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NO20033540D0 - 6-substituerte pyrido-pyrimidiner - Google Patents

6-substituerte pyrido-pyrimidiner

Info

Publication number
NO20033540D0
NO20033540D0 NO20033540A NO20033540A NO20033540D0 NO 20033540 D0 NO20033540 D0 NO 20033540D0 NO 20033540 A NO20033540 A NO 20033540A NO 20033540 A NO20033540 A NO 20033540A NO 20033540 D0 NO20033540 D0 NO 20033540D0
Authority
NO
Norway
Prior art keywords
pyrimidines
substituted pyrido
pyrido
substituted
Prior art date
Application number
NO20033540A
Other languages
English (en)
Other versions
NO326133B1 (no
NO20033540L (no
Inventor
Jeffrey Jian Chen
James Patrick Dunn
David Michael Goldstein
Christophe Martin Stahl
Original Assignee
Hoffmann La Roche
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Hoffmann La Roche filed Critical Hoffmann La Roche
Publication of NO20033540L publication Critical patent/NO20033540L/no
Publication of NO20033540D0 publication Critical patent/NO20033540D0/no
Publication of NO326133B1 publication Critical patent/NO326133B1/no

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04Ortho-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/04Drugs for disorders of the alimentary tract or the digestive system for ulcers, gastritis or reflux esophagitis, e.g. antacids, inhibitors of acid secretion, mucosal protectants
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00Drugs for disorders of the respiratory system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P17/00Drugs for dermatological disorders
    • A61P17/06Antipsoriatics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P19/00Drugs for skeletal disorders
    • A61P19/02Drugs for skeletal disorders for joint disorders, e.g. arthritis, arthrosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/28Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00Drugs for immunological or allergic disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurosurgery (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Dermatology (AREA)
  • Rheumatology (AREA)
  • Immunology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Hospice & Palliative Care (AREA)
  • Cardiology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
NO20033540A 2001-02-12 2003-08-11 6-substituerte pyrido-pyrimidiner, fremgangsmate for fremstilling av slike, farmasoytiske preparater inneholdende slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom NO326133B1 (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US26837501P 2001-02-12 2001-02-12
US33465401P 2001-11-30 2001-11-30
PCT/EP2002/001106 WO2002064594A2 (en) 2001-02-12 2002-02-04 6-substituted pyrido-pyrimidines

Publications (3)

Publication Number Publication Date
NO20033540L NO20033540L (no) 2003-08-11
NO20033540D0 true NO20033540D0 (no) 2003-08-11
NO326133B1 NO326133B1 (no) 2008-10-06

Family

ID=26953040

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20033540A NO326133B1 (no) 2001-02-12 2003-08-11 6-substituerte pyrido-pyrimidiner, fremgangsmate for fremstilling av slike, farmasoytiske preparater inneholdende slike samt anvendelse av slike for fremstilling av medikament for behandling av sykdom

Country Status (31)

Country Link
US (3) US6696566B2 (no)
EP (1) EP1361880B1 (no)
JP (1) JP4064818B2 (no)
KR (1) KR100639772B1 (no)
CN (1) CN100376571C (no)
AR (1) AR035854A1 (no)
AT (1) ATE305303T1 (no)
AU (1) AU2002256615B2 (no)
BR (1) BRPI0207172B8 (no)
CA (1) CA2434834C (no)
CZ (1) CZ20032416A3 (no)
DE (1) DE60206363T2 (no)
DK (1) DK1361880T3 (no)
ES (1) ES2249574T3 (no)
HR (1) HRP20030624B1 (no)
HU (1) HU229604B1 (no)
IL (2) IL156872A0 (no)
JO (1) JO2410B1 (no)
MA (1) MA26993A1 (no)
MX (1) MXPA03007166A (no)
MY (1) MY131518A (no)
NO (1) NO326133B1 (no)
NZ (1) NZ526961A (no)
PA (1) PA8539201A1 (no)
PE (1) PE20020976A1 (no)
PL (1) PL366918A1 (no)
RU (1) RU2269527C2 (no)
SK (1) SK11322003A3 (no)
WO (1) WO2002064594A2 (no)
YU (1) YU63703A (no)
ZA (1) ZA200305938B (no)

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PL218692B1 (pl) 2002-01-22 2015-01-30 Warner Lambert Co Podstawiony 2-(pirydyn-2-yloamino)pirydo[2,3-d]pirymidyn-7-on oraz jego zastosowanie do leczenia zaburzenia lub stanu spowodowanego nieprawidłową proliferacją komórek
JP2006503802A (ja) 2002-04-03 2006-02-02 エフ.ホフマン−ラ ロシュ アーゲー イミダゾ縮合化合物
JP4252534B2 (ja) 2002-08-06 2009-04-08 エフ.ホフマン−ラ ロシュ アーゲー p−38MAPキナーゼインヒビターとしての6−アルコキシ−ピリド−ピリミジン類
JP2006516548A (ja) 2002-12-30 2006-07-06 アンジオテック インターナショナル アクツィエン ゲゼルシャフト 迅速ゲル化ポリマー組成物からの薬物送達法
WO2004076412A2 (en) * 2003-02-26 2004-09-10 Sugen, Inc. Aminoheteroaryl compounds as protein kinase inhibitors
BRPI0409405A (pt) * 2003-04-16 2006-04-25 Hoffmann La Roche compostos 7-aza-quinazolina substituìdos
EP1685131B1 (en) * 2003-11-13 2007-03-07 F. Hoffmann-La Roche AG Hydroxyalkyl substituted pyrido-7-pyrimidin-7-ones
US20090131430A1 (en) * 2004-11-23 2009-05-21 Palle Venkata P Pyrido'2,3-dipyrimidines as anti-inflammatory agents
US20060142312A1 (en) * 2004-12-23 2006-06-29 Pfizer Inc C6-aryl and heteroaryl substituted pyrido[2,3-D] pyrimidin-7-ones
US20090036472A1 (en) * 2005-02-02 2009-02-05 Palle Venkata P Azabicyclo derivatives as anti-inflammatory agents
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ATE449097T1 (de) * 2005-07-21 2009-12-15 Hoffmann La Roche Pyridoä2,3-düpyrimidin-2,4-diamin-verbindungen als ptpib-hemmer
ES2351939T3 (es) * 2005-08-09 2011-02-14 Irm Llc Compuestos y composiciones como inhibidores de proteínas cinasas.
EP1917245A1 (de) 2005-08-21 2008-05-07 Abbott GmbH & Co. KG Heterocyclische verbindungen und ihre verwendung als bindungspartner für 5-ht5-rezeptoren
JO2783B1 (en) * 2005-09-30 2014-03-15 نوفارتيس ايه جي Compounds 2-Amino-7, 8-dihydro-6H-Bayredo (3,4-D) Pyrimidine-5-Ones
AU2007268749B2 (en) * 2006-05-26 2012-07-26 Taisho Pharmaceutical Co., Ltd. Novel heterocyclic compound or salt thereof and intermediate thereof
WO2008150260A1 (en) * 2007-06-06 2008-12-11 Gpc Biotech, Inc. 8-oxy-2-aminopyrido (2, 3-d) pyrimidin-7-one derivatives as kinase inhibitors and anticancer agents
WO2008078249A1 (en) * 2006-12-21 2008-07-03 Ranbaxy Laboratories Limited Anti-inflammatory agents
CA2685597C (en) 2007-05-07 2012-10-02 Amgen Inc. Pyrazolo-pyridinone and pyrazolo-pyrazinone compounds as p38 modulators, process for their preparation, and their pharmaceutical use
JP2010529973A (ja) 2007-06-15 2010-09-02 エフ.ホフマン−ラ ロシュ アーゲー 3−アミノ−ペンタン−1,5−ジオールの新規製造方法
US8367671B2 (en) 2008-03-21 2013-02-05 Amgen Inc. Pyrazolo[3.4-B]pyrazine compounds as p38 modulators and methods of use as anti-inflamatory agents
EP2112150B1 (en) 2008-04-22 2013-10-16 Forma Therapeutics, Inc. Improved raf inhibitors
WO2010046273A2 (en) * 2008-10-22 2010-04-29 F. Hoffmann-La Roche Ag Pyrimidinyl pyridone inhibitors of jnk
WO2010071846A2 (en) 2008-12-19 2010-06-24 Afraxis, Inc. Compounds for treating neuropsychiatric conditions
CN102648200A (zh) * 2009-10-09 2012-08-22 亚弗克希斯公司 用于治疗cns病症的8-乙基-6-(芳基)吡啶并[2,3-d]嘧啶-7(8h)-酮
JP5797664B2 (ja) * 2009-12-18 2015-10-21 テンプル・ユニバーシティ−オブ・ザ・コモンウェルス・システム・オブ・ハイアー・エデュケイションTemple University−Of The Commonwealth System Of Higher Education 置換ピリド[2,3−d]ピリミジン−7(8H)−オン及びそれらの治療用の使用
EP3172214B1 (en) 2014-07-26 2020-05-13 Sunshine Lake Pharma Co., Ltd. 2-amino-pyrido[2,3-d]pyrimidin-7(8h)-one derivatives as cdk inhibitors and uses thereof
JP7349790B2 (ja) * 2016-06-08 2023-09-25 サポート-ヴェンチャー ゲゼルシャフト ミット ベシュレンクター ハフトゥング がんを治療するための薬学的組み合わせ
MA45920B1 (fr) 2016-08-15 2021-08-31 Pfizer Inhibiteurs de pyridopyrimidinone cdk2/4/6
JP2019528273A (ja) 2016-08-17 2019-10-10 サポート−ヴェンチャー ゲゼルシャフト ミット ベシュレンクター ハフトゥング 聴力損失を予防又は治療する方法
US11117858B2 (en) 2017-01-11 2021-09-14 The General Hospital Corporation Voltage gated sodium channel imaging agents
US11576916B2 (en) * 2017-04-04 2023-02-14 Kinarus Ag Methods of preventing or treating ophthalmic diseases
CN115322193A (zh) 2017-08-31 2022-11-11 达纳-法伯癌症研究所股份有限公司 Egfr和/或her2抑制剂和使用方法
PT3691620T (pt) 2017-10-05 2022-10-06 Fulcrum Therapeutics Inc Os inibidores da quinase p38 reduzem a expressão de dux4 e genes a jusante para o tratamento de fshd
US10342786B2 (en) 2017-10-05 2019-07-09 Fulcrum Therapeutics, Inc. P38 kinase inhibitors reduce DUX4 and downstream gene expression for the treatment of FSHD
WO2020006210A1 (en) * 2018-06-27 2020-01-02 Tufts Medical Center, Inc. Pyridopyrimidine compounds and methods of their use
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YU63703A (sh) 2001-02-12 2006-05-25 F. Hoffmann-La Roche Ag. 6-supstituisani pirido-pirimidini
PL218692B1 (pl) * 2002-01-22 2015-01-30 Warner Lambert Co Podstawiony 2-(pirydyn-2-yloamino)pirydo[2,3-d]pirymidyn-7-on oraz jego zastosowanie do leczenia zaburzenia lub stanu spowodowanego nieprawidłową proliferacją komórek

Also Published As

Publication number Publication date
ES2249574T3 (es) 2006-04-01
MXPA03007166A (es) 2003-11-18
HUP0303458A2 (hu) 2004-01-28
US20040116698A1 (en) 2004-06-17
DE60206363D1 (de) 2006-02-09
RU2269527C2 (ru) 2006-02-10
HU229604B1 (en) 2014-02-28
BRPI0207172B1 (pt) 2019-04-09
CA2434834C (en) 2010-09-14
KR100639772B1 (ko) 2006-10-30
NO326133B1 (no) 2008-10-06
JP2004525896A (ja) 2004-08-26
US20030171584A1 (en) 2003-09-11
HUP0303458A3 (en) 2012-12-28
PL366918A1 (en) 2005-02-07
NZ526961A (en) 2005-03-24
ATE305303T1 (de) 2005-10-15
ZA200305938B (en) 2005-01-26
JP4064818B2 (ja) 2008-03-19
NO20033540L (no) 2003-08-11
RU2003125887A (ru) 2005-03-20
US7449581B2 (en) 2008-11-11
BR0207172A (pt) 2004-03-30
US7169794B2 (en) 2007-01-30
YU63703A (sh) 2006-05-25
MY131518A (en) 2007-08-30
BRPI0207172B8 (pt) 2021-05-25
JO2410B1 (en) 2007-06-17
US20070135458A1 (en) 2007-06-14
WO2002064594A2 (en) 2002-08-22
PA8539201A1 (es) 2004-08-31
DE60206363T2 (de) 2006-07-06
AR035854A1 (es) 2004-07-21
HRP20030624B1 (en) 2007-03-31
DK1361880T3 (da) 2006-01-23
CZ20032416A3 (cs) 2004-07-14
MA26993A1 (fr) 2004-12-20
PE20020976A1 (es) 2002-10-29
WO2002064594A3 (en) 2003-01-09
KR20040018254A (ko) 2004-03-02
HK1066170A1 (en) 2005-03-18
US6696566B2 (en) 2004-02-24
EP1361880A2 (en) 2003-11-19
IL156872A0 (en) 2004-02-08
EP1361880B1 (en) 2005-09-28
AU2002256615B2 (en) 2007-09-13
SK11322003A3 (en) 2004-10-05
CN1503672A (zh) 2004-06-09
CN100376571C (zh) 2008-03-26
CA2434834A1 (en) 2002-08-22
IL156872A (en) 2009-07-20
HRP20030624A2 (en) 2005-06-30

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