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UY31010A1 - Nuevo régimen de drospirenona/17b-estradiol, producto farmacéutico combinado y conjunto de elementos (kit) para su aplicacion - Google Patents

Nuevo régimen de drospirenona/17b-estradiol, producto farmacéutico combinado y conjunto de elementos (kit) para su aplicacion

Info

Publication number
UY31010A1
UY31010A1 UY31010A UY31010A UY31010A1 UY 31010 A1 UY31010 A1 UY 31010A1 UY 31010 A UY31010 A UY 31010A UY 31010 A UY31010 A UY 31010A UY 31010 A1 UY31010 A1 UY 31010A1
Authority
UY
Uruguay
Prior art keywords
estradiol
pharmaceutical product
drospirenona
kit
elements
Prior art date
Application number
UY31010A
Other languages
English (en)
Inventor
Joachim Marr
Bernd Doesterberg
Rolf Schoermann
Hartmut Blode
Vladimir Hanes
Original Assignee
Bayer Schering Pharma Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39745001&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=UY31010(A1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Bayer Schering Pharma Ag filed Critical Bayer Schering Pharma Ag
Publication of UY31010A1 publication Critical patent/UY31010A1/es

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/56Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/58Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
    • A61K31/585Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/12Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P15/00Drugs for genital or sexual disorders; Contraceptives
    • A61P15/18Feminine contraceptives

Landscapes

  • Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Medicinal Chemistry (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Reproductive Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Endocrinology (AREA)
  • Gynecology & Obstetrics (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)

Abstract

Un producto farmacéutico combinado de al menos 21 unidades de dosificacion diarias consecutivas que contienen entre 2,0 mg y 3,0 mg de drospirenona y entre 1,0 y 2,0 mg de 17 B(Bet)-estradiol en cada unidad de dosifiacion diaria seguido por unidades de dosificacion diarias intermitentes que contienen la misma cantidad, o una cantidad menor, de drospirenona ( es decir, entre 0,5mg y 3,0 mg) como unidades de dosificacion diarias consecutivas, en donde cada unidad de dosifiacion diaria intermitente está prededida por al menos un día sin administracion de drospirenona.
UY31010A 2007-04-05 2008-04-07 Nuevo régimen de drospirenona/17b-estradiol, producto farmacéutico combinado y conjunto de elementos (kit) para su aplicacion UY31010A1 (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US91032607P 2007-04-05 2007-04-05
US3528508P 2008-03-10 2008-03-10
US4049408P 2008-03-28 2008-03-28

Publications (1)

Publication Number Publication Date
UY31010A1 true UY31010A1 (es) 2008-11-28

Family

ID=39745001

Family Applications (1)

Application Number Title Priority Date Filing Date
UY31010A UY31010A1 (es) 2007-04-05 2008-04-07 Nuevo régimen de drospirenona/17b-estradiol, producto farmacéutico combinado y conjunto de elementos (kit) para su aplicacion

Country Status (15)

Country Link
US (1) US20090023693A1 (es)
EP (1) EP2150257A2 (es)
JP (1) JP2010523512A (es)
CN (1) CN101674837A (es)
AR (1) AR065971A1 (es)
AU (1) AU2008235006A1 (es)
BR (1) BRPI0810049A2 (es)
CA (1) CA2683093A1 (es)
CL (1) CL2008000999A1 (es)
IL (1) IL201302A0 (es)
MX (1) MX2009010763A (es)
PE (1) PE20090805A1 (es)
TW (1) TW200904452A (es)
UY (1) UY31010A1 (es)
WO (1) WO2008122439A2 (es)

Families Citing this family (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US8617597B2 (en) 2006-07-06 2013-12-31 Bayer Intellectual Property Gmbh Pharmaceutical composition containing a tetrahydrofolic acid
JP5951480B2 (ja) 2009-04-14 2016-07-13 ラボラトワール・アシュエールア−ファルマLaboratoire Hra−Pharma オンデマンド避妊方法
ES2533584T3 (es) * 2010-04-15 2015-04-13 Bayer Intellectual Property Gmbh Formas de dosificación oral sólidas de dosis baja para TSH
BR112012026115B1 (pt) * 2010-04-15 2019-12-24 Bayer Ip Gmbh forma de dosagem oral sólida, seu uso, e unidade de acondicionamento
CN108025014B (zh) * 2015-06-23 2021-10-22 莱昂实验室制药股份有限公司 用于过重女性患者的基于屈螺酮的避孕药

Family Cites Families (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
RS50262B2 (sr) * 1999-08-31 2018-10-31 Bayer Pharma AG Farmaceutska kombinacija etinilestradiola i drospirenona za primenu kao kontraceptivnog sredstva
US20020132801A1 (en) * 2001-01-11 2002-09-19 Schering Aktiengesellschaft Drospirenone for hormone replacement therapy
UY29527A1 (es) * 2005-05-13 2006-12-29 Schering Ag Composicinn farmaccutica que contienen gestrgenos y/o estrngenos y 5-metil - (6s) - tetrhidrofolato.

Also Published As

Publication number Publication date
JP2010523512A (ja) 2010-07-15
MX2009010763A (es) 2009-10-28
CA2683093A1 (en) 2008-10-16
US20090023693A1 (en) 2009-01-22
AU2008235006A1 (en) 2008-10-16
CN101674837A (zh) 2010-03-17
IL201302A0 (en) 2010-05-31
WO2008122439A3 (en) 2009-07-23
TW200904452A (en) 2009-02-01
AR065971A1 (es) 2009-07-15
PE20090805A1 (es) 2009-07-25
CL2008000999A1 (es) 2008-10-10
BRPI0810049A2 (pt) 2015-05-05
WO2008122439A2 (en) 2008-10-16
EP2150257A2 (en) 2010-02-10

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Legal Events

Date Code Title Description
109 Application deemed to be withdrawn

Effective date: 20170919