PE20090805A1 - COMBINACION DE DROSPIRENONA Y 17ß-ESTRADIOL COMO CONTRACEPTIVO ORAL - Google Patents
COMBINACION DE DROSPIRENONA Y 17ß-ESTRADIOL COMO CONTRACEPTIVO ORALInfo
- Publication number
- PE20090805A1 PE20090805A1 PE2008000621A PE2008000621A PE20090805A1 PE 20090805 A1 PE20090805 A1 PE 20090805A1 PE 2008000621 A PE2008000621 A PE 2008000621A PE 2008000621 A PE2008000621 A PE 2008000621A PE 20090805 A1 PE20090805 A1 PE 20090805A1
- Authority
- PE
- Peru
- Prior art keywords
- combination
- drospirenone
- estradiol
- oral contraceptive
- contraceptive
- Prior art date
Links
- VOXZDWNPVJITMN-ZBRFXRBCSA-N 17β-estradiol Chemical compound OC1=CC=C2[C@H]3CC[C@](C)([C@H](CC4)O)[C@@H]4[C@@H]3CCC2=C1 VOXZDWNPVJITMN-ZBRFXRBCSA-N 0.000 title abstract 4
- METQSPRSQINEEU-UHFFFAOYSA-N dihydrospirorenone Natural products CC12CCC(C3(CCC(=O)C=C3C3CC33)C)C3C1C1CC1C21CCC(=O)O1 METQSPRSQINEEU-UHFFFAOYSA-N 0.000 title abstract 3
- METQSPRSQINEEU-HXCATZOESA-N drospirenone Chemical compound C([C@]12[C@H]3C[C@H]3[C@H]3[C@H]4[C@@H]([C@]5(CCC(=O)C=C5[C@@H]5C[C@@H]54)C)CC[C@@]31C)CC(=O)O2 METQSPRSQINEEU-HXCATZOESA-N 0.000 title abstract 3
- 229960004845 drospirenone Drugs 0.000 title abstract 3
- 229940127234 oral contraceptive Drugs 0.000 title 1
- 239000003539 oral contraceptive agent Substances 0.000 title 1
- 229960005309 estradiol Drugs 0.000 abstract 1
- 229940011871 estrogen Drugs 0.000 abstract 1
- 239000000262 estrogen Substances 0.000 abstract 1
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
- A61K31/58—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin
- A61K31/585—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids containing heterocyclic rings, e.g. danazol, stanozolol, pancuronium or digitogenin containing lactone rings, e.g. oxandrolone, bufalin
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/12—Drugs for genital or sexual disorders; Contraceptives for climacteric disorders
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P15/00—Drugs for genital or sexual disorders; Contraceptives
- A61P15/18—Feminine contraceptives
Landscapes
- Health & Medical Sciences (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Veterinary Medicine (AREA)
- Animal Behavior & Ethology (AREA)
- Chemical & Material Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Pharmacology & Pharmacy (AREA)
- Medicinal Chemistry (AREA)
- Epidemiology (AREA)
- Bioinformatics & Cheminformatics (AREA)
- General Chemical & Material Sciences (AREA)
- Reproductive Health (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Organic Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Engineering & Computer Science (AREA)
- Endocrinology (AREA)
- Gynecology & Obstetrics (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Abstract
REFERIDA A UNA COMBINACION FARMACEUTICA QUE COMPRENDE ENTRE 2,0 MG Y 3,0 MG DE DROSPIRENONA Y ENTRE 1,0 MG Y 2,0 MG DE 17BETA-ESTRADIOL, DONDE ADEMAS DEL ESTROGENO Y LA DROSPIRENONA DICHA COMBINACION TAMBIEN PUEDE CONTENER TETRAHIDROFOLATO Y METAFOLINA. DICHA COMBINACION ES UTIL EN LA CONTRACEPCION ORAL FEMENINA
Applications Claiming Priority (3)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US91032607P | 2007-04-05 | 2007-04-05 | |
| US3528508P | 2008-03-10 | 2008-03-10 | |
| US4049408P | 2008-03-28 | 2008-03-28 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| PE20090805A1 true PE20090805A1 (es) | 2009-07-25 |
Family
ID=39745001
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| PE2008000621A PE20090805A1 (es) | 2007-04-05 | 2008-04-07 | COMBINACION DE DROSPIRENONA Y 17ß-ESTRADIOL COMO CONTRACEPTIVO ORAL |
Country Status (15)
| Country | Link |
|---|---|
| US (1) | US20090023693A1 (es) |
| EP (1) | EP2150257A2 (es) |
| JP (1) | JP2010523512A (es) |
| CN (1) | CN101674837A (es) |
| AR (1) | AR065971A1 (es) |
| AU (1) | AU2008235006A1 (es) |
| BR (1) | BRPI0810049A2 (es) |
| CA (1) | CA2683093A1 (es) |
| CL (1) | CL2008000999A1 (es) |
| IL (1) | IL201302A0 (es) |
| MX (1) | MX2009010763A (es) |
| PE (1) | PE20090805A1 (es) |
| TW (1) | TW200904452A (es) |
| UY (1) | UY31010A1 (es) |
| WO (1) | WO2008122439A2 (es) |
Families Citing this family (5)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US8617597B2 (en) | 2006-07-06 | 2013-12-31 | Bayer Intellectual Property Gmbh | Pharmaceutical composition containing a tetrahydrofolic acid |
| EP2419108B1 (en) | 2009-04-14 | 2016-08-17 | Laboratoire HRA Pharma | Method for on-demand contraception |
| US20130140210A1 (en) * | 2010-04-15 | 2013-06-06 | Bayer Intellectual Property Gmbh | Low-dosed solid oral dosage forms for hrt |
| BR112012026115B1 (pt) | 2010-04-15 | 2019-12-24 | Bayer Ip Gmbh | forma de dosagem oral sólida, seu uso, e unidade de acondicionamento |
| CN108025014B (zh) * | 2015-06-23 | 2021-10-22 | 莱昂实验室制药股份有限公司 | 用于过重女性患者的基于屈螺酮的避孕药 |
Family Cites Families (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| SI1214076T1 (en) * | 1999-08-31 | 2004-06-30 | Schering Aktiengesellschaft | Pharmaceutical combination of ethinylestradiol and drospirenone for use as a contraceptive |
| US20020132801A1 (en) * | 2001-01-11 | 2002-09-19 | Schering Aktiengesellschaft | Drospirenone for hormone replacement therapy |
| UY29527A1 (es) * | 2005-05-13 | 2006-12-29 | Schering Ag | Composicinn farmaccutica que contienen gestrgenos y/o estrngenos y 5-metil - (6s) - tetrhidrofolato. |
-
2008
- 2008-04-07 US US12/098,831 patent/US20090023693A1/en not_active Abandoned
- 2008-04-07 UY UY31010A patent/UY31010A1/es not_active Application Discontinuation
- 2008-04-07 MX MX2009010763A patent/MX2009010763A/es unknown
- 2008-04-07 BR BRPI0810049 patent/BRPI0810049A2/pt not_active IP Right Cessation
- 2008-04-07 CA CA002683093A patent/CA2683093A1/en not_active Abandoned
- 2008-04-07 AU AU2008235006A patent/AU2008235006A1/en not_active Abandoned
- 2008-04-07 CN CN200880014865A patent/CN101674837A/zh active Pending
- 2008-04-07 CL CL200800999A patent/CL2008000999A1/es unknown
- 2008-04-07 WO PCT/EP2008/002823 patent/WO2008122439A2/en not_active Ceased
- 2008-04-07 PE PE2008000621A patent/PE20090805A1/es not_active Application Discontinuation
- 2008-04-07 TW TW097112528A patent/TW200904452A/zh unknown
- 2008-04-07 EP EP08735133A patent/EP2150257A2/en not_active Withdrawn
- 2008-04-07 JP JP2010501448A patent/JP2010523512A/ja active Pending
- 2008-04-07 AR ARP080101436A patent/AR065971A1/es unknown
-
2009
- 2009-10-01 IL IL201302A patent/IL201302A0/en unknown
Also Published As
| Publication number | Publication date |
|---|---|
| EP2150257A2 (en) | 2010-02-10 |
| AR065971A1 (es) | 2009-07-15 |
| CL2008000999A1 (es) | 2008-10-10 |
| WO2008122439A2 (en) | 2008-10-16 |
| CN101674837A (zh) | 2010-03-17 |
| BRPI0810049A2 (pt) | 2015-05-05 |
| MX2009010763A (es) | 2009-10-28 |
| JP2010523512A (ja) | 2010-07-15 |
| IL201302A0 (en) | 2010-05-31 |
| US20090023693A1 (en) | 2009-01-22 |
| WO2008122439A3 (en) | 2009-07-23 |
| TW200904452A (en) | 2009-02-01 |
| AU2008235006A1 (en) | 2008-10-16 |
| CA2683093A1 (en) | 2008-10-16 |
| UY31010A1 (es) | 2008-11-28 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| FC | Refusal |