UY32036A - Derivados de ciclohexil-amida, composiciones farmacéuticas que los contienen, su preparación y aplicaciones - Google Patents
Derivados de ciclohexil-amida, composiciones farmacéuticas que los contienen, su preparación y aplicacionesInfo
- Publication number
- UY32036A UY32036A UY0001032036A UY32036A UY32036A UY 32036 A UY32036 A UY 32036A UY 0001032036 A UY0001032036 A UY 0001032036A UY 32036 A UY32036 A UY 32036A UY 32036 A UY32036 A UY 32036A
- Authority
- UY
- Uruguay
- Prior art keywords
- derivatives
- ciclohexil
- amida
- contain
- applications
- Prior art date
Links
- 239000008194 pharmaceutical composition Substances 0.000 title 1
- 102400000739 Corticotropin Human genes 0.000 abstract 1
- 101800000414 Corticotropin Proteins 0.000 abstract 1
- 239000005557 antagonist Substances 0.000 abstract 1
- IDLFZVILOHSSID-OVLDLUHVSA-N corticotropin Chemical compound C([C@@H](C(=O)N[C@@H](CO)C(=O)N[C@@H](CCSC)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC=1NC=NC=1)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CC=1C2=CC=CC=C2NC=1)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C(C)C)C(=O)NCC(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N[C@@H](CCCNC(N)=N)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](C(C)C)C(=O)N[C@@H](CC=1C=CC(O)=CC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(N)=O)C(=O)NCC(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC(O)=O)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CO)C(=O)N[C@@H](C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](C)C(=O)N[C@@H](CC=1C=CC=CC=1)C(=O)N1[C@@H](CCC1)C(=O)N[C@@H](CC(C)C)C(=O)N[C@@H](CCC(O)=O)C(=O)N[C@@H](CC=1C=CC=CC=1)C(O)=O)NC(=O)[C@@H](N)CO)C1=CC=C(O)C=C1 IDLFZVILOHSSID-OVLDLUHVSA-N 0.000 abstract 1
- 229960000258 corticotropin Drugs 0.000 abstract 1
- PAFZNILMFXTMIY-UHFFFAOYSA-N cyclohexylamine Chemical class NC1CCCCC1 PAFZNILMFXTMIY-UHFFFAOYSA-N 0.000 abstract 1
Classifications
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Abstract
Se describen derivados de ciclohexil-amida como antagonistas del receptor del factor de liberación de corticotropina (CRF-1).
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| EP08162006 | 2008-08-07 | ||
| US20513909P | 2009-01-14 | 2009-01-14 | |
| EP09150543 | 2009-01-14 |
Publications (1)
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| UY32036A true UY32036A (es) | 2010-03-26 |
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| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| UY0001032036A UY32036A (es) | 2008-08-07 | 2009-08-05 | Derivados de ciclohexil-amida, composiciones farmacéuticas que los contienen, su preparación y aplicaciones |
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| US (3) | US8273900B2 (es) |
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| JP (1) | JP5527745B2 (es) |
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| CN (1) | CN102143940B (es) |
| AR (1) | AR072969A1 (es) |
| AU (1) | AU2009279089B2 (es) |
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| CA (1) | CA2732887A1 (es) |
| CO (1) | CO6351776A2 (es) |
| EA (1) | EA020921B1 (es) |
| EC (1) | ECSP11010814A (es) |
| ES (1) | ES2582576T3 (es) |
| HN (1) | HN2011000372A (es) |
| IL (1) | IL210834A0 (es) |
| MA (1) | MA32534B1 (es) |
| MX (1) | MX2011001375A (es) |
| MY (1) | MY151568A (es) |
| PE (1) | PE20110237A1 (es) |
| SV (1) | SV2011003832A (es) |
| TN (1) | TN2011000040A1 (es) |
| TW (1) | TW201011001A (es) |
| UY (1) | UY32036A (es) |
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Families Citing this family (27)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8273900B2 (en) * | 2008-08-07 | 2012-09-25 | Novartis Ag | Organic compounds |
| WO2011092293A2 (en) * | 2010-02-01 | 2011-08-04 | Novartis Ag | Cyclohexyl amide derivatives as crf receptor antagonists |
| CN102753527B (zh) * | 2010-02-02 | 2014-12-24 | 诺华股份有限公司 | 用作crf受体拮抗剂的环己基酰胺衍生物 |
| RU2639876C2 (ru) | 2010-03-30 | 2017-12-25 | Версеон Корпорейшн | Мультизамещенные ароматические соединения в качестве ингибиторов тромбина |
| AU2011348220B2 (en) | 2010-12-22 | 2017-09-07 | The Salk Institute For Biological Studies | Cyclic CRF antagonist peptides |
| UY34094A (es) | 2011-05-27 | 2013-01-03 | Novartis Ag | Derivados de la piperidina 3-espirocíclica como agonistas de receptores de la ghrelina |
| EP2567959B1 (en) | 2011-09-12 | 2014-04-16 | Sanofi | 6-(4-hydroxy-phenyl)-3-styryl-1h-pyrazolo[3,4-b]pyridine-4-carboxylic acid amide derivatives as kinase inhibitors |
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| 109 | Application deemed to be withdrawn |
Effective date: 20181112 |