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NO20052761L - Spirocykliske cykloheksanderivater. - Google Patents

Spirocykliske cykloheksanderivater.

Info

Publication number
NO20052761L
NO20052761L NO20052761A NO20052761A NO20052761L NO 20052761 L NO20052761 L NO 20052761L NO 20052761 A NO20052761 A NO 20052761A NO 20052761 A NO20052761 A NO 20052761A NO 20052761 L NO20052761 L NO 20052761L
Authority
NO
Norway
Prior art keywords
cyclohexane derivatives
spirocyclic cyclohexane
spirocyclic
preparation
derivatives
Prior art date
Application number
NO20052761A
Other languages
English (en)
Other versions
NO20052761D0 (no
NO331818B1 (no
Inventor
Babette-Yvonne Koegel
Bernd Sundermann
Elmar Josef Friderichs
Claudia Hinze
Otto Aulenbacher
Stefan Oberboersch
Werner Engelberger
Klaus Linz
Hans Schick
Helmut Sonnenschein
Birgitta Henkel
Valerie Sarah Rose
Michael Jonathan Lipkin
Original Assignee
Gruenenthal Gmbh
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=32185555&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=NO20052761(L) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Gruenenthal Gmbh filed Critical Gruenenthal Gmbh
Publication of NO20052761L publication Critical patent/NO20052761L/no
Publication of NO20052761D0 publication Critical patent/NO20052761D0/no
Publication of NO331818B1 publication Critical patent/NO331818B1/no

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/10—Spiro-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04—Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • A—HUMAN NECESSITIES
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00—Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/14—Prodigestives, e.g. acids, enzymes, appetite stimulants, antidyspeptics, tonics, antiflatulents
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • A—HUMAN NECESSITIES
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    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C309/04—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing only one sulfo group
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C309/00—Sulfonic acids; Halides, esters, or anhydrides thereof
    • C07C309/01—Sulfonic acids
    • C07C309/02—Sulfonic acids having sulfo groups bound to acyclic carbon atoms
    • C07C309/03—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
    • C07C309/06—Sulfonic acids having sulfo groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton containing halogen atoms, or nitro or nitroso groups bound to the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/235—Saturated compounds containing more than one carboxyl group
    • C07C59/245—Saturated compounds containing more than one carboxyl group containing hydroxy or O-metal groups
    • C07C59/255—Tartaric acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/235—Saturated compounds containing more than one carboxyl group
    • C07C59/245—Saturated compounds containing more than one carboxyl group containing hydroxy or O-metal groups
    • C07C59/265—Citric acid
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
    • C07D491/02—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00 in which the condensed system contains two hetero rings
    • C07D491/10—Spiro-condensed systems
    • C07D491/107—Spiro-condensed systems with only one oxygen atom as ring hetero atom in the oxygen-containing ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D493/00—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system
    • C07D493/02—Heterocyclic compounds containing oxygen atoms as the only ring hetero atoms in the condensed system in which the condensed system contains two hetero rings
    • C07D493/10—Spiro-condensed systems
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D495/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms
    • C07D495/02—Heterocyclic compounds containing in the condensed system at least one hetero ring having sulfur atoms as the only ring hetero atoms in which the condensed system contains two hetero rings
    • C07D495/10—Spiro-condensed systems

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  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
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  • Neurology (AREA)
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  • Pain & Pain Management (AREA)
  • Addiction (AREA)
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  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Anesthesiology (AREA)
  • Urology & Nephrology (AREA)
  • Reproductive Health (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Endocrinology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Dermatology (AREA)
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  • Psychology (AREA)
  • Nutrition Science (AREA)
  • Gynecology & Obstetrics (AREA)
  • Child & Adolescent Psychology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Det er beskrevet spirosykliske sykloheksanderivater, fremgangsmåter for deres fremstilling, legemidler inneholdende disse forbindelsene og anvendelsen av spirosykliske sykloheksanderivater for fremstilling av legemidler.
NO20052761A 2002-11-11 2005-06-07 Spirosykliske sykloheksanderivater, fremgangsmater for fremstilling derav, anvendelse derav samt medikament inneholdende minst en slik forbindelse. NO331818B1 (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE2002152667 DE10252667A1 (de) 2002-11-11 2002-11-11 Spirocyclische Cyclohexan-Derivate
PCT/EP2003/012305 WO2004043967A1 (de) 2002-11-11 2003-11-05 Spirocyclische cyclohexan-derivate

Publications (3)

Publication Number Publication Date
NO20052761L true NO20052761L (no) 2005-06-07
NO20052761D0 NO20052761D0 (no) 2005-06-07
NO331818B1 NO331818B1 (no) 2012-04-10

Family

ID=32185555

Family Applications (2)

Application Number Title Priority Date Filing Date
NO20052761A NO331818B1 (no) 2002-11-11 2005-06-07 Spirosykliske sykloheksanderivater, fremgangsmater for fremstilling derav, anvendelse derav samt medikament inneholdende minst en slik forbindelse.
NO20093060A NO331776B1 (no) 2002-11-11 2009-09-24 Spirosykliske sykloheksanderivater, fremgangsmater for fremstilling derav, anvendelse derav samt medikamenter inneholdende derivatene.

Family Applications After (1)

Application Number Title Priority Date Filing Date
NO20093060A NO331776B1 (no) 2002-11-11 2009-09-24 Spirosykliske sykloheksanderivater, fremgangsmater for fremstilling derav, anvendelse derav samt medikamenter inneholdende derivatene.

Country Status (27)

Country Link
US (6) US7547707B2 (no)
EP (4) EP1560835B1 (no)
JP (4) JP4728645B2 (no)
KR (2) KR101075817B1 (no)
CN (2) CN100577664C (no)
AR (2) AR041932A1 (no)
AT (1) ATE441650T1 (no)
AU (2) AU2003296563B2 (no)
BR (2) BRPI0318811B8 (no)
CA (1) CA2505555C (no)
CO (1) CO5580765A2 (no)
CY (2) CY1110558T1 (no)
DE (2) DE10252667A1 (no)
DK (2) DK1560835T3 (no)
EC (1) ECSP055786A (no)
ES (4) ES2587185T3 (no)
IL (2) IL168473A (no)
MX (1) MXPA05004959A (no)
NO (2) NO331818B1 (no)
NZ (1) NZ540575A (no)
PE (1) PE20040830A1 (no)
PL (2) PL215227B1 (no)
PT (2) PT2062898E (no)
RU (1) RU2354656C2 (no)
SI (2) SI1560835T1 (no)
WO (1) WO2004043967A1 (no)
ZA (1) ZA200504725B (no)

Families Citing this family (101)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US7776314B2 (en) 2002-06-17 2010-08-17 Grunenthal Gmbh Abuse-proofed dosage system
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EP1560835B1 (de) 2009-09-02
HK1130491A1 (en) 2009-12-31
DK2062898T3 (da) 2013-10-28
PE20040830A1 (es) 2004-11-17
CN1735619A (zh) 2006-02-15
BRPI0318811B8 (pt) 2021-05-25
EP2062898A2 (de) 2009-05-27
PL390420A1 (pl) 2010-04-26
IL203141A (en) 2012-04-30
EP2233487A1 (de) 2010-09-29
SI2062898T1 (sl) 2013-11-29
EP2116544B1 (de) 2016-05-18
EP2116544A3 (de) 2010-09-22
JP2006508114A (ja) 2006-03-09
CN101693714A (zh) 2010-04-14
RU2354656C2 (ru) 2009-05-10
AU2003296563A1 (en) 2004-06-03
JP5442565B2 (ja) 2014-03-12
NO331776B1 (no) 2012-03-26
JP5539821B2 (ja) 2014-07-02
US20090163716A1 (en) 2009-06-25
CN100577664C (zh) 2010-01-06
SI1560835T1 (sl) 2010-01-29
ATE441650T1 (de) 2009-09-15
ES2587013T3 (es) 2016-10-20
NO20093060L (no) 2005-06-07
PL217804B1 (pl) 2014-08-29
EP2116544A2 (de) 2009-11-11
CY1114616T1 (el) 2016-10-05
AU2003296563B2 (en) 2010-03-11
HK1146044A1 (zh) 2011-05-13
US8053576B2 (en) 2011-11-08
US7799931B2 (en) 2010-09-21
ES2333956T3 (es) 2010-03-03
CA2505555A1 (en) 2004-05-27
BR0315296A (pt) 2005-08-30
JP4728645B2 (ja) 2011-07-20
ES2587185T3 (es) 2016-10-21
NO331818B1 (no) 2012-04-10
BRPI0315296B1 (pt) 2018-10-09
US9120797B2 (en) 2015-09-01
AU2010200219A1 (en) 2010-02-11
DE10252667A1 (de) 2004-05-27
CY1110558T1 (el) 2015-04-29

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