EE200100161A - Segamisest sõltumatud toimeainet aeglustatult vabastavad mitmeosalised ravimvormid ja nende valmistamismeetodid - Google Patents

Segamisest sõltumatud toimeainet aeglustatult vabastavad mitmeosalised ravimvormid ja nende valmistamismeetodid

Info

Publication number: EE200100161A
Authority: EE; Estonia
Prior art keywords: processes; slow; preparation; release; active compound
Prior art date: 1998-09-18

Application number

EEP200100161A

Other languages

English (en)

Inventor

Kanikanti Venkata-Rangarao

Rupp Roland

Brendel Erich

Weisemann Claus

Chantraine Ernst

Original Assignee

Bayer Aktiengesellschaft

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1998-09-18

Filing date

1999-09-17

Publication date

2002-08-15

1999-09-17 Application filed by Bayer Aktiengesellschaft filed Critical Bayer Aktiengesellschaft

2002-08-15 Publication of EE200100161A publication Critical patent/EE200100161A/et

2006-10-16 Publication of EE04700B1 publication Critical patent/EE04700B1/et

Classifications

- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
- A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
- A61K31/4422—1,4-Dihydropyridines, e.g. nifedipine, nicardipine
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K9/00—Medicinal preparations characterised by special physical form
- A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
- A61K9/16—Agglomerates; Granulates; Microbeadlets ; Microspheres; Pellets; Solid products obtained by spray drying, spray freeze drying, spray congealing,(multiple) emulsion solvent evaporation or extraction
- A61K9/1605—Excipients; Inactive ingredients
- A61K9/1629—Organic macromolecular compounds
- A61K9/1652—Polysaccharides, e.g. alginate, cellulose derivatives; Cyclodextrin
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
- A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis

Landscapes

Health & Medical Sciences (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Public Health (AREA)
Chemical & Material Sciences (AREA)
General Health & Medical Sciences (AREA)
Animal Behavior & Ethology (AREA)
Medicinal Chemistry (AREA)
Life Sciences & Earth Sciences (AREA)
Epidemiology (AREA)
Heart & Thoracic Surgery (AREA)
Organic Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
General Chemical & Material Sciences (AREA)
Chemical Kinetics & Catalysis (AREA)
Cardiology (AREA)
Vascular Medicine (AREA)
Urology & Nephrology (AREA)
Medicinal Preparation (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Nonmetallic Welding Materials (AREA)
General Preparation And Processing Of Foods (AREA)

EEP200100161A 1998-09-18 1999-09-17 Segamisest sõltumatud toimeainet aeglustatult vabastavad mitmeosalised ravimvormid ja nende valmistamismeetodid EE04700B1 (et)

Applications Claiming Priority (2)

Application Number	Priority Date	Filing Date	Title
DE19842753A DE19842753A1 (de)	1998-09-18	1998-09-18	Agitationsunabhängige pharmazeutische Retardzubereitungen und Verfahren zu ihrer Herstellung
PCT/EP1999/006882 WO2000016748A1 (de)	1998-09-18	1999-09-17	Agitationsunabhängige pharmazeutische multiple-unit-retardzubereitungen und verfahren zu ihrer herstellung

Publications (2)

Publication Number	Publication Date
EE200100161A true EE200100161A (et)	2002-08-15
EE04700B1 EE04700B1 (et)	2006-10-16

Family

ID=7881376

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
EEP200100161A EE04700B1 (et)	1998-09-18	1999-09-17	Segamisest sõltumatud toimeainet aeglustatult vabastavad mitmeosalised ravimvormid ja nende valmistamismeetodid

Country Status (29)

Country	Link
US (1)	US6805881B1 (et)
EP (1)	EP1113787B1 (et)
JP (1)	JP2002526437A (et)
KR (1)	KR100660072B1 (et)
CN (1)	CN1178650C (et)
AT (1)	ATE260645T1 (et)
AU (2)	AU5861499A (et)
BG (1)	BG105325A (et)
BR (1)	BR9913839A (et)
CA (1)	CA2344372C (et)
DE (2)	DE19842753A1 (et)
DK (1)	DK1113787T3 (et)
EE (1)	EE04700B1 (et)
ES (1)	ES2215404T3 (et)
HK (1)	HK1040932B (et)
HR (1)	HRP20010198A2 (et)
HU (1)	HUP0103669A3 (et)
ID (1)	ID28735A (et)
IL (2)	IL141532A0 (et)
NO (1)	NO20011211L (et)
NZ (1)	NZ510563A (et)
PL (1)	PL195543B1 (et)
PT (1)	PT1113787E (et)
RU (1)	RU2235540C2 (et)
SK (1)	SK285099B6 (et)
TR (1)	TR200100756T2 (et)
UA (1)	UA73097C2 (et)
WO (2)	WO2000016747A1 (et)
ZA (1)	ZA200101485B (et)

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DE19962924A1 (de)	1999-12-24	2001-07-05	Bayer Ag	Substituierte Oxazolidinone und ihre Verwendung
DE10026698A1 (de)	2000-05-30	2001-12-06	Basf Ag	Selbstemulgierende Wirkstoffformulierung und Verwendung dieser Formulierung
US20020044962A1 (en) *	2000-06-06	2002-04-18	Cherukuri S. Rao	Encapsulation products for controlled or extended release
DE10129725A1 (de) *	2001-06-20	2003-01-02	Bayer Ag	Kombinationstherapie substituierter Oxazolidinone
AR034813A1 (es) †	2001-07-20	2004-03-17	Novartis Ag	Composiciones farmaceuticas y uso de las mismas
US7718189B2 (en) *	2002-10-29	2010-05-18	Transave, Inc.	Sustained release of antiinfectives
DE10300111A1 (de) *	2003-01-07	2004-07-15	Bayer Healthcare Ag	Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
US8025899B2 (en)	2003-08-28	2011-09-27	Abbott Laboratories	Solid pharmaceutical dosage form
US8377952B2 (en)	2003-08-28	2013-02-19	Abbott Laboratories	Solid pharmaceutical dosage formulation
DE10355461A1 (de)	2003-11-27	2005-06-23	Bayer Healthcare Ag	Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
DE102004062475A1 (de) *	2004-12-24	2006-07-06	Bayer Healthcare Ag	Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung
EP1830886B1 (en)	2004-12-27	2016-04-13	Eisai R&D Management Co., Ltd.	Method for stabilizing anti-dementia drug
US20070129402A1 (en) *	2004-12-27	2007-06-07	Eisai Research Institute	Sustained release formulations
EP1685841A1 (en)	2005-01-31	2006-08-02	Bayer Health Care Aktiengesellschaft	Prevention and treatment of thromboembolic disorders
DE102005012561B4 (de)	2005-03-18	2008-06-19	Christian Beer	Verfahren zum Betrieb eines Werkstück-Transfersystems
DE102005045518A1 (de) *	2005-09-23	2007-03-29	Bayer Healthcare Ag	2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
EP1934208B1 (de)	2005-10-04	2011-03-23	Bayer Schering Pharma Aktiengesellschaft	Neue polymorphe form von 5-chlor-n-({ ( 5s )-2-0x0-3-[4-( 3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl} -methyl)-2-thiophencarboxamid
DE102005047561A1 (de)	2005-10-04	2007-04-05	Bayer Healthcare Ag	Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung
DE102005047558A1 (de) *	2005-10-04	2008-02-07	Bayer Healthcare Ag	Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
CN100448432C (zh) *	2006-10-26	2009-01-07	徐竹青	高溶出度尼莫地平分散片的制备方法
DE102006051625A1 (de) *	2006-11-02	2008-05-08	Bayer Materialscience Ag	Kombinationstherapie substituierter Oxazolidinone
US7952167B2 (en) *	2007-04-27	2011-05-31	Taiwan Semiconductor Manufacturing Company, Ltd.	Scribe line layout design
TWI478712B (zh)	2008-09-30	2015-04-01	Astellas Pharma Inc	釋控性醫藥組成物
TWI468191B (zh) *	2009-01-28	2015-01-11	Novartis Ag	有機化合物之調配物
US20100247646A1 (en) *	2009-03-26	2010-09-30	Ranbaxy Laboratories Limited	Extended release tablets of nisoldipine
JP5849947B2 (ja)	2010-03-29	2016-02-03	アステラス製薬株式会社	放出制御医薬組成物
EP4247354A4 (en) *	2020-11-18	2025-02-19	Fb-Hrs, Llc	COMPOSITIONS CONTAINING DOFETILIDE AND MEXILETINE AND THEIR USES
US12097189B1 (en)	2024-02-09	2024-09-24	Astellas Pharma Inc.	Pharmaceutical composition for modified release

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JPS5482525A (en)	1977-12-13	1979-06-30	Aisan Ind Co Ltd	Exhaust gas recirculation system
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DE3612212A1 (de)	1986-04-11	1987-10-15	Basf Ag	Verfahren zur herstellung von festen pharmazeutischen formen
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JPS63222121A (ja) *	1987-03-10	1988-09-16	Nippon Soda Co Ltd	徐放性ゲル製剤
DE3720757A1 (de)	1987-06-24	1989-01-05	Bayer Ag	Dhp-manteltablette
JPH02167229A (ja) *	1988-09-01	1990-06-27	Kureha Chem Ind Co Ltd	かわらたけ由来の蛋白多糖体の粒状製剤
DE3830353A1 (de)	1988-09-07	1990-03-15	Basf Ag	Verfahren zur kontinuierlichen herstellung von festen pharmazeutischen formen
JPH03101615A (ja) *	1989-09-14	1991-04-26	Sumitomo Pharmaceut Co Ltd	胃内滞留型持続性製剤
JPH03145418A (ja)	1989-10-27	1991-06-20	Sumitomo Pharmaceut Co Ltd	塩基性薬物塩酸塩の徐放性製剤
JP3078859B2 (ja) *	1990-02-23	2000-08-21	武田薬品工業株式会社	安定な放出制御性製剤用コーティング剤
ES2111065T5 (es)	1991-04-16	2005-06-16	Nippon Shinyaku Company, Limited	Procedimiento para producir una dispersion solida.
DE4138513A1 (de)	1991-11-23	1993-05-27	Basf Ag	Feste pharmazeutische retardform
JP3059004B2 (ja) *	1992-09-18	2000-07-04	ダイセル化学工業株式会社	アルカリ水溶液に対する溶解性の高い低置換度ヒドロキシプロピルセルロース及びその製造法
DE4413350A1 (de)	1994-04-18	1995-10-19	Basf Ag	Retard-Matrixpellets und Verfahren zu ihrer Herstellung
SE9402422D0 (sv) *	1994-07-08	1994-07-08	Astra Ab	New beads for controlled release and a pharmaceutical preparation containing the same
FR2725624B1 (fr)	1994-10-14	1997-01-17	Jouveinal Inst Rech	Procede de preparation de formes pharmaceutiques a liberation controlee
DE19504831A1 (de)	1995-02-14	1996-09-05	Basf Ag	Feste Wirkstoffzubereitungen enthaltend Hydroxypropylcellulose

1998
- 1998-09-18 DE DE19842753A patent/DE19842753A1/de not_active Withdrawn
1999
- 1999-09-08 AU AU58614/99A patent/AU5861499A/en not_active Abandoned
- 1999-09-08 WO PCT/EP1999/006608 patent/WO2000016747A1/de not_active Ceased
- 1999-09-17 JP JP2000573709A patent/JP2002526437A/ja not_active Ceased
- 1999-09-17 UA UA2001042576A patent/UA73097C2/uk unknown
- 1999-09-17 BR BR9913839-5A patent/BR9913839A/pt not_active Application Discontinuation
- 1999-09-17 HK HK02102756.8A patent/HK1040932B/zh not_active IP Right Cessation
- 1999-09-17 IL IL14153299A patent/IL141532A0/xx not_active IP Right Cessation
- 1999-09-17 EP EP99948770A patent/EP1113787B1/de not_active Expired - Lifetime
- 1999-09-17 KR KR1020017003495A patent/KR100660072B1/ko not_active Expired - Fee Related
- 1999-09-17 SK SK372-2001A patent/SK285099B6/sk unknown
- 1999-09-17 NZ NZ510563A patent/NZ510563A/xx unknown
- 1999-09-17 CN CNB998110299A patent/CN1178650C/zh not_active Expired - Fee Related
- 1999-09-17 DE DE59908764T patent/DE59908764D1/de not_active Expired - Lifetime
- 1999-09-17 AU AU61918/99A patent/AU750617B2/en not_active Ceased
- 1999-09-17 HU HU0103669A patent/HUP0103669A3/hu unknown
- 1999-09-17 US US09/787,229 patent/US6805881B1/en not_active Expired - Fee Related
- 1999-09-17 EE EEP200100161A patent/EE04700B1/et not_active IP Right Cessation
- 1999-09-17 DK DK99948770T patent/DK1113787T3/da active
- 1999-09-17 ID IDW20010651A patent/ID28735A/id unknown
- 1999-09-17 PT PT99948770T patent/PT1113787E/pt unknown
- 1999-09-17 WO PCT/EP1999/006882 patent/WO2000016748A1/de not_active Ceased
- 1999-09-17 CA CA002344372A patent/CA2344372C/en not_active Expired - Fee Related
- 1999-09-17 AT AT99948770T patent/ATE260645T1/de not_active IP Right Cessation
- 1999-09-17 ES ES99948770T patent/ES2215404T3/es not_active Expired - Lifetime
- 1999-09-17 PL PL99346535A patent/PL195543B1/pl unknown
- 1999-09-17 TR TR2001/00756T patent/TR200100756T2/xx unknown
- 1999-09-17 HR HR20010198A patent/HRP20010198A2/hr not_active Application Discontinuation
- 1999-09-17 RU RU2001110355/15A patent/RU2235540C2/ru not_active IP Right Cessation
2001
- 2001-02-20 IL IL141532A patent/IL141532A/en unknown
- 2001-02-22 ZA ZA200101485A patent/ZA200101485B/en unknown
- 2001-03-09 NO NO20011211A patent/NO20011211L/no not_active Application Discontinuation
- 2001-03-09 BG BG105325A patent/BG105325A/bg unknown

Also Published As

Publication number	Publication date
HUP0103669A3 (en)	2006-07-28
JP2002526437A (ja)	2002-08-20
BG105325A (bg)	2001-11-30
IL141532A (en)	2007-03-08
ATE260645T1 (de)	2004-03-15
US6805881B1 (en)	2004-10-19
CA2344372C (en)	2009-12-22
ZA200101485B (en)	2002-02-22
WO2000016748A1 (de)	2000-03-30
HRP20010198A2 (en)	2002-04-30
EP1113787A1 (de)	2001-07-11
SK285099B6 (sk)	2006-06-01
DE19842753A1 (de)	2000-03-23
UA73097C2 (en)	2005-06-15
HK1040932A1 (en)	2002-06-28
NO20011211D0 (no)	2001-03-09
DK1113787T3 (da)	2004-05-17
PL346535A1 (en)	2002-02-11
CN1317959A (zh)	2001-10-17
CA2344372A1 (en)	2000-03-30
NO20011211L (no)	2001-03-09
KR20010073172A (ko)	2001-07-31
HUP0103669A2 (hu)	2002-01-28
RU2235540C2 (ru)	2004-09-10
WO2000016747A1 (de)	2000-03-30
SK3722001A3 (en)	2001-10-08
IL141532A0 (en)	2002-03-10
HK1040932B (zh)	2005-08-05
TR200100756T2 (tr)	2001-07-23
BR9913839A (pt)	2001-06-12
DE59908764D1 (de)	2004-04-08
PL195543B1 (pl)	2007-09-28
AU5861499A (en)	2000-04-10
ES2215404T3 (es)	2004-10-01
AU6191899A (en)	2000-04-10
CN1178650C (zh)	2004-12-08
AU750617B2 (en)	2002-07-25
KR100660072B1 (ko)	2006-12-22
NZ510563A (en)	2002-10-25
EE04700B1 (et)	2006-10-16
PT1113787E (pt)	2004-07-30
EP1113787B1 (de)	2004-03-03
ID28735A (id)	2001-06-28

Publication	Publication Date	Title
EE04700B1 (et)	2006-10-16	Segamisest sõltumatud toimeainet aeglustatult vabastavad mitmeosalised ravimvormid ja nende valmistamismeetodid
IL135130A0 (en)	2001-05-20	Pharmaceutical preparation comprising clodronate as active ingredient and silicified microcrystalline cellulose as excipient
NO995006D0 (no)	1999-10-14	Nye forbindelser
CA2427815A1 (en)	2002-05-10	Controlled release hydrocodone formulations
YU35893A (sh)	1997-03-07	Formulacije oksidona sa kontrolisanim otpuštanjem i njihova upotreba
ES2172239T3 (es)	2002-09-16	Sistema osmotico de liberacion de farmacos.
BG104727A (en)	2001-05-31	Pharmaceutical composition of topiramate
BR9405843A (pt)	1996-01-16	Processo para reduzir perda óssea e uso de um composto
HUP0002296A2 (hu)	2001-10-28	Sertralinsók és a sertralin elnyújtott felszabadulását biztosító dózisformák
BR9612291A (pt)	1999-07-13	Forma de dosagem sólida bioadesiva
TR200000129T2 (tr)	2000-07-21	Yepyeni spiroazabisiklik heterosiklik bileşikler.
ZA200205512B (en)	2004-02-10	Novel substituted benzimidazole dosage forms and methods of using same.
BR9916361A (pt)	2002-11-05	Forma de dosagem de tabletes de liberação controlada, formulação de tablete de liberação controlada, composição granular para prensagem em uma forma de dosagem de tablete de liberação controlada, e, métodos para preparar uma composição granular, para preparar uma forma de dosagem de tabletes de liberação controlada de divalproex sódio e para tratar epilepsia
AU3533395A (en)	1996-04-26	Oral sustained-release preparation
IS3789A7 (is)	1992-06-08	Aðferð við framleiðslu lyfjaskammta í föstu formimeð tempraðri losun virks þáttar
PT1121109E (pt)	2006-09-29	Formulacao bifasica contendo tramadol
IL110025A0 (en)	1994-10-07	Phosphonosuccinic acid derivatives, processes for the preparation thereof and pharmaceutical compositions containing them
MY133957A (en)	2007-11-30	"compounds useful for the treatment or prevention of a disease mediated by the alpha-2b-adrenoceptor"
HU0100122D0 (en)	2001-03-28	Use of tiludronic acid and derivatives thereof in poultry for preparation of a medicinal product for preventing and treating osteoporosis

Legal Events

Date	Code	Title	Description
2007-02-15	KB4A	Valid patent at the end of a year	Effective date: 20061231
2008-02-15	KB4A	Valid patent at the end of a year	Effective date: 20071231
2008-06-16	MM4A	Lapsed by not paying the annual fees	Effective date: 20070917