 2005-12-19

Family

ID=33299939

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20054371A NO20054371L (no) 2003-04-11 2005-09-21 Somatostatin-dopamin kimaere analoger

Country Status (19)

Country Link
US (2) US7517853B2 (fr)
EP (1) EP1617856B1 (fr)
JP (2) JP4579235B2 (fr)
KR (3) KR100795425B1 (fr)
CN (2) CN1771049A (fr)
AR (1) AR041769A1 (fr)
AU (1) AU2004229437B2 (fr)
BR (1) BRPI0409359A (fr)
CA (1) CA2521965A1 (fr)
ES (1) ES2450645T3 (fr)
IL (1) IL170742A0 (fr)
MX (1) MXPA05010868A (fr)
NO (1) NO20054371L (fr)
NZ (2) NZ542297A (fr)
RU (1) RU2329273C2 (fr)
SG (1) SG175448A1 (fr)
TW (2) TWI350838B (fr)
WO (1) WO2004091490A2 (fr)
ZA (1) ZA200508145B (fr)

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* Cited by examiner, † Cited by third party
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KR100795425B1 (ko) * 2003-04-11 2008-01-17 소시에떼 더 콘세이유 더 레세르세 에 다플리까띠옹 시엔띠피끄, 에스.아.에스. 소마토스타틴-도파민 키메라 유사체
ATE536368T1 (de) * 2006-10-20 2011-12-15 Ipsen Pharma Sas Konjugate von zytotoxischen verbindungen mit peptiden
GB0721333D0 (en) * 2007-10-31 2007-12-12 Motac Neuroscience Ltd Medicaments
EP2296687A4 (fr) * 2008-05-14 2012-12-26 Ipsen Pharma Sas Compositions pharmaceutiques de conjugués somatostatine-dopamine
WO2011104627A1 (fr) 2010-02-24 2011-09-01 Ipsen Pharma S.A.S. Métabolites de dop2-d-lys(dop2)-cyclo[cys-tyr-d-trp-lys-abu-cys]-thr-nh2
RU2457215C1 (ru) * 2011-04-07 2012-07-27 Закрытое Акционерное Общество "Фарм-Синтез" Октапептид для получения радиофармацевтических средств, радиофармацевтическое средство на его основе и способ диагностики опухолей, экспрессирующих соматостатиновые рецепторы
ES2663869T3 (es) * 2011-12-23 2018-04-17 Ipsen Manufacturing Ireland Limited Procedimiento para la síntesis de análogos de la grelina
CN102898397B (zh) * 2012-09-26 2014-12-10 江苏华益科技有限公司 (4aR,10bR)-3,4,4a,5,6,10b-六氢-2H-萘并[1,2-b][1,4]噁嗪-9-醇类物质及其盐酸盐合成方法
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SG175448A1 (en) 2011-11-28
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EP1617856B1 (fr) 2014-01-15
AR041769A1 (es) 2005-06-01
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AU2004229437B2 (en) 2007-12-06
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