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NO20011211L - Multippel enhet for kontrollert mateffektuavhengig frigivelse av farmasöytiske preparater og fremgangsmåter for fremstilling avsamme - Google Patents

Multippel enhet for kontrollert mateffektuavhengig frigivelse av farmasöytiske preparater og fremgangsmåter for fremstilling avsamme

Info

Publication number
NO20011211L
NO20011211L NO20011211A NO20011211A NO20011211L NO 20011211 L NO20011211 L NO 20011211L NO 20011211 A NO20011211 A NO 20011211A NO 20011211 A NO20011211 A NO 20011211A NO 20011211 L NO20011211 L NO 20011211L
Authority
NO
Norway
Prior art keywords
methods
pharmaceutical preparations
multiple unit
food effect
dependent release
Prior art date
Application number
NO20011211A
Other languages
English (en)
Other versions
NO20011211D0 (no
Inventor
Venkata-Rangarao Kanikanti
Roland Rupp Haferbusch
Erich Brendel
Claus Weisemann
Ernst Chantraine
Original Assignee
Bayer Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Ag filed Critical Bayer Ag
Publication of NO20011211D0 publication Critical patent/NO20011211D0/no
Publication of NO20011211L publication Critical patent/NO20011211L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/4422—1,4-Dihydropyridines, e.g. nifedipine, nicardipine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
    • A61K9/1605—Excipients; Inactive ingredients
    • A61K9/1629—Organic macromolecular compounds
    • A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

  • Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Urology & Nephrology (AREA)
  • Vascular Medicine (AREA)
  • Cardiology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nonmetallic Welding Materials (AREA)
  • General Preparation And Processing Of Foods (AREA)

Abstract

Foreliggende oppfinnelse angår oralt administrerbare multi-enhets vedvarende frigivelses doseformer som har kontrollert agitasjonsuavhengig frigivelse av aktiv forbindelse og fremgangsmåter for deres fremstilling ved anvendelse av en utvalgt eroderbar hydrofil polymer (HPC) og en begrensning av maksimumstørrelsen for aktiv forbindelse-inneholdende polymerpartikler på < 3 mm.
NO20011211A 1998-09-18 2001-03-09 Multippel enhet for kontrollert mateffektuavhengig frigivelse av farmasöytiske preparater og fremgangsmåter for fremstilling avsamme NO20011211L (no)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
DE19842753A DE19842753A1 (de) 1998-09-18 1998-09-18 Agitationsunabhängige pharmazeutische Retardzubereitungen und Verfahren zu ihrer Herstellung
PCT/EP1999/006882 WO2000016748A1 (de) 1998-09-18 1999-09-17 Agitationsunabhängige pharmazeutische multiple-unit-retardzubereitungen und verfahren zu ihrer herstellung

Publications (2)

Publication Number Publication Date
NO20011211D0 NO20011211D0 (no) 2001-03-09
NO20011211L true NO20011211L (no) 2001-03-09

Family

ID=7881376

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20011211A NO20011211L (no) 1998-09-18 2001-03-09 Multippel enhet for kontrollert mateffektuavhengig frigivelse av farmasöytiske preparater og fremgangsmåter for fremstilling avsamme

Country Status (29)

Country Link
US (1) US6805881B1 (no)
EP (1) EP1113787B1 (no)
JP (1) JP2002526437A (no)
KR (1) KR100660072B1 (no)
CN (1) CN1178650C (no)
AT (1) ATE260645T1 (no)
AU (2) AU5861499A (no)
BG (1) BG105325A (no)
BR (1) BR9913839A (no)
CA (1) CA2344372C (no)
DE (2) DE19842753A1 (no)
DK (1) DK1113787T3 (no)
EE (1) EE04700B1 (no)
ES (1) ES2215404T3 (no)
HK (1) HK1040932B (no)
HR (1) HRP20010198A2 (no)
HU (1) HUP0103669A3 (no)
ID (1) ID28735A (no)
IL (2) IL141532A0 (no)
NO (1) NO20011211L (no)
NZ (1) NZ510563A (no)
PL (1) PL195543B1 (no)
PT (1) PT1113787E (no)
RU (1) RU2235540C2 (no)
SK (1) SK285099B6 (no)
TR (1) TR200100756T2 (no)
UA (1) UA73097C2 (no)
WO (2) WO2000016747A1 (no)
ZA (1) ZA200101485B (no)

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DE19962924A1 (de) * 1999-12-24 2001-07-05 Bayer Ag Substituierte Oxazolidinone und ihre Verwendung
DE10026698A1 (de) 2000-05-30 2001-12-06 Basf Ag Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung
US20020044962A1 (en) * 2000-06-06 2002-04-18 Cherukuri S. Rao Encapsulation products for controlled or extended release
DE10129725A1 (de) * 2001-06-20 2003-01-02 Bayer Ag Kombinationstherapie substituierter Oxazolidinone
AR034813A1 (es) † 2001-07-20 2004-03-17 Novartis Ag Composiciones farmaceuticas y uso de las mismas
US7718189B2 (en) * 2002-10-29 2010-05-18 Transave, Inc. Sustained release of antiinfectives
DE10300111A1 (de) * 2003-01-07 2004-07-15 Bayer Healthcare Ag Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
US8377952B2 (en) 2003-08-28 2013-02-19 Abbott Laboratories Solid pharmaceutical dosage formulation
US8025899B2 (en) 2003-08-28 2011-09-27 Abbott Laboratories Solid pharmaceutical dosage form
DE10355461A1 (de) 2003-11-27 2005-06-23 Bayer Healthcare Ag Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
DE102004062475A1 (de) * 2004-12-24 2006-07-06 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung
KR100866720B1 (ko) 2004-12-27 2008-11-05 에자이 알앤드디 매니지먼트 가부시키가이샤 항치매 약물의 안정화 방법
US20070129402A1 (en) * 2004-12-27 2007-06-07 Eisai Research Institute Sustained release formulations
EP1685841A1 (en) * 2005-01-31 2006-08-02 Bayer Health Care Aktiengesellschaft Prevention and treatment of thromboembolic disorders
DE102005012561B4 (de) 2005-03-18 2008-06-19 Christian Beer Verfahren zum Betrieb eines Werkstück-Transfersystems
DE102005045518A1 (de) * 2005-09-23 2007-03-29 Bayer Healthcare Ag 2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
DE102005047561A1 (de) * 2005-10-04 2007-04-05 Bayer Healthcare Ag Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung
RU2578602C2 (ru) 2005-10-04 2016-03-27 Байер Интеллектуэль Проперти Гмбх Способ получения 5-хлор-n-(5s)-2-оксо-3-[4-(3-оксо-морфолинил)-фенил]-1,3-оксазолидин-5-ил}-метил)-2-тиофенкарбоксамида в модификации ii (варианты)
DE102005047558A1 (de) * 2005-10-04 2008-02-07 Bayer Healthcare Ag Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
CN100448432C (zh) * 2006-10-26 2009-01-07 徐竹青 高溶出度尼莫地平分散片的制备方法
DE102006051625A1 (de) * 2006-11-02 2008-05-08 Bayer Materialscience Ag Kombinationstherapie substituierter Oxazolidinone
US7952167B2 (en) * 2007-04-27 2011-05-31 Taiwan Semiconductor Manufacturing Company, Ltd. Scribe line layout design
TWI478712B (zh) 2008-09-30 2015-04-01 Astellas Pharma Inc 釋控性醫藥組成物
MX2011007779A (es) * 2009-01-28 2011-08-12 Novartis Ag Formulaciones galenicas de compuestos organicos.
US20100247646A1 (en) * 2009-03-26 2010-09-30 Ranbaxy Laboratories Limited Extended release tablets of nisoldipine
TR201802207T4 (tr) 2010-03-29 2018-03-21 Astellas Pharma Inc Kontrollü Salımlı Farmasötik Bileşim.
JP2023553274A (ja) * 2020-11-18 2023-12-21 エフビー－エイチアールエス リミテッド ライアビリティ カンパニー ドフェチリド及びメキシレチンを含有する組成物並びにその使用
US12097189B1 (en) 2024-02-09 2024-09-24 Astellas Pharma Inc. Pharmaceutical composition for modified release

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Also Published As

Publication number Publication date
SK285099B6 (sk) 2006-06-01
AU750617B2 (en) 2002-07-25
ZA200101485B (en) 2002-02-22
ATE260645T1 (de) 2004-03-15
IL141532A0 (en) 2002-03-10
AU6191899A (en) 2000-04-10
IL141532A (en) 2007-03-08
DK1113787T3 (da) 2004-05-17
CA2344372C (en) 2009-12-22
ES2215404T3 (es) 2004-10-01
CN1317959A (zh) 2001-10-17
HUP0103669A2 (hu) 2002-01-28
US6805881B1 (en) 2004-10-19
NO20011211D0 (no) 2001-03-09
RU2235540C2 (ru) 2004-09-10
PT1113787E (pt) 2004-07-30
AU5861499A (en) 2000-04-10
EE04700B1 (et) 2006-10-16
EP1113787B1 (de) 2004-03-03
ID28735A (id) 2001-06-28
BR9913839A (pt) 2001-06-12
WO2000016748A1 (de) 2000-03-30
CN1178650C (zh) 2004-12-08
PL195543B1 (pl) 2007-09-28
CA2344372A1 (en) 2000-03-30
TR200100756T2 (tr) 2001-07-23
DE19842753A1 (de) 2000-03-23
UA73097C2 (en) 2005-06-15
EP1113787A1 (de) 2001-07-11
HK1040932A1 (en) 2002-06-28
JP2002526437A (ja) 2002-08-20
HRP20010198A2 (en) 2002-04-30
EE200100161A (et) 2002-08-15
HK1040932B (zh) 2005-08-05
KR100660072B1 (ko) 2006-12-22
HUP0103669A3 (en) 2006-07-28
WO2000016747A1 (de) 2000-03-30
BG105325A (bg) 2001-11-30
NZ510563A (en) 2002-10-25
SK3722001A3 (en) 2001-10-08
PL346535A1 (en) 2002-02-11
DE59908764D1 (de) 2004-04-08
KR20010073172A (ko) 2001-07-31

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