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NO20050164L - Nye quinuklidin-amid-derivater - Google Patents

Nye quinuklidin-amid-derivater

Info

Publication number
NO20050164L
NO20050164L NO20050164A NO20050164A NO20050164L NO 20050164 L NO20050164 L NO 20050164L NO 20050164 A NO20050164 A NO 20050164A NO 20050164 A NO20050164 A NO 20050164A NO 20050164 L NO20050164 L NO 20050164L
Authority
NO
Norway
Prior art keywords
amide derivatives
chj
well
quinuclidine amide
new quinuclidine
Prior art date
Application number
NO20050164A
Other languages
English (en)
Inventor
Maria Prat Quinones
Original Assignee
Almirall Prodesfarma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Almirall Prodesfarma Ag filed Critical Almirall Prodesfarma Ag
Publication of NO20050164L publication Critical patent/NO20050164L/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/08Bridged systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/02Drugs for disorders of the nervous system for peripheral neuropathies
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D453/00Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids
    • C07D453/02Heterocyclic compounds containing quinuclidine or iso-quinuclidine ring systems, e.g. quinine alkaloids containing not further condensed quinuclidine ring systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Urology & Nephrology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)

Abstract

Nye kvinuklidinamidderivater som har den kjemiske struktur med generell formel (I) (I) samt farmasøytisk akseptable salter derav innbefattende kvaternære salter av formel (II) (II) Ri Rfi¿(CHJ¿-A- {CHJ¿¿NtvcH.W X \<CHJ7 S er beskrevet, så vel som fremgangsmåter for deres fremstilling, farmasøytiske sammensetninger omfattende disse og deres bruk i terapi som antagonister for M3 muskarine reseptorer.
NO20050164A 2002-07-02 2005-01-12 Nye quinuklidin-amid-derivater NO20050164L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
ES200201539A ES2204295B1 (es) 2002-07-02 2002-07-02 Nuevos derivados de quinuclidina-amida.
PCT/EP2003/006708 WO2004005285A1 (en) 2002-07-02 2003-06-25 New quinuclidine amide derivatives

Publications (1)

Publication Number Publication Date
NO20050164L true NO20050164L (no) 2005-04-04

Family

ID=30011350

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20050164A NO20050164L (no) 2002-07-02 2005-01-12 Nye quinuklidin-amid-derivater

Country Status (24)

Country Link
US (2) US7488735B2 (no)
EP (1) EP1519933B1 (no)
JP (1) JP2005533826A (no)
CN (1) CN100404533C (no)
AR (1) AR040351A1 (no)
AT (1) ATE467631T1 (no)
AU (1) AU2003242757B2 (no)
BR (1) BR0312216A (no)
CA (1) CA2492535A1 (no)
DE (1) DE60332534D1 (no)
EC (1) ECSP045519A (no)
ES (1) ES2204295B1 (no)
IL (1) IL165923A (no)
MX (1) MXPA04012271A (no)
MY (1) MY130803A (no)
NO (1) NO20050164L (no)
NZ (1) NZ537341A (no)
PE (1) PE20040644A1 (no)
RU (1) RU2314306C2 (no)
TW (1) TW200402420A (no)
UA (1) UA80832C2 (no)
UY (1) UY27870A1 (no)
WO (1) WO2004005285A1 (no)
ZA (1) ZA200410404B (no)

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Also Published As

Publication number Publication date
CN100404533C (zh) 2008-07-23
US20080234316A1 (en) 2008-09-25
RU2005102585A (ru) 2005-10-10
BR0312216A (pt) 2005-04-12
MY130803A (en) 2007-07-31
ATE467631T1 (de) 2010-05-15
ES2204295B1 (es) 2005-08-01
US7488735B2 (en) 2009-02-10
CN1678610A (zh) 2005-10-05
DE60332534D1 (de) 2010-06-24
ES2204295A1 (es) 2004-04-16
ECSP045519A (es) 2005-03-10
RU2314306C2 (ru) 2008-01-10
AU2003242757B2 (en) 2009-01-08
WO2004005285A1 (en) 2004-01-15
PE20040644A1 (es) 2004-09-18
UA80832C2 (en) 2007-11-12
AU2003242757A1 (en) 2004-01-23
MXPA04012271A (es) 2005-04-08
CA2492535A1 (en) 2004-01-15
ZA200410404B (en) 2005-09-05
JP2005533826A (ja) 2005-11-10
UY27870A1 (es) 2003-10-31
EP1519933B1 (en) 2010-05-12
NZ537341A (en) 2006-04-28
IL165923A (en) 2010-06-30
US7718670B2 (en) 2010-05-18
EP1519933A1 (en) 2005-04-06
AR040351A1 (es) 2005-03-30
US20060167042A1 (en) 2006-07-27
TW200402420A (en) 2004-02-16
IL165923A0 (en) 2006-01-15

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