NO20053201D0 - Nye heterocykliske fluorglukosidderivater, legemidler inneholdende disse forbindelser og deres anvendelse. - Google Patents

Nye heterocykliske fluorglukosidderivater, legemidler inneholdende disse forbindelser og deres anvendelse.

Info

Publication number: NO20053201D0
Authority: NO; Norway
Prior art keywords: fluoroglucose; derivatives; compounds; drugs containing; new heterocyclic
Prior art date: 2002-12-12

Application number

NO20053201A

Other languages

English (en)

Other versions

NO20053201L (no

NO330299B1 (no

Inventor

Heiner Glombik

Hubert Heuer

Werner Kramer

Wendelin Frick

Harm Brummerhop

Oliver Plettenburg

Original Assignee

Aventis Pharma Gmbh

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

2002-12-12

Filing date

2005-06-30

Publication date

2005-06-30

2005-06-30 Application filed by Aventis Pharma Gmbh filed Critical Aventis Pharma Gmbh

2005-06-30 Publication of NO20053201D0 publication Critical patent/NO20053201D0/no

2005-08-04 Publication of NO20053201L publication Critical patent/NO20053201L/no

2011-03-28 Publication of NO330299B1 publication Critical patent/NO330299B1/no

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
- C07H17/02—Heterocyclic radicals containing only nitrogen as ring hetero atoms
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/70—Carbohydrates; Sugars; Derivatives thereof
- A61K31/7042—Compounds having saccharide radicals and heterocyclic rings
- A61K31/7052—Compounds having saccharide radicals and heterocyclic rings having nitrogen as a ring hetero atom, e.g. nucleosides, nucleotides
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P13/00—Drugs for disorders of the urinary system
- A61P13/12—Drugs for disorders of the urinary system of the kidneys
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A61P17/06—Antipsoriatics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P19/00—Drugs for skeletal disorders
- A61P19/08—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease
- A61P19/10—Drugs for skeletal disorders for bone diseases, e.g. rachitism, Paget's disease for osteoporosis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/04—Anorexiants; Antiobesity agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P3/00—Drugs for disorders of the metabolism
- A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
- A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/10—Antimycotics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/18—Antivirals for RNA viruses for HIV
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P35/00—Antineoplastic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P37/00—Drugs for immunological or allergic disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P5/00—Drugs for disorders of the endocrine system
- A61P5/48—Drugs for disorders of the endocrine system of the pancreatic hormones
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
- C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals

Landscapes

Health & Medical Sciences (AREA)
Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
General Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Medicinal Chemistry (AREA)
Pharmacology & Pharmacy (AREA)
Animal Behavior & Ethology (AREA)
Public Health (AREA)
Veterinary Medicine (AREA)
Chemical Kinetics & Catalysis (AREA)
General Chemical & Material Sciences (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Bioinformatics & Cheminformatics (AREA)
Diabetes (AREA)
Molecular Biology (AREA)
Genetics & Genomics (AREA)
Biotechnology (AREA)
Biochemistry (AREA)
Hematology (AREA)
Obesity (AREA)
Biomedical Technology (AREA)
Neurology (AREA)
Neurosurgery (AREA)
Physical Education & Sports Medicine (AREA)
Endocrinology (AREA)
Rheumatology (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Virology (AREA)
Heart & Thoracic Surgery (AREA)
Urology & Nephrology (AREA)
Cardiology (AREA)
Orthopedic Medicine & Surgery (AREA)
Pulmonology (AREA)
Emergency Medicine (AREA)
Psychiatry (AREA)
Hospice & Palliative Care (AREA)
Child & Adolescent Psychology (AREA)

NO20053201A 2002-12-12 2005-06-30 Heterocykliske fluorglukosidderivater, anvendelser derav, legemidler inneholdende forbindelsene samt fremgangsmate for fremstilling av legemidlene. NO330299B1 (no)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE10258008A DE10258008B4 (de)	2002-12-12	2002-12-12	Heterocyclische Fluorglycosidderivate, diese Verbindungen enthaltende Arzneimittel und Verfahren zur Herstellung dieser Arzneimittel
PCT/EP2003/013455 WO2004052903A1 (de)	2002-12-12	2003-11-28	Neue heterocyclische fluorglykosidderivate, diese verbindungen enthaltende arzneimittel und deren verwendung

Publications (3)

Publication Number	Publication Date
NO20053201D0 true NO20053201D0 (no)	2005-06-30
NO20053201L NO20053201L (no)	2005-08-04
NO330299B1 NO330299B1 (no)	2011-03-28

Family

ID=32477575

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
NO20053201A NO330299B1 (no)	2002-12-12	2005-06-30	Heterocykliske fluorglukosidderivater, anvendelser derav, legemidler inneholdende forbindelsene samt fremgangsmate for fremstilling av legemidlene.

Country Status (42)

Country	Link
US (2)	US20040259819A1 (no)
EP (1)	EP1572708B1 (no)
JP (1)	JP4806193B2 (no)
KR (1)	KR101160061B1 (no)
CN (1)	CN1304406C (no)
AR (1)	AR042437A1 (no)
AT (1)	ATE323713T1 (no)
AU (1)	AU2003289911B2 (no)
BR (1)	BR0317283A (no)
CA (1)	CA2508226C (no)
CR (1)	CR7820A (no)
CY (1)	CY1105621T1 (no)
DE (2)	DE10258008B4 (no)
DK (1)	DK1572708T3 (no)
EC (1)	ECSP055853A (no)
ES (1)	ES2261993T3 (no)
GT (1)	GT200300268A (no)
HN (1)	HN2003000408A (no)
HR (1)	HRP20050532A2 (no)
IL (1)	IL168876A (no)
JO (1)	JO2353B1 (no)
MA (1)	MA27560A1 (no)
ME (1)	MEP40908A (no)
MX (1)	MXPA05005821A (no)
MY (1)	MY139302A (no)
NO (1)	NO330299B1 (no)
NZ (1)	NZ540695A (no)
OA (1)	OA12972A (no)
PA (1)	PA8592301A1 (no)
PE (1)	PE20040771A1 (no)
PL (1)	PL212080B1 (no)
PT (1)	PT1572708E (no)
RS (1)	RS50908B (no)
RU (1)	RU2339641C2 (no)
SI (1)	SI1572708T1 (no)
SV (1)	SV2004001690A (no)
TN (1)	TNSN05160A1 (no)
TW (1)	TWI320044B (no)
UA (1)	UA81136C2 (no)
UY (1)	UY28122A1 (no)
WO (1)	WO2004052903A1 (no)
ZA (1)	ZA200503365B (no)

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US7723309B2 (en)	2005-05-03	2010-05-25	Boehringer Ingelheim International Gmbh	Crystalline forms of 1-chloro-4-(β-D-glucopyranos-1-yl)-2-[4-((R)-tetrahydrofuran-3-yloxy)-benzyl]-benzene, a method for its preparation and the use thereof for preparing medicaments
US7772191B2 (en)	2005-05-10	2010-08-10	Boehringer Ingelheim International Gmbh	Processes for preparing of glucopyranosyl-substituted benzyl-benzene derivatives and intermediates therein
DE102005026762A1 (de)	2005-06-09	2006-12-21	Sanofi-Aventis Deutschland Gmbh	Azolopyridin-2-on-derivate als Inhibitoren von Lipasen und Phospholipasen
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JP5175191B2 (ja)	2005-08-30	2013-04-03	ベーリンガーインゲルハイムインターナショナルゲゼルシャフトミットベシュレンクテルハフツング	グリコピラノシル置換ベンジルベンゼン誘導体、該化合物を含有する医薬品及びその使用と製造方法
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Publication number	Publication date
CR7820A (es)	2008-11-25
ES2261993T3 (es)	2006-11-16
NO20053201L (no)	2005-08-04
UA81136C2 (en)	2007-12-10
RS20050432A (sr)	2007-06-04
WO2004052903A1 (de)	2004-06-24
MA27560A1 (fr)	2005-10-03
CN1723214A (zh)	2006-01-18
JP2006510644A (ja)	2006-03-30
NO330299B1 (no)	2011-03-28
PE20040771A1 (es)	2005-01-21
PL375790A1 (en)	2005-12-12
SI1572708T1 (sl)	2006-08-31
EP1572708A1 (de)	2005-09-14
HK1084123A1 (en)	2006-07-21
JP4806193B2 (ja)	2011-11-02
HRP20050532A2 (en)	2006-09-30
UY28122A1 (es)	2004-07-30
EP1572708B1 (de)	2006-04-19
MEP40908A (en)	2011-02-10
ATE323713T1 (de)	2006-05-15
AU2003289911A1 (en)	2004-06-30
HN2003000408A (es)	2006-01-07
ECSP055853A (es)	2005-09-20
KR20050085482A (ko)	2005-08-29
CY1105621T1 (el)	2010-12-22
ZA200503365B (en)	2006-11-29
GT200300268A (es)	2004-03-03
TNSN05160A1 (en)	2007-05-14
MXPA05005821A (es)	2005-08-29
CN1304406C (zh)	2007-03-14
US20100261664A1 (en)	2010-10-14
DK1572708T3 (da)	2006-08-21
JO2353B1 (en)	2006-12-12
RS50908B (sr)	2010-08-31
AR042437A1 (es)	2005-06-22
OA12972A (en)	2006-10-13
AU2003289911B2 (en)	2009-09-17
TW200418870A (en)	2004-10-01
IL168876A (en)	2010-06-30
KR101160061B1 (ko)	2012-06-26
BR0317283A (pt)	2005-11-08
US20040259819A1 (en)	2004-12-23
DE10258008B4 (de)	2006-02-02
NZ540695A (en)	2007-02-23
CA2508226A1 (en)	2004-06-24
DE10258008A1 (de)	2004-07-08
MY139302A (en)	2009-09-30
PT1572708E (pt)	2006-07-31
RU2339641C2 (ru)	2008-11-27
CA2508226C (en)	2011-12-20
DE50303067D1 (de)	2006-05-24
RU2005121893A (ru)	2006-01-20
PA8592301A1 (es)	2004-07-26
PL212080B1 (pl)	2012-08-31
TWI320044B (en)	2010-02-01
SV2004001690A (es)	2004-03-19

Publication	Publication Date	Title
NO20053201D0 (no)	2005-06-30	Nye heterocykliske fluorglukosidderivater, legemidler inneholdende disse forbindelser og deres anvendelse.
DK1523488T3 (da)	2009-03-16	Nye thiophenglycosidderivater, fremgangsmåder til deres fremstilling, lægemidler indeholdende disse forbindelser og deres anvendelse
DK1572707T3 (da)	2006-08-14	Hidtil ukendte aromatiske fluorglycosidderivater, lægemidler indeholdende disse forbindelser og anvendelse heraf
NO20052855D0 (no)	2005-06-13	Fosfonoksykinazolinderivater og farmasoytisk anvendelse derav.
NO20053356D0 (no)	2005-07-11	Aminindazolderivater og anvendelse derav som kinaseinhibitorer.
NO20043733L (no)	2004-10-20	Aryl-5-tio-Β-D-glukopyranosid-derivater og legemidler for diabetes inneholdende de samme
NO20052496D0 (no)	2005-05-24	Selekterte CGRP antagonister, fremgangsmater for fremstilling derav og anvendelse derav som medikamenter.
DK1558578T3 (da)	2013-06-17	Nye Alkynforbindelser med MCH-antagonistisk virkning og lægemiddel indeholdende disse forbindelser.
DK1400518T3 (da)	2007-03-26	Heterocycliske forbindelser og lægemidler
DK1562946T3 (da)	2010-09-20	Nye xanthinderivater, deres fremstilling og deres anvendelse som lægemiddel
DK1758914T3 (da)	2008-03-17	Hidtil ukendte fluorglycosidderivater af pyrazoler, lægemidler indeholdende disse forbindelser og anvendelse heraf
DK1730131T3 (da)	2012-08-13	Glucopyranosyl-substituerede benzol-derivater, lægemiddel indeholdende disse forbindelser, deres anvendelse og fremgangsmåder til deres fremstilling
NO20021689L (no)	2002-05-30	5-leddede heterocykliske derivater, fremstilling derav og anvendelse som medikamenter
NO20054244D0 (no)	2005-09-13	Nitrogeninneholdende heterocykliske derivater og legemidler inneholdende de samme som den aktive bestanddel
NO20051645L (no)	2005-05-19	Nye aminoindozolderivater som medisin og farmakologiske preparater inneholdende disse
DK1581532T3 (da)	2010-08-16	Pyrazolo-3,4-B pyridinforbindelser og deres anvendelse som phosphodiesterase inhibitorer
NO20024742D0 (no)	2002-10-02	Heterocykliske forbindelser, deres fremstilling og anvendelse
NO20030302D0 (no)	2003-01-20	Nye heteroarylderivater og deres anvendelse som medikamenter
NO20045064L (no)	2005-02-23	Indol-, azaindol- og beslektede heterocykliske 4-alkenyl-piperidin-amider
DK1500654T3 (da)	2006-06-06	Benzoxazinonderivater, fremstilling deraf og anvendelse deraf som lægemidler
DK1511734T3 (da)	2010-08-02	Forbindelser, præparater og fremgangsmåder
DK1674456T3 (da)	2008-10-27	Nye 1,4-benzothiazepin-1,1-dioxid-derivater med forbedrede egenskaber, fremgangsmåde til deres fremstilling, lægemidler indeholdende disse forbindelser og deres anvendelse
DK1603915T3 (da)	2010-08-30	Substituerede 8-pyridinyl-dihydrospiro-cycloalkyl-pyrimido- 1,2-a-pyrimidin-6-on og 8-pyrimidinyl-dihydrospiro-cycloalkyl-pyrimido-1,2-a-pyrimidin-6-on-derivater og deres anvendelse mod neurogenerative sygdomme
DK2107069T3 (da)	2013-04-15	Nye insulinderivater
NO20043349L (no)	2004-10-05	Kumarinderivater, fremgangsmate for deres framstilling og anvendelse derav

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