ZA200204166B - Oxazolidinones having a sulfoximine functionality and their use as antimicrobial agents. - Google Patents

Oxazolidinones having a sulfoximine functionality and their use as antimicrobial agents.

Info

Publication number: ZA200204166B
Authority: ZA; South Africa
Prior art keywords: oxazolidinones; antimicrobial agents; sulfoximine; functionality; sulfoximine functionality
Prior art date: 1999-12-21

Application number

ZA200204166A

Other languages

English (en)

Inventor

Jackson B Hester Jr

David L Alexander

Original Assignee

Upjohn Co

Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)

1999-12-21

Filing date

2002-05-24

Publication date

2003-10-29

2002-05-24 Application filed by Upjohn Co filed Critical Upjohn Co

2003-10-29 Publication of ZA200204166B publication Critical patent/ZA200204166B/xx

Classifications

- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing aromatic rings
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P17/00—Drugs for dermatological disorders
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P27/00—Drugs for disorders of the senses
- A61P27/02—Ophthalmic agents
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
- C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
- C07D417/10—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a carbon chain containing aromatic rings

Landscapes

Chemical & Material Sciences (AREA)
Organic Chemistry (AREA)
Health & Medical Sciences (AREA)
Life Sciences & Earth Sciences (AREA)
Public Health (AREA)
General Chemical & Material Sciences (AREA)
Medicinal Chemistry (AREA)
Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
Chemical Kinetics & Catalysis (AREA)
Pharmacology & Pharmacy (AREA)
Veterinary Medicine (AREA)
Animal Behavior & Ethology (AREA)
General Health & Medical Sciences (AREA)
Oncology (AREA)
Communicable Diseases (AREA)
Engineering & Computer Science (AREA)
Bioinformatics & Cheminformatics (AREA)
Ophthalmology & Optometry (AREA)
Dermatology (AREA)
Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
Plural Heterocyclic Compounds (AREA)

ZA200204166A 1999-12-21 2002-05-24 Oxazolidinones having a sulfoximine functionality and their use as antimicrobial agents. ZA200204166B (en)

Applications Claiming Priority (1)

Application Number	Priority Date	Filing Date	Title
US17191699P	1999-12-21	1999-12-21

Publications (1)

Publication Number	Publication Date
ZA200204166B true ZA200204166B (en)	2003-10-29

Family

ID=22625632

Family Applications (1)

Application Number	Title	Priority Date	Filing Date
ZA200204166A ZA200204166B (en)	1999-12-21	2002-05-24	Oxazolidinones having a sulfoximine functionality and their use as antimicrobial agents.

Country Status (22)

Country	Link
US (1)	US20010046987A1 (sk)
EP (1)	EP1242417A1 (sk)
JP (1)	JP2003518117A (sk)
KR (1)	KR20020067557A (sk)
CN (1)	CN1221548C (sk)
AR (1)	AR029211A1 (sk)
AU (1)	AU782078B2 (sk)
BR (1)	BR0016605A (sk)
CA (1)	CA2389482A1 (sk)
CO (1)	CO5251427A1 (sk)
CZ (1)	CZ20022142A3 (sk)
EA (1)	EA005567B1 (sk)
HU (1)	HUP0203869A2 (sk)
IL (1)	IL150348A0 (sk)
MX (1)	MXPA02006233A (sk)
NO (1)	NO20022973L (sk)
NZ (1)	NZ519725A (sk)
PE (1)	PE20010931A1 (sk)
PL (1)	PL356478A1 (sk)
SK (1)	SK7572002A3 (sk)
WO (1)	WO2001046185A1 (sk)
ZA (1)	ZA200204166B (sk)

Families Citing this family (27)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
GB9928568D0 (en)	1999-12-03	2000-02-02	Zeneca Ltd	Chemical compounds
DE19962924A1 (de)	1999-12-24	2001-07-05	Bayer Ag	Substituierte Oxazolidinone und ihre Verwendung
GB0009803D0 (en)	2000-04-25	2000-06-07	Astrazeneca Ab	Chemical compounds
GB0108794D0 (en) *	2001-04-07	2001-05-30	Astrazeneca Ab	Chemical compound
GB0108764D0 (en) *	2001-04-07	2001-05-30	Astrazeneca Ab	Chemical compounds
ATE332299T1 (de) *	2001-04-07	2006-07-15	Astrazeneca Ab	Eine sulfonimid-gruppe enthaltende oxazolidinone als antibiotika
GB0108793D0 (en) *	2001-04-07	2001-05-30	Astrazeneca Ab	Chemical compounds
DE10129725A1 (de)	2001-06-20	2003-01-02	Bayer Ag	Kombinationstherapie substituierter Oxazolidinone
US7141588B2 (en)	2002-02-25	2006-11-28	Pfizer, Inc.	N-aryl-2-oxazolidinone-5-carboxamides and their derivatives
AR038536A1 (es)	2002-02-25	2005-01-19	Upjohn Co	N-aril-2-oxazolidinona-5- carboxamidas y sus derivados
TW200403240A (en)	2002-06-28	2004-03-01	Upjohn Co	Difluorothioacetamides of oxazolidinones as antibacterial agents
US6875784B2 (en) *	2002-10-09	2005-04-05	Pharmacia & Upjohn Company	Antimibicrobial [3.1.0.] bicyclic oxazolidinone derivatives
DE10300111A1 (de) *	2003-01-07	2004-07-15	Bayer Healthcare Ag	Verfahren zur Herstellung von 5-Chlor-N-({(5S)-2-oxo-3-[4-(3-oxo-4-morpholinyl)-phenyl]-1,3-oxazolidin-5-yl}-methyl)-2-thiophencarboxamid
CA2521685A1 (en)	2003-04-09	2004-10-21	Pharmacia & Upjohn Company Llc	Antimicrobial [3.1.0] bicyclohexylphenyl-oxazolidinone derivatives and analogues
US7304050B2 (en)	2003-09-16	2007-12-04	Pfizer Inc.	Antibacterial agents
US7265140B2 (en) *	2003-09-23	2007-09-04	Pfizer Inc	Acyloxymethylcarbamate prodrugs of oxazolidinones
DE10355461A1 (de)	2003-11-27	2005-06-23	Bayer Healthcare Ag	Verfahren zur Herstellung einer festen, oral applizierbaren pharmazeutischen Zusammensetzung
JP2008521792A (ja) *	2004-11-29	2008-06-26	ファルマシア・アンド・アップジョン・カンパニー・エルエルシー	抗菌薬としてのジアゼピンオキサゾリジノン
DE102004062475A1 (de) *	2004-12-24	2006-07-06	Bayer Healthcare Ag	Feste, oral applizierbare pharmazeutische Darreichungsformen mit modifizierter Freisetzung
EP1685841A1 (en)	2005-01-31	2006-08-02	Bayer Health Care Aktiengesellschaft	Prevention and treatment of thromboembolic disorders
ATE449773T1 (de)	2005-06-29	2009-12-15	Pharmacia & Upjohn Co Llc	Homomorpholinoxazolidinone als antibakterielle mittel
DE102005045518A1 (de) *	2005-09-23	2007-03-29	Bayer Healthcare Ag	2-Aminoethoxyessigsäure-Derivate und ihre Verwendung
DE102005047558A1 (de) *	2005-10-04	2008-02-07	Bayer Healthcare Ag	Kombinationstherapie substituierter Oxazolidinone zur Prophylaxe und Behandlung von cerebralen Durchblutungsstörungen
PT1934208E (pt)	2005-10-04	2011-06-01	Bayer Schering Pharma Ag	Nova forma polimorfa de 5-cloro-n-({(5s)-2-oxo-3-[4-(3- oxo-4-morfolinil)-fenil]-1,3-oxazolidin-5-il}-metil)-2- tiofenocarboxamida
DE102005047561A1 (de)	2005-10-04	2007-04-05	Bayer Healthcare Ag	Feste, oral applizierbare pharmazeutische Darreichungsformen mit schneller Wirkstofffreisetzung
DE102007028319A1 (de) *	2007-06-20	2008-12-24	Bayer Healthcare Ag	Substituierte Oxazolidinone und ihre Verwendung
WO2021184339A1 (en) *	2020-03-20	2021-09-23	Merck Sharp & Dohme Corp.	Oxazolidinone compound and methods of use thereof as an antibacterial agent

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number	Priority date	Publication date	Assignee	Title
US5688792A (en) *	1994-08-16	1997-11-18	Pharmacia & Upjohn Company	Substituted oxazine and thiazine oxazolidinone antimicrobials
MY115155A (en) *	1993-09-09	2003-04-30	Upjohn Co	Substituted oxazine and thiazine oxazolidinone antimicrobials.
JPH10508844A (ja) *	1994-11-15	1998-09-02	ファルマシア・アンド・アップジョン・カンパニー	二環式オキサジンおよびチアジンオキサゾリジノン抗菌剤
DE69616366T2 (de) *	1995-09-01	2002-07-04	Upjohn Co	Phenyloxazolidinone mit einer c-c-bindung zu 4-8 gliedrigen heterocyclen
KR20010013192A (ko) *	1997-05-30	2001-02-26	로렌스 티. 마이젠헬더	티오카보닐 작용기를 갖는 옥사졸리디논 항균제

2000
- 2000-12-12 NZ NZ519725A patent/NZ519725A/en unknown
- 2000-12-12 EP EP00983792A patent/EP1242417A1/en not_active Withdrawn
- 2000-12-12 IL IL15034800A patent/IL150348A0/xx unknown
- 2000-12-12 KR KR1020027007958A patent/KR20020067557A/ko not_active Withdrawn
- 2000-12-12 CZ CZ20022142A patent/CZ20022142A3/cs unknown
- 2000-12-12 WO PCT/US2000/032451 patent/WO2001046185A1/en not_active Ceased
- 2000-12-12 AU AU20502/01A patent/AU782078B2/en not_active Ceased
- 2000-12-12 JP JP2001547095A patent/JP2003518117A/ja active Pending
- 2000-12-12 CN CNB008160449A patent/CN1221548C/zh not_active Expired - Fee Related
- 2000-12-12 MX MXPA02006233A patent/MXPA02006233A/es unknown
- 2000-12-12 SK SK757-2002A patent/SK7572002A3/sk unknown
- 2000-12-12 CA CA002389482A patent/CA2389482A1/en not_active Abandoned
- 2000-12-12 HU HU0203869A patent/HUP0203869A2/hu unknown
- 2000-12-12 EA EA200200699A patent/EA005567B1/ru not_active IP Right Cessation
- 2000-12-12 BR BR0016605-7A patent/BR0016605A/pt not_active IP Right Cessation
- 2000-12-12 PL PL00356478A patent/PL356478A1/xx not_active Application Discontinuation
- 2000-12-14 US US09/736,858 patent/US20010046987A1/en not_active Abandoned
- 2000-12-19 PE PE2000001363A patent/PE20010931A1/es not_active Application Discontinuation
- 2000-12-20 AR ARP000106795A patent/AR029211A1/es unknown
- 2000-12-20 CO CO00096639A patent/CO5251427A1/es not_active Application Discontinuation
2002
- 2002-05-24 ZA ZA200204166A patent/ZA200204166B/xx unknown
- 2002-06-20 NO NO20022973A patent/NO20022973L/no not_active Application Discontinuation

Also Published As

Publication number	Publication date
EP1242417A1 (en)	2002-09-25
NO20022973D0 (no)	2002-06-20
NO20022973L (no)	2002-08-20
EA200200699A1 (ru)	2003-02-27
BR0016605A (pt)	2003-02-25
EA005567B1 (ru)	2005-04-28
AR029211A1 (es)	2003-06-18
IL150348A0 (en)	2002-12-01
CN1221548C (zh)	2005-10-05
HUP0203869A2 (hu)	2003-07-28
PL356478A1 (en)	2004-06-28
CA2389482A1 (en)	2001-06-28
US20010046987A1 (en)	2001-11-29
MXPA02006233A (es)	2002-12-05
PE20010931A1 (es)	2001-08-29
CO5251427A1 (es)	2003-02-28
NZ519725A (en)	2004-05-28
SK7572002A3 (en)	2002-12-03
CZ20022142A3 (cs)	2002-11-13
AU2050201A (en)	2001-07-03
KR20020067557A (ko)	2002-08-22
CN1391572A (zh)	2003-01-15
AU782078B2 (en)	2005-06-30
WO2001046185A1 (en)	2001-06-28
JP2003518117A (ja)	2003-06-03

Publication	Publication Date	Title
ZA200204166B (en)	2003-10-29	Oxazolidinones having a sulfoximine functionality and their use as antimicrobial agents.
AU2001286878A1 (en)	2002-03-13	Oxazolidinones and their use as antibacterial agents
MXPA03000503A (es)	2003-10-14	Derivados de oxazolidinona como antimicrobianos.
HUS1300061I1 (hu)	2017-08-28	Herbicid kompozíció
MXPA02006460A (es)	2003-09-22	Trifluorometilpirrolcarboxamidas y trifluorometilpirroltioamidas como fungicidas.
HUP0203143A3 (en)	2004-12-28	Synergistic herbicidal composition and its use
IL150393A0 (en)	2002-12-01	3-aminoquinazolin-2,4-dione antibacterial agents
MX244938B (es)	2007-04-12	Toallas antimicrobianas que proveen reduccion inmediata mejorada de germenes.
ZA200101733B (en)	2001-05-09	Plastic implant.
AU4344600A (en)	2000-11-14	Antimicrobial
ZA997876B (en)	2001-06-25	A disposable absorbent article.
MXPA02006325A (es)	2003-09-22	Maquina precortadora y biseladora.
ZA200108294B (en)	2002-12-24	Stretchable nonwoven material.
HUP0201795A3 (en)	2003-10-28	Disinfectants
ZA200001416B (en)	2000-10-24	Pesticidal compositions.
MXPA02003660A (es)	2003-10-14	Composicion herbicida y adyuvante.
ZA200202530B (en)	2003-06-25	Fabric care composition.
AU7236500A (en)	2000-12-05	Antimicrobial copolymers
AU2002216249A1 (en)	2002-07-01	Antimicrobial agents
ZA200109902B (en)	2003-05-28	Stable biocidal compositions.
GB9927160D0 (en)	2000-01-12	Gardening implement
AU5630800A (en)	2001-01-09	Antimicrobial agents
AU2362401A (en)	2001-06-18	N-phenylcarbamates having a microbicide, insecticide and acaricide effect
MXPA02002850A (es)	2003-12-11	Fungicidas.
ZA200107483B (en)	2003-01-29	Synergistic insecticidal compositions.